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公开(公告)号:US4058523A
公开(公告)日:1977-11-15
申请号:US723444
申请日:1976-09-15
申请人: Takashi Mori , Sakae Takaku , Nobuhiro Oi , Minoru Shindo , Takeaki Hirano , Shigeyuki Kataoka , Kouji Furuno
发明人: Takashi Mori , Sakae Takaku , Nobuhiro Oi , Minoru Shindo , Takeaki Hirano , Shigeyuki Kataoka , Kouji Furuno
IPC分类号: C07C233/12 , C07D295/12 , C07D295/10 , A61K31/165 , A61K31/535 , C07C103/78
CPC分类号: C07D295/12 , C07C233/12
摘要: Bis(benzamido)-benzene derivatives having various pharmaceutical activities such as activity for preventing and treating peptic ulcer, peripheral vasodilating action, hypotensive activity and analgesic activity and represented by the formula ##STR1## wherein X, Y, Z, R.sub.1, R.sub.2 and R.sub.3 are as defined hereinafter and a process for preparing the same are disclosed.
摘要翻译: 具有各种药物活性的双(苯甲酰氨基) - 苯衍生物,例如用于预防和治疗消化性溃疡的活性,外周血管扩张作用,降血压活性和止痛活性,并由式
表示,其中X,Y,Z,R 1,R 2和R 3 如下所述,并公开了其制备方法。 -
公开(公告)号:US4092431A
公开(公告)日:1978-05-30
申请号:US791889
申请日:1977-04-28
申请人: Takashi Mori , Sakae Takaku , Nobuhiro Oi , Minoru Shindo , Takeaki Hirano , Shigeyuki Kataoka , Kouji Furuno
发明人: Takashi Mori , Sakae Takaku , Nobuhiro Oi , Minoru Shindo , Takeaki Hirano , Shigeyuki Kataoka , Kouji Furuno
IPC分类号: A61K31/165 , A61P1/04
CPC分类号: A61K31/165 , Y10S514/925 , Y10S514/927
摘要: A pharmaceutical composition for prevention and treatment of gastritis and peptic ulcer of mammals including human beings which contains a bis(benzamido)benzene derivative represented by the formula ##STR1## wherein X and Y are as defined hereinbelow, or an acid addition salt thereof, as an active ingredient, and a method of the use thereof are disclosed.
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公开(公告)号:US4038416A
公开(公告)日:1977-07-26
申请号:US612500
申请日:1975-09-11
申请人: Takashi Mori , Sakae Takaku , Nobuhiro Oi , Minoru Shindo , Takeaki Hirano , Shigeyuki Kataoka , Kouji Furuno
发明人: Takashi Mori , Sakae Takaku , Nobuhiro Oi , Minoru Shindo , Takeaki Hirano , Shigeyuki Kataoka , Kouji Furuno
IPC分类号: A61K31/165 , A61P1/04
CPC分类号: A61K31/165 , Y10S514/925 , Y10S514/927
摘要: A pharmaceutical composition for prevention and treatment of gastritis and peptic ulcer of mammals including human beings which contains a bis(benzamido)-benzene derivative represented by the formula ##STR1## wherein X and Y are as defined hereinbelow or an acid addition salt thereof as an active ingredient, and a method of the use thereof are disclosed.
摘要翻译: 一种用于预防和治疗包括人的哺乳动物的胃炎和消化性溃疡的药物组合物,其包含由下式表示的式(I)所示的双(苯甲酰氨基)苯衍生物或其酸加成盐, 公开了一种活性成分及其使用方法。
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