HALOSUBSTITUTED ARYLOXYALKYLIMIDAZOLINES FOR USE AS PESTICIDES

    公开(公告)号:US20100280088A1

    公开(公告)日:2010-11-04

    申请号:US12677825

    申请日:2008-09-09

    CPC分类号: C07D233/16 A01N43/50

    摘要: The present invention relates to novel imidazoline derivatives and their use as insecticidal, acaricidal, molluscicidal and nematocidal agents. The invention also extends to insecticidal, acaricidal, molluscicidal and nematicidal compositions comprising such imidazoline derivatives, and to methods of using such derivatives and/or compositions to combat and control insect, acarine, mollusc and nematode pests. A compound of formula (I) and salts and N-oxides thereof, wherein: R1 is C1-10 alkyl; R2 is chloro, bromo or iodo; R3 is C2-5 alkyl, C1-5 haloalkyl, C1-6 hydroxyalkyl, C1-5alkoxy-(C1-3)-alkyl, di-(C1-5 alkoxy)-(C1-3)-alkyl, C1-5alkylthio-(C1-3)-alkyl; C1-5 alkylsulfinyl-(C1-3)alkyl; C2-5 alkenyl, C1-5 haloalkenyl, C2-5 alkinyl, C3-6 cycloalkyl, C3-6 cycloalkenyl, hydroxy, C1-5 alkoxy, C1-5haloalkoxy, C1-5alkylthio, C1-5 haloalkylthio, formyl, cyano, bromo, or iodo; Z is hydrogen, hydroxy, nitro cyano, rhodano, formyl, G-, G-S—, G-S—S—, G-A-, R7R8N—, R7R8N—S—, R7R8N-A-, G-O-A-, G-S-A-, (R10O)(R11O)P(X)—, (R10O)(R11S)P(X)—, (R10O)(R11)P(X)—, (R10S)(R11S)P(X)—, (R10O)(R14R15N)P(X)—, (R11)(R14R15N)P(X)—, (R14R15N)(R16R17N)P(X)—, G-N═CH—, G-O—N═CH—, N≡C—N═CH—, or Z is a group of formula (II), wherein B is S—, S—S—, S(O)—, C(O)—, or (CH2)n—; n is an integer from 1 to 6; and R1, R2, and R3 are as defined above; and G is optionally substituted C1-10alkyl, optionally substituted C2-10 alkenyl, optionally substituted C2-10 alkynyl, optionally substituted C3-7 cycloalkyl, optionally substituted C3-7 cycloalkenyl, optionally substituted aryl, optionally substituted heteroaryl or optionally substituted heterocyclyl; A is S(O), SO2, C(O) or C(S).

    Phenoxymethyl imidazoline derivatives and their use as pesticides
    4.
    发明授权
    Phenoxymethyl imidazoline derivatives and their use as pesticides 失效
    苯氧基甲基咪唑啉衍生物及其作为农药的用途

    公开(公告)号:US08110593B2

    公开(公告)日:2012-02-07

    申请号:US12526977

    申请日:2008-01-18

    摘要: The present invention relates to imidazoline derivatives and their use as insecticidal, acaricidal, molluscicidal and nematocidal agents. The invention also extends to insecticidal, acaricidal, molluscicidal and nematicidal compositions comprising such imidazoline derivatives, and to methods of using such derivatives and/or compositions to combat and control insect, acarine, mollusc and nematode pests. In particular the present invention relates to imidazolines with alkyl, cycloalkyl, alkenyl, cycloalkenyl, alkynyl, aryl, heteroaryl or heterocyclyl substituents.

    摘要翻译: 本发明涉及咪唑啉衍生物及其作为杀虫,杀螨,杀软体动物和杀线虫剂的用途。 本发明还延伸到包含这种咪唑啉衍生物的杀虫,杀螨,杀软体动物和杀线虫组合物,以及使用这些衍生物和/或组合物来对抗和控制昆虫,螨虫,软体动物和线虫的害虫的方法。 特别地,本发明涉及具有烷基,环烷基,烯基,环烯基,炔基,芳基,杂芳基或杂环基取代基的咪唑啉。

    NITROSUBSTITUTED ARYLOXYALKYLIMIDAZOLINES FOR USE AS PESTICIDES
    5.
    发明申请
    NITROSUBSTITUTED ARYLOXYALKYLIMIDAZOLINES FOR USE AS PESTICIDES 审中-公开
    用作杀虫剂的硝基苯甲酰胺基咪唑啉

    公开(公告)号:US20100267795A1

    公开(公告)日:2010-10-21

    申请号:US12741741

    申请日:2008-10-24

    摘要: The present invention relates to imidazoline derivatives and their use as insecticidal and acaricidal agents. The invention also extends to insecticidal and acaricidal compositions comprising such imidazoline derivatives, and to methods of using such derivatives and/or compositions to combat and control insect and acarine pests. In particular the present invention relates to phenoxy-imidazoline derivatives wherein the phenoxy moiety is substituted with a nitro group. A method of combating and/or controlling an insect or acarid pest, which comprises applying to said pest, or to the locus of said pest, or to a plant susceptible to attack by said pest, a compound of formula (I): or salt or N-oxide thereof.

    摘要翻译: 本发明涉及咪唑啉衍生物及其作为杀虫剂和杀螨剂的用途。 本发明还延伸到包含这种咪唑啉衍生物的杀虫和杀螨组合物,以及使用这些衍生物和/或组合物来对抗和控制昆虫和螨类害虫的方法。 特别地,本发明涉及苯氧基 - 咪唑啉衍生物,其中苯氧基部分被硝基取代。 一种防治昆虫或螨类害虫的方法,其包括向所述有害生物或所述有害生物所在地或向所述有害生物易受攻击的植物施用式(I)化合物或盐 或N-氧化物。

    CHEMICAL COMPOUNDS
    6.
    发明申请
    CHEMICAL COMPOUNDS 失效
    化学化合物

    公开(公告)号:US20100120881A1

    公开(公告)日:2010-05-13

    申请号:US12526977

    申请日:2008-01-18

    摘要: The present invention relates to imidazoline derivatives and their use as insecticidal, acaricidal, molluscicidal and nematocidal agents. The invention also extends to insecticidal, acaricidal, molluscicidal and nematicidal compositions comprising such imidazoline derivatives, and to methods of using such derivatives and/or compositions to combat and control insect, acarine, mollusc and nematode pests. In particular the present invention relates to imidazolines with alkyl, cycloalkyl, alkenyl, cycloalkenyl, alkynyl, aryl, heteroaryl or heterocyclyl substituents.

    摘要翻译: 本发明涉及咪唑啉衍生物及其作为杀虫,杀螨,杀软体动物和杀线虫剂的用途。 本发明还延伸到包含这种咪唑啉衍生物的杀虫,杀螨,杀软体动物和杀线虫组合物,以及使用这些衍生物和/或组合物来对抗和控制昆虫,螨虫,软体动物和线虫的害虫的方法。 特别地,本发明涉及具有烷基,环烷基,烯基,环烯基,炔基,芳基,杂芳基或杂环基取代基的咪唑啉。

    Chemical compounds
    7.
    发明授权
    Chemical compounds 失效
    化合物

    公开(公告)号:US08309739B2

    公开(公告)日:2012-11-13

    申请号:US13105596

    申请日:2011-05-11

    IPC分类号: C07D277/18

    摘要: The use of a compound of formula I wherein X is (i), (ii) or (iii) Y is O, S(O)m, NR3, CR5R6, CR5R6—CR7R8, O—CR7R8, S(O)m—CR7R8, NR3—CR7R8, CR5R6—O, CR5R6—S(O)m, CR5R6—NR3, SO2—NR3, NR3—SO2, NR3—O or O—NR3; m is 0, 1, or 2; the ring (T) is a 5- or 6-membered aromatic or heteroaromatic ring; R1 to R10 are specified organic groups and n and is 0, 1, 2, 3 or 4; or salts or N-oxides thereof or compositions containing them in controlling insects, acarines, nematodes or molluscs. Novel compounds are also provided.

    摘要翻译: 其中X是(i),(ii)或(iii)Y的式I化合物是O,S(O)m,NR 3,CR 5 R 6,CR 5 R 6 -CR 7 R 8,O-CR 7 R 8,S(O) CR7R8,NR3-CR7R8,CR5R6-O,CR5R6-S(O)m,CR5R6-NR3,SO2-NR3,NR3-SO2,NR3-O或O-NR3; m为0,1或2; 环(T)是5或6元芳族或杂芳族环; R1至R10为指定的有机基团,n为0,1,2,3或4; 或其盐或N-氧化物或含有它们的组合物来控制昆虫,螨类,线虫或软体动物。 还提供了新的化合物。

    Halosubstituted aryloxyalkylimidazolines for use as pesticides
    8.
    发明授权
    Halosubstituted aryloxyalkylimidazolines for use as pesticides 失效
    用作农药的卤代芳氧基烷基咪唑啉

    公开(公告)号:US08455663B2

    公开(公告)日:2013-06-04

    申请号:US12677825

    申请日:2008-09-09

    IPC分类号: C07D233/22 C07C255/13

    CPC分类号: C07D233/16 A01N43/50

    摘要: The present invention relates to novel imidazoline derivatives and their use as insecticidal, acaricidal, molluscicidal and nematocidal agents. The invention also extends to insecticidal, acaricidal, molluscicidal and nematicidal compositions comprising such imidazoline derivatives, and to methods of using such derivatives and/or compositions to combat and control insect, acarine, mollusc and nematode pests. A compound of formula (I) and salts and N-oxides thereof, wherein: R1 is C1-10 alkyl; R2 is chloro, bromo or iodo; R3 is C2-5 alkyl, C1-5 haloalkyl, C1-6 hydroxyalkyl, C1-5alkoxy-(C1-3)-alkyl, di-(C1-5 alkoxy)-(C1-3)-alkyl, C1-5alkylthio-(C1-3)-alkyl; C1-5 alkylsulfinyl-(C1-3)alkyl; C2-5 alkenyl, C1-5 haloalkenyl, C2-5 alkinyl, C3-6 cycloalkyl, C3-6 cycloalkenyl, hydroxy, C1-5 alkoxy, C1-5haloalkoxy, C1-5alkylthio, C1-5 haloalkylthio, formyl, cyano, bromo, or iodo; Z is hydrogen, hydroxy, nitro cyano, rhodano, formyl, G-, G-S—, G-S—S—, G-A-, R7R8N—, R7R8N—S—, R7R8N-A-, G-O-A-, G-S-A-, (R10O)(R11O)P(X)—, (R10O)(R11S)P(X)—, (R10O)(R11)P(X)—, (R10S)(R11S)P(X)—, (R10O)(R14R15N)P(X)—, (R11)(R14R15N)P(X)—, (R14R15N)(R16R17N)P(X)—, G-N═CH—, G-O—N═CH—, N≡C—N═CH—, or Z is a group of formula (II), wherein B is S—, S—S—, S(O)—, C(O)—, or (CH2)n—; n is an integer from 1 to 6; and R1, R2, and R3 are as defined above; and G is optionally substituted C1-10alkyl, optionally substituted C2-10 alkenyl, optionally substituted C2-10 alkynyl, optionally substituted C3-7 cycloalkyl, optionally substituted C3-7 cycloalkenyl, optionally substituted aryl, optionally substituted heteroaryl or optionally substituted heterocyclyl; A is S(O), SO2, C(O) or C(S).

    摘要翻译: 本发明涉及新的咪唑啉衍生物及其作为杀虫,杀螨,杀软体动物和杀线虫剂的用途。 本发明还延伸到包含这种咪唑啉衍生物的杀虫,杀螨,杀软体动物和杀线虫组合物,以及使用这些衍生物和/或组合物来对抗和控制昆虫,螨虫,软体动物和线虫的害虫的方法。 式(I)化合物及其盐和N-氧化物,其中:R1为C1-10烷基; R2是氯,溴或碘; R3是C2-5烷基,C1-5卤代烷基,C1-6羟基烷基,C1-5烷氧基 - (C1-3) - 烷基,二 - (C1-5烷氧基) - (C1-3) - 烷基,C1-5烷硫基 - (C 1-3) - 烷基; C 1-5烷基亚磺酰基 - (C 1-3)烷基; C2-5烯基,C1-5卤代烯基,C2-5炔基,C3-6环烷基,C3-6环烯基,羟基,C1-5烷氧基,C1-5卤代烷氧基,C1-5烷硫基,C1-5卤代烷硫基,甲酰基,氰基,溴 ,或碘; Z是氢,羟基,硝基氰基,罗丹明,甲酰基,G-,GS-,GSS-,GA-,R7R8N-,R7R8N-S-,R7R8N-A-,GOA-,GSA-,(R10O) P(X) - ,(R10O)(R11S)P(X) - ,(R10O)(R11)P(X) - ,(R10S)(R11S)P(X) - ,(R10O)(R14R15N) X) - ,(R11)(R14R15N)P(X) - ,(R14R15N)(R16R17N)P(X) - ,GN = CH-,GON = CH-,N = CN = CH-,或Z为基团 其中B为S-,SS-,S(O) - ,C(O) - 或(CH 2)n - )的式(II) n是1至6的整数; 并且R 1,R 2和R 3如上所定义; 任选取代的C 2-10炔基,任选取代的C 3-7环烷基,任选取代的C 3-7环烯基,任选取代的芳基,任选取代的杂芳基或任选取代的杂环基; A是S(O),SO 2,C(O)或C(S)。

    PHENOXYMETHYL IMIDAZOLINE DERIVATIVES AND THEIR USE AS PESTICIDES
    9.
    发明申请
    PHENOXYMETHYL IMIDAZOLINE DERIVATIVES AND THEIR USE AS PESTICIDES 审中-公开
    苯甲基咪唑衍生物及其作为杀虫剂的用途

    公开(公告)号:US20100120882A1

    公开(公告)日:2010-05-13

    申请号:US12527213

    申请日:2008-01-28

    IPC分类号: A01N43/50 C07D233/22

    CPC分类号: C07D233/22 C07C255/16

    摘要: The present invention relates to imidazoline derivatives and their use as insecticidal, acaricidal, molluscicidal and nematocidal agents. The invention also extends to insecticidal, acaricidal, molluscicidal and nematicidal compositions comprising such imidazoline derivatives, and to methods of using such derivatives and/or compositions to combat and control insect, acarine, mollusc and nematode pests. In particular the present invention relates to imidazolines with alkyl and fluoro substituents.

    摘要翻译: 本发明涉及咪唑啉衍生物及其作为杀虫,杀螨,杀软体动物和杀线虫剂的用途。 本发明还延伸到包含这种咪唑啉衍生物的杀虫,杀螨,杀软体动物和杀线虫组合物,以及使用这些衍生物和/或组合物来对抗和控制昆虫,螨虫,软体动物和线虫的害虫的方法。 特别地,本发明涉及具有烷基和氟取代基的咪唑啉。