Glycopeptide antibiotic derivative
    2.
    发明授权
    Glycopeptide antibiotic derivative 有权
    糖肽抗生素衍生物

    公开(公告)号:US08933012B2

    公开(公告)日:2015-01-13

    申请号:US12224443

    申请日:2007-05-25

    CPC分类号: C07K9/008 A61K38/00 A61K38/04

    摘要: The present invention provides a novel glycopeptide antibiotic derivative.These derivatives are represented by the formula (I) or a pharmaceutically acceptable salt or solvate thereof, wherein RA is —X1—Ar1—X2—Y—X3—Ar2 wherein X1, X2 and X3 are single bond; heteroatom-containing group selected from the group consisting of —N═, ═N—, —NR1— (R1 is hydrogen or lower alkyl), —O—, —S—, —SO— and —SO2—, or a linkage thereof; or alkylene or alkenylene optionally substituted and optionally interrupted by one or more of said heteroatom-containing group; Y is —NR2CO—, —CONR2— (R2 is hydrogen or lower alkyl), or a group of the formula (II) wherein R3 is alkylene; Ar1 and Ar2 are a carbocycle or a heterocycle which is optionally substituted and may have an unsaturated bond; RB is —NHNRXRY or —NRZORW wherein RX is hydrogen or lower alkyl; RY is hydrogen, optionally substituted lower alkyl, C(═NH)NH2, CSNH2, COCONH2, CN, optionally substituted heterocyclic group, and optionally substituted carbamoyl; RZ is hydrogen or lower alkyl; RW is hydrogen, optionally substituted lower alkyl, optionally substituted lower alkenyl, optionally substituted heterocyclic group, optionally substituted heterocyclic carbonyl or optionally substituted carbamoyl; RC is hydrogen or optionally substituted alkyl, wherein said alkyl may be interrupted by a heteroatom-containing group selected from N═, ═N—, —NR1— (R1 is hydrogen or lower alkyl), —O—, —S—, —SO— and —SO2—; and R is optionally substituted alkyl.

    摘要翻译: 本发明提供了一种新型糖肽抗生素衍生物。 这些衍生物由式(I)表示或其药学上可接受的盐或溶剂化物,其中RA为-X1-Ar1-X2-Y-X3-Ar2,其中X1,X2和X3为单键; 选自-N =,N-,-NR1-(R 1为氢或低级烷基), - O - , - S - , - SO-和-SO 2 - 的杂原子的基团,或其连接基 ; 或任选被取代并任选被一个或多个所述含杂原子基团中断的亚烷基或亚烯基; Y是-NR 2 CO-,-CONR 2 - (R 2是氢或低级烷基)或式(II)的基团,其中R 3是亚烷基; Ar1和Ar2是任选被取代并可具有不饱和键的碳环或杂环; RB是-NHNRXRY或-NRZORW,其中RX是氢或低级烷基; RY是氢,任选取代的低级烷基,C(= NH)NH 2,CSNH 2,COCONH 2,CN,任选取代的杂环基和任选取代的氨基甲酰基; RZ是氢或低级烷基; RW是氢,任选取代的低级烷基,任选取代的低级烯基,任选取代的杂环基,任选取代的杂环羰基或任选取代的氨基甲酰基; RC是氢或任选取代的烷基,其中所述烷基可以被选自N =,N-,-NR1-(R 1是氢或低级烷基),-O - , - S - , - SO-和-SO 2 - ; R是任选取代的烷基。

    Information processing apparatus and display control method
    3.
    发明授权
    Information processing apparatus and display control method 有权
    信息处理装置及显示控制方法

    公开(公告)号:US08294725B2

    公开(公告)日:2012-10-23

    申请号:US12777119

    申请日:2010-05-10

    IPC分类号: G09G5/36

    摘要: According to one embodiment, an information processing apparatus comprises video memories each corresponding to each of the display devices, a determination module configured to determine whether an access that satisfies conditions preset with respect to display of the display devices exists in at least one of the video memories, and a changing module configured to change, when the determination module determines that the access that satisfies conditions preset with respect to display of the display devices does not exist in at least one of the video memories, an operation state of a display device corresponding to the at least one of the video memories determined that an access does not exist, from a first operation state to a second operation state having a power consumption lower than a power consumption of the first operation state.

    摘要翻译: 根据一个实施例,信息处理设备包括每个对应于每个显示设备的视频存储器,确定模块被配置为确定满足关于显示设备的显示的预设条件的访问是否存在于视频的至少一个中 存储器和改变模块,其被配置为当所述确定模块确定满足关于所述显示设备的显示预设的条件的访问不存在于所述视频存储器的至少一个中时,改变对应于所述显示设备的操作状态 将确定存在不存在的视频存储器中的至少一个从第一操作状态转换为具有低于第一操作状态的功耗的功耗的第二操作状态。

    Information processing apparatus and display control method
    4.
    再颁专利
    Information processing apparatus and display control method 失效
    信息处理装置及显示控制方法

    公开(公告)号:USRE41104E1

    公开(公告)日:2010-02-09

    申请号:US12330245

    申请日:2008-12-08

    申请人: Tsutomu Iwaki

    发明人: Tsutomu Iwaki

    IPC分类号: H04N9/74

    摘要: When the fact that the display mode of motion picture data is a full screen mode is detected, the display control mode for sending a video signal generated by a graphics controller to an LCD is switched from a normal mode for sending the video signal to the LCD without interposition of a high quality video engine to a high quality mode for sending the video signal to the LCD with interposition of the high quality video engine. The high quality video engine enlarges the screen size of the video signal in either linear scaling mode or nonlinear scaling mode designated by a user. Scaling is validated only in the case were motion picture data are displayed in the full screen mode.

    摘要翻译: 当检测到运动图像数据的显示模式是全屏模式的事实时,将由图形控制器产生的视频信号发送到LCD的显示控制模式从用于将视频信号发送到LCD的正常模式切换 而不需要将高质量视频引擎插入高品质模式,用于通过插入高质量视频引擎将视频信号发送到LCD。 高质量视频引擎以用户指定的线性缩放模式或非线性缩放模式放大视频信号的屏幕尺寸。 仅在运动图像数据以全屏模式显示的情况下,缩放才被验证。

    Information processing apparatus and video signal output control method
    5.
    发明授权
    Information processing apparatus and video signal output control method 有权
    信息处理装置和视频信号输出控制方法

    公开(公告)号:US07649735B2

    公开(公告)日:2010-01-19

    申请号:US11485365

    申请日:2006-07-13

    申请人: Tsutomu Iwaki

    发明人: Tsutomu Iwaki

    IPC分类号: G06F1/16

    CPC分类号: G06F1/1632

    摘要: A video signal output control method in an information processing apparatus which being to be locked to an external unit by a lock mechanism, the video signal output control method includes detecting the state of the lock mechanism, and stopping the output of the video signal to the external unit, when the lock mechanism is in the unlocked state.

    摘要翻译: 一种视频信号输出控制方法,在通过锁定机构锁定到外部单元的信息处理装置中,视频信号输出控制方法包括检测锁定机构的状态,并停止将视频信号输出到 外部单元,当锁定机构处于未锁定状态时。

    Glycopeptide Antibiotic Derivative
    6.
    发明申请
    Glycopeptide Antibiotic Derivative 有权
    糖肽抗生素衍生物

    公开(公告)号:US20090286717A1

    公开(公告)日:2009-11-19

    申请号:US12224443

    申请日:2007-05-25

    IPC分类号: A61K38/00 C07K9/00 A61P43/00

    CPC分类号: C07K9/008 A61K38/00 A61K38/04

    摘要: The present invention provides a novel glycopeptide antibiotic derivative.These derivatives are represented by the formula (I) or a pharmaceutically acceptable salt or solvate thereof, wherein RA is —X1—Ar1—X2—Y—X3—Ar2 wherein X1, X2 and X3 are single bond; heteroatom-containing group selected from the group consisting of —N═, ═N—, —NR1— (R1 is hydrogen or lower alkyl), —O—, —S—, —SO— and —SO2—, or a linkage thereof; or alkylene or alkenylene optionally substituted and optionally interrupted by one or more of said heteroatom-containing group; Y is —NR2CO—, —CONR2— (R2 is hydrogen or lower alkyl), or a group of the formula (II) wherein R3 is alkylene; Ar1 and Ar2 are a carbocycle or a heterocycle which is optionally substituted and may have an unsaturated bond; RB is —NHNRXRY or —NRZORW wherein RX is hydrogen or lower alkyl; RY is hydrogen, optionally substituted lower alkyl, C(═NH)NH2, CSNH2, COCONH2, CN, optionally substituted heterocyclic group, and optionally substituted carbamoyl; RZ is hydrogen or lower alkyl; RW is hydrogen, optionally substituted lower alkyl, optionally substituted lower alkenyl, optionally substituted heterocyclic group, optionally substituted heterocyclic carbonyl or optionally substituted carbamoyl; RC is hydrogen or optionally substituted alkyl, wherein said alkyl may be interrupted by a heteroatom-containing group selected from N═, ═N—, —NR1— (R1 is hydrogen or lower alkyl), —O—, —S—, —SO— and —SO2—; and R is optionally substituted alkyl.

    摘要翻译: 本发明提供了一种新型糖肽抗生素衍生物。 这些衍生物由式(I)表示或其药学上可接受的盐或溶剂化物,其中RA为-X1-Ar1-X2-Y-X3-Ar2,其中X1,X2和X3为单键; 选自-N-,-N-,-NR1-(R 1为氢或低级烷基), - , - - , - S - , - SO - 和-SO 2 - 或其连接基团 ; 或任选被取代并任选被一个或多个所述含杂原子基团中断的亚烷基或亚烯基; Y是-NR 2 CO-,-CONR 2 - (R 2是氢或低级烷基)或式(II)的基团,其中R 3是亚烷基; Ar1和Ar2是任选被取代并可具有不饱和键的碳环或杂环; RB是-NHNRXRY或-NRZORW,其中RX是氢或低级烷基; RY是氢,任选取代的低级烷基,C(-NH)NH 2,CSNH 2,COCONH 2,CN,任选取代的杂环基和任选取代的氨基甲酰基; RZ是氢或低级烷基; RW是氢,任选取代的低级烷基,任选取代的低级烯基,任选取代的杂环基,任选取代的杂环羰基或任选取代的氨基甲酰基; RC是氢或任选取代的烷基,其中所述烷基可以被选自N-,-N-,-NR1-(R 1是氢或低级烷基),-O - , - S - , - SO-和-SO 2 - ; R是任选取代的烷基。

    Information processing apparatus and display control method
    7.
    发明申请
    Information processing apparatus and display control method 审中-公开
    信息处理装置及显示控制方法

    公开(公告)号:US20070242159A1

    公开(公告)日:2007-10-18

    申请号:US11812397

    申请日:2007-06-19

    申请人: Tsutomu Iwaki

    发明人: Tsutomu Iwaki

    IPC分类号: H04N5/46 H04N9/74

    摘要: An information processing apparatus including: a display that is capable of displaying moving image data in a full screen mode; a first signal processing section that generates a signal for forming the moving image data to be displayed on the display; a second signal processing section that executes image quality processing for the signal generated by the first signal processing section; a determination section that determines whether or not a display mode to display the moving image data is the full screen mode based on a relationship between a screen size of the moving image data and a screen size of the display; and a control section that enables the signal subjected to the image quality processing by the second signal processing section to be output to the display when the determination section determines that the display mode to display the moving image data is the full screen mode.

    摘要翻译: 一种信息处理设备,包括:能够以全屏模式显示运动图像数据的显示器; 第一信号处理部,其生成用于形成要在显示器上显示的运动图像数据的信号; 第二信号处理部,对由所述第一信号处理部生成的信号进行图像质量处理; 确定部分,其基于所述运动图像数据的屏幕尺寸和所述显示器的屏幕尺寸之间的关系,确定显示所述运动图像数据的显示模式是否为全屏模式; 以及控制部,其使得当所述判定部判定为显示所述运动图像数据的显示模式为全屏模式时,能够将由所述第二信号处理部进行了图像质量处理的信号输出到所述显示。

    Battery electrode producing method, and battery electrode
    8.
    发明申请
    Battery electrode producing method, and battery electrode 有权
    电池电极的制造方法和电池电极

    公开(公告)号:US20070207388A1

    公开(公告)日:2007-09-06

    申请号:US11712473

    申请日:2007-03-01

    IPC分类号: H01M4/74 H01M4/32 H01M4/04

    摘要: A method of producing an electrode includes the steps of filling an active material in an electrode substrate made of woven or non-woven fabric having its fiber surface coated with metal, and pressing the electrode substrate to obtain an electrode, wherein the pressing is performed using the electrode substrate having a thickness of less than 2.0 t when the thickness of the electrode after the pressing is t. This ensues that the electrode substrate has a thickness allowing the active material of a sufficient amount to be filled therein, and a battery electrode in which the filled active material is unlikely to peel off from the electrode substrate can be produced. Accordingly, a battery electrode having a desired thickness and desired capacity and that can suppress degradation in battery performance due to repeated charge and discharge, and its producing method are provided.

    摘要翻译: 电极的制造方法包括以下步骤:将活性物质填充在由金属纤维表面涂覆的织造或无纺布制成的电极基板中,并按压电极基板以获得电极,其中使用 当压制后的电极的厚度为t时,电极基板的厚度小于2.0t。 因此,可以制造电极基板的厚度,使得能够填充足够量的活性物质,并且可以制造填充的活性物质不易从电极基板剥离的电池电极。 因此,提供了具有期望的厚度和期望容量并且可以抑制由于反复充放电引起的电池性能劣化的电池电极及其制造方法。

    Hydrogen storage alloy electrode
    9.
    发明授权
    Hydrogen storage alloy electrode 失效
    氢存储合金电极

    公开(公告)号:US5149383A

    公开(公告)日:1992-09-22

    申请号:US677572

    申请日:1991-03-29

    IPC分类号: H01M4/38

    CPC分类号: H01M4/383 Y10S420/90

    摘要: The present invention provides a hydrogen storage alloy electrode made of a pentanary or higher multi-component hydrogen storage alloy or a hydride thereof where the alloy comprises at least Zr, Mn, Cr, Ni, and M where M is one or more elements selected from V an Mo, and a major component of the alloy phase is C.sub.15 (MgCu.sub.2) type Laves phase. This hydrogen storage alloy electrode may be enhanced in its performance by subjecting the alloy after the production thereof to a homogenizing heat-treatment at a temperature of 900.degree. to 1300.degree. C. in vacuum or in an inert gaseous atmosphere.