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    Pyridazine compounds for controlling invertebrate pests
    3.
    发明授权
    Pyridazine compounds for controlling invertebrate pests 有权
    用于控制无脊椎害虫的哒嗪化合物

    公开(公告)号：US08710056B2

    公开(公告)日：2014-04-29

    申请号：US13382229

    申请日：2010-07-01

    申请人： Ronan Le Vezouet ,  Sebastian Soergel ,  Christian Defieber ,  Steffen Gross ,  Karsten Koerber ,  Deborah L. Culbertson ,  Douglas D. Anspaugh

    发明人： Ronan Le Vezouet ,  Sebastian Soergel ,  Christian Defieber ,  Steffen Gross ,  Karsten Koerber ,  Deborah L. Culbertson ,  Douglas D. Anspaugh

    IPC分类号： A01N43/58 ,  A61K31/50 ,  A01N43/80 ,  A01N25/00 ,  A01N43/08 ,  A01N43/10 ,  C07D207/20 ,  C07D327/02 ,  C07D275/02 ,  C07D277/18 ,  C07D417/12 ,  C07D261/18 ,  C07D261/02 ,  A61K31/42

    CPC分类号： C07D417/12 ,  A01N43/80 ,  A01N53/00 ,  C07D413/12

    摘要： The present invention relates to pyridazine compounds of formulae I or II and the salts and N-oxides thereof, wherein A is a substituted or unsubstituted isoxazole or isothiazole radical; V is C(Rv) or N; W is C(Rw) or N; with the proviso that either V or W is N; Rt, Ru, Rv, Rw are H, halogen, C1-C4-alkyl and the like; X1 is S, O or NR1a, wherein R1a is selected H, C1-C10-alkyl and the like; X2 is OR2a, NR2bR2c, S(O)mR2d, wherein m is 0, 1 or 2, R2a is C1-C4-alkyl, C1-C4-haloalkyl and the like, R2b, R2c are H, C1-C4-alkyl, C1-C4-haloalkyl and the like, or R2b and R2c together with the nitrogen atom to which they are bound form a heterocycle, and R2d is C1-C4-alkyl, C1-C4-haloalkyl, C3-C6-cycloalkyl and the like; and R1 is H, CN, C1-C10-alkyl and the like. The present invention further relates to a method for controlling invertebrate pests, to a method for protecting plant propagation material and/or the plants which grow therefrom, to plant propagation material, comprising at least one compound according to the present invention, to a method for treating or protecting an animal from infestation or infection by parasites and to an agricultural composition containing at least one compound according to the present invention.

    摘要翻译： 本发明涉及式I或II的哒嗪化合物及其盐和N-氧化物，其中A是取代或未取代的异恶唑或异噻唑基; V是C（Rv）或N; W是C（Rw）或N; 条件是V或W为N; R 1，R u，R v，R w为H，卤素，C 1 -C 4 - 烷基等; X1是S，O或NR1a，其中R1a选自H，C1-C10-烷基等; X2是OR2a，NR2bR2c，S（O）mR2d，其中m是0,1或2，R2a是C1-C4-烷基，C1-C4-卤代烷基等，R2b，R2c是H，C1-C4-烷基， C1-C4卤代烷基等，或R2b和R2c与它们所结合的氮原子一起形成杂环，R2d是C1-C4-烷基，C1-C4卤代烷基，C3-C6-环烷基等 ; R1为H，CN，C1-C10-烷基等。 本发明还涉及一种控制无脊椎害虫的方法，一种用于保护植物繁殖材料和/或从其生长的植物的方法，包括至少一种根据本发明的化合物的植物繁殖材料的方法， 治疗或保护动物免受寄生虫侵袭或感染，以及含有至少一种本发明化合物的农药组合物。

    Whitening Agent And Skin External Preparation
    6.
    发明申请
    Whitening Agent And Skin External Preparation 审中-公开
    美白剂和皮肤外用剂

    公开(公告)号：US20100324096A1

    公开(公告)日：2010-12-23

    申请号：US12866472

    申请日：2009-02-06

    申请人： Naoto Hanyu ,  Tomoko Saito ,  Takako Shibata ,  Kiyoshi Sato ,  Kimihiro Ogino

    发明人： Naoto Hanyu ,  Tomoko Saito ,  Takako Shibata ,  Kiyoshi Sato ,  Kimihiro Ogino

    IPC分类号： A61K8/49 ,  C07D277/18 ,  C07D417/12 ,  A61Q19/02

    CPC分类号： A61K31/4439 ,  A61K8/4946 ,  A61K31/506 ,  A61Q19/02

    摘要： The present invention provides a compound having an excellent inhibitory action on melanin production and being useful as a whitening agent, and a skin external preparation containing the compound. The whitening agent of the present invention comprises, as an active ingredient, a heterocyclic compound represented by formula (1) or a pharmacologically acceptable salt thereof: wherein A is C1-6 alkyl, C5-6 cycloalkyl, benzyl, benzylcarbonyl, benzoyl, phenyl, pyridyl or pyrimidyl; Ra is H, C1-6 alkyl, or C2-6 alkenyl; “” represents a single bond or a double bond wherein n=1 or 2; Y is S or O; and R3 and R4 are each independently H, C1-6 alkyl, hydroxy-C1-6 alkyl, C2-7 acyl, phenyl, pyridyl, pyrimidyl, etc.;with the proviso that at least one R3 is a group other than C1-3 alkyl in the case where: the hetero ring containing Y is a thiazoline ring; R4═Ra═H; X1═X2═CH; and either p =0 or R5═C1-6 alkyl.

    摘要翻译： 本发明提供对黑素生成具有优异抑制作用并可用作增白剂的化合物和含有该化合物的皮肤外用制剂。 本发明的增白剂作为活性成分，含有式（1）表示的杂环化合物或其药理学上可接受的盐：其中A为C1-6烷基，C5-6环烷基，苄基，苄基羰基，苯甲酰基，苯基 ，吡啶基或嘧啶基; R a是H，C 1-6烷基或C 2-6烯基; “”表示单键或双键，其中n = 1或2; Y为S或O; 并且R 3和R 4各自独立地为H，C 1-6烷基，羟基-C 1-6烷基，C 2-7酰基，苯基，吡啶基，嘧啶基等;条件是至少一个R 3是除C1- 3烷基，其中：含有Y的杂环是噻唑啉环; R4 = R = X1 = X2 = CH; 和p = 0或R5 = C1-6烷基。