N-ACRYLIMINO HETEROCYCLIC COMPOUNDS
    1.
    发明申请
    N-ACRYLIMINO HETEROCYCLIC COMPOUNDS 审中-公开
    N-丙烯酰胺杂环化合物

    公开(公告)号:US20160235069A1

    公开(公告)日:2016-08-18

    申请号:US15023176

    申请日:2014-09-19

    Applicant: BASF SE

    Abstract: The present invention relates to N-acrylimino compound of formula (I): wherein X is O or S, in particular O; Het is a 5- or 6-membered carbon-bound or nitrogen-bound heterocyclic ring, W1-W2-W3-W4 represents a carbon chain group connected to N and C═N, and thus forming a saturated, unsaturated, or partially unsaturated 5 or 6 membered nitrogen containing heterocycle, wherein W1, W2, W3 and W4 each individually represent CRvRw, R1, R2 may be hydrogen, halogen, etc. R3 is selected from the group consisting of hydrogen, halogen, CN, C1-C6-alkyl, etc. R4 is selected from the group consisting of hydrogen, halogen, CN, C1-C10-alkyl, etc. R5 is selected from the group consisting of hydrogen CN, C1-C10-alkyl, C2-C10-alkenyl C3-C8-cycloalkyl, S(O)nNR9aR9b, O—NR9aR9b, NR9aR9b, NR9a NR9aR9b, NR9aC(═O)R7a, NR9aC(═S)R7a, NR9aC(═O)NR9aR9b, NR9aC(═S)NR9aR9b, C(═O)OR8, C(═O)NR9aR9b, C(═S)NR9aR9b, C(═O)R7a, C(═S)R7a, a moitey Q-phenyl, where the phenyl ring is optionally substituted with 1, 2, 3, 4 or 5 identical or different substituents R10, and a moiety Q-Het# where Het# represents a 3- to 10-membered saturated, partly saturated or unsaturated aromatic heterocyclic ring. The invention also relates to the use of the N-acrylimino heterocyclic compounds, their stereoisomers, their tautomers and their salts, for combating invertebrate pests. Furthermore the invention relates also to methods of combating invertebrate pests, which comprises applying such compounds.

    Abstract translation: 本发明涉及式(I)的N-丙烯酰亚氨基化合物:其中X是O或S,特别是O; Het是5或6元碳键或氮键合的杂环,W1-W2-W3-W4表示与N和C = N连接的碳链基团,因此形成饱和的,不饱和的或部分不饱和的 5或6元含氮杂环,其中W1,W2,W3和W4各自独立地表示CRvRw,R1,R2可以是氢,卤素等。R3选自氢,卤素,CN,C1-C6- 烷基等.R 4选自氢,卤素,CN,C 1 -C 10 - 烷基等。R 5选自氢CN,C 1 -C 10 - 烷基,C 2 -C 10 - 烯基C3- C 9 - 环烷基,S(O)n NR 9 a R 9 b,O-NR 9 a R 9 b,NR 9 a R 9 b,NR 9 a NR 9 a R 9 b,NR 9 a C(= O)R 7a,NR 9 a C(≡S)R 7a,NR 9 a C(≡O)NR 9 a R 9 b,NR 9 a C(≡S)NR 9 a R 9 b,C O)OR 8,C(= O)NR 9 a R 9 b,C(= S)NR 9 a R 9 b,C(= O)R 7a,C(= O)R 7a,其中苯环任选被1,2, 3,4或5个相同或不同的取代基R10,和其中Het#表示a的部分Q-Het# 3-至10-元饱和,部分饱和或不饱和的芳族杂环。 本发明还涉及N-丙烯酰胺杂环化合物,其立体异构体,其互变异构体及其盐的用途,用于对抗无脊椎动物害虫。 此外,本发明还涉及防治无脊椎害虫的方法,其包括施用这样的化合物。

    Substituted Pyrimidinium Compounds and Derivatives for Combating Animal Pests
    2.
    发明申请
    Substituted Pyrimidinium Compounds and Derivatives for Combating Animal Pests 有权
    取代的嘧啶鎓化合物和衍生物用于防治动物害虫

    公开(公告)号:US20160058009A1

    公开(公告)日:2016-03-03

    申请号:US14783600

    申请日:2014-04-11

    Applicant: BASF SE

    Abstract: Substituted pyrimidinium compounds of the general formula (I) and their uses for combating animal pestsThe present invention relates to substituted pyrimidinium compounds of formula (I), to the stereoisomers, salts, tautomers and N-oxides thereof and to compositions comprising such compounds. The invention also relates to methods and uses of these substituted pyrimidinium compounds and of compositions thereof, for combating and controlling animal pests. Furthermore the invention relates also to pesticidal methods of applying such substituted pyrimidinium compounds.The substituted pyrimidinium compounds of the present invention are defined by the following general formula (I): wherein X, Y, Z, R1, R2, A and Het are defined as in the description.

    Abstract translation: 通式(I)的取代嘧啶化合物及其用于对抗动物害虫的用途本发明涉及式(I)的取代嘧啶鎓化合物,其立体异构体,盐,互变异构体和N-氧化物以及包含这些化合物的组合物。 本发明还涉及这些取代的嘧啶鎓化合物及其组合物用于对抗和控制动物害虫的方法和用途。 此外,本发明还涉及施用这种取代的嘧啶鎓化合物的杀虫方法。 本发明的取代的嘧啶鎓化合物由以下通式(I)定义:其中X,Y,Z,R 1,R 2,A和Het如描述中所定义。

    N-Acylimino Heterocyclic Compounds
    3.
    发明申请

    公开(公告)号:US20190142004A1

    公开(公告)日:2019-05-16

    申请号:US16245471

    申请日:2019-01-11

    Applicant: BASF SE

    Abstract: The present invention relates to N-acylimino compound of formula (I): wherein X is O or S, in particular O; m is an integer selected from 0, 1, 2, 3, 4, 5 or 6; Het is a 5 or 6 membered carbon-bound or nitrogen-bound heterocyclic ring, W1-W2-W3-W4 represents a carbon chain group connected to N and C═N, and thus forming a saturated, unsaturated, or partially unsaturated 5 or 6 membered nitrogen containing heterocycle, wherein W1, W2, W3 and W4 each individually represent CRvRw, R1, R2 may be hydrogen, halogen, etc. R3 may be hydrogen, halogen, CN, C1-C6-alkyl, etc. R4a, R4b if present, may be hydrogen, halogen, C1-C6-alkyl, etc. R5 may be hydrogen, halogen, C1-C6-alkyl, C1-C6-alkenyl, C1-C6-alkinyl, C3-C8-cycloalkyl, S(O)nNR9aR9b, NR9aR9b, C(═O)OR8, C(═O)NR9aR9b, C(═S)NR9aR9b, C(═O)R7a, C(═S)R7a, NR9a—C(═O)R7a, NR9a—C(═S)R7a, NR9a—S(O)nR8a, a moitey Q-phenyl, where the phenyl ring is optionally substituted with one or more, e.g. 1, 2, 3, 4 or 5 identical or different substituents R10, or a moiety Q-Het#, or R3 and R5 together may also form with the carbon atom they are bound to, a 3, 4, 5 or 6 membered saturated partially unsaturated carbocycle or heterocycle. The invention also relates to the use of the N-acylimino heterocyclic compounds, their stereoisomers, their tautomers and their salts, for combating invertebrate pests. Furthermore the invention relates also to methods of combating invertebrate pests, which comprises applying such compounds.

    Pesticide Compounds
    4.
    发明申请
    Pesticide Compounds 有权
    农药化合物

    公开(公告)号:US20160157491A1

    公开(公告)日:2016-06-09

    申请号:US14903887

    申请日:2014-07-14

    Applicant: BASF SE

    Abstract: The present invention relates to novel compounds of the formula I and the N-oxides, stereoisomers, tautomers and agriculturally or veterinarily acceptable salts thereof wherein C1 is C or CH; C2 is C or CH; A1 is N or C; A2 is N, C(R2), N(R3), O, S or C(R4,R5); and A3 is N, O, S, N(R6), C(R7) or C(R8,R9); where one or two non-adjacent bonds in the 5-membered ring formed by C1, C2, A1, A2 and A3 are double bonds, while the others are single bonds, provided that the bond between A1 and A2 or the bond between A1 and C1 or the bond between A2 and A3 or the bond between C1 and C2 or the bond between A3 and C2 is a double bond further provided that at least one of A1, A2 and A3 is N, N(R3) or N(R6), and where Ar, R1, R2, R3, R4, R5, R6, R7, R8, R9 and (R)k are as defined in the claims and in the description, which are useful for combating or controlling invertebrate pests, in particular arthropod pests and nematodes. The invention also relates to a method for controlling invertebrate pests by using these compounds and to plant propagation material and to an agricultural and a veterinary composition comprising said compounds.

    Abstract translation: 本发明涉及式I的新化合物和N-氧化物,立体异构体,互变异构体及其农业或兽医学上可接受的盐,其中C 1是C或CH; C2是C或CH; A1为N或C; A2是N,C(R2),N(R3),O,S或C(R4,R5); 并且A3是N,O,S,N(R6),C(R7)或C(R8,R9); 其中由C1,C2,A1,A2和A3形成的5元环中一个或两个不相邻的键是双键,而其它的是单键,条件是A1和A2之间的键或A1和 C1或A2和A3之间的键或C1和C2之间的键或A3和C2之间的键是双键,进一步规定A1,A2和A3中的至少一个是N,N(R3)或N(R6) ,其中Ar,R 1,R 2,R 3,R 4,R 5,R 6,R 7,R 8,R 9,R 6,R 7,R 8,R 9和(R)k如权利要求书和说明书中所定义,其可用于防治或控制无脊椎害虫, 节肢动物害虫和线虫。 本发明还涉及通过使用这些化合物和植物繁殖材料以及包含所述化合物的农业和兽用组合物来控制无脊椎害虫的方法。

    N-SUBSTITUTED ACYL-IMINO-PYRIDINE COMPOUNDS AND DERIVATIVES FOR COMBATING ANIMAL PESTS
    6.
    发明申请
    N-SUBSTITUTED ACYL-IMINO-PYRIDINE COMPOUNDS AND DERIVATIVES FOR COMBATING ANIMAL PESTS 审中-公开
    N-取代的亚氨基 - 吡啶化合物和用于组合动物饲料的衍生物

    公开(公告)号:US20160050923A1

    公开(公告)日:2016-02-25

    申请号:US14784126

    申请日:2014-04-15

    Applicant: BASF SE

    Abstract: The invention relates to N-substituted acyl-imino-pyridine compounds of formula (I), to the enantiomers, diastereomers and salts thereof and to compositions comprising such compounds. The invention also relates to methods and uses of these N-substituted acyl-imino-pyridine compounds, and of compositions comprising thereof, for combating and controlling animal pests. Furthermore the invention relates also to pesticidal methods of applying such N-substituted acyl-imino-pyridine compounds.The N-substituted acyl-imino-pyridine compounds of the present invention are defined by the following formula I: wherein p, X, Y, W1, W2, W3, W4, Het, R1, R2, R3a, R3b, R4a, R4b and R5 are defined as in the description.

    Abstract translation: 本发明涉及式(I)的N-取代酰基 - 亚氨基 - 吡啶化合物,其涉及其对映体,非对映异构体和盐以及包含这些化合物的组合物。 本发明还涉及这些N-取代的酰基 - 亚氨基 - 吡啶化合物及其组合物的方法和用途,用于对抗和控制动物害虫。 此外,本发明还涉及施用这种N-取代的酰基 - 亚氨基 - 吡啶化合物的杀虫方法。 本发明的N-取代酰基亚氨基 - 吡啶化合物由下式I定义:其中p,X,Y,W1,W2,W3,W4,Het,R1,R2,R3a,R3b,R4a,R4b 和R5如说明书中所定义。

    N-ACYLIMINO HETEROCYCLIC COMPOUNDS
    7.
    发明申请
    N-ACYLIMINO HETEROCYCLIC COMPOUNDS 有权
    N-乙酰氨基杂环化合物

    公开(公告)号:US20160297793A1

    公开(公告)日:2016-10-13

    申请号:US15038272

    申请日:2014-11-21

    Applicant: BASF SE

    Abstract: The present invention relates to N-acylimino compound of formula (I): wherein X is O or S, in particular O; Y is a single bond, O, S or NR5; Het is a 5 or 6 membered carbon-bound or nitrogen-bound heterocyclic ring, W1—W2—W3—W4 represents a carbon chain group connected to N and C═N, and thus forming a saturated, unsaturated, or partially unsaturated 5 or 6 membered nitrogen containing heterocycle, wherein W1, W2, W3 and W4 each individually represent CRvRw; R1, R2 may be hydrogen, halogen, etc.; R3 may be hydrogen, CN, C1-C6-alkyl, etc.; R4 may be of hydrogen, C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkinyl, C3-C8-cycloalkyl, Q-phenyl, Q′-O-phenyl, Q′-S-phenyl, where the phenyl ring is optionally substituted with one or more, e.g. 1, 2, 3, 4 or 5 identical or different substituents R10, and the moieties Q-Het#, Q′-O-Het# and Q′-S-Het# where Het# represents a heterocyclic radical and where Q and Q′ are C1-C6-alkandiyl, C2-C6-alkendiyl, or C2-C6-alkyndiyl, and where Q may also be a single bond; R3 and R4 together may also may also a bivalent radical, selected from the group consisting of C2-C5-alkandiyl, C2-C5-alkendiyl, Q″-C1-C4-alkandiyl and Q″-C2-C4-alkendiyl, where Q″ is O or S. The invention also relates to the use of the N-acylimino heterocyclic compounds, their stereoisomers, their tautomers and their salts, for combating invertebrate pests. Furthermore the invention relates also to methods of combating invertebrate pests, which comprises applying such compounds.

    Abstract translation: 本发明还涉及N-酰基亚氨基杂环化合物,其立体异构体,其互变异构体及其盐的用途,用于防治无脊椎动物害虫。 此外,本发明还涉及防治无脊椎害虫的方法,其包括施用这样的化合物。

    N-Acylimino Heterocyclic Compounds
    8.
    发明申请
    N-Acylimino Heterocyclic Compounds 审中-公开
    N-酰基亚氨基杂环化合物

    公开(公告)号:US20160227777A1

    公开(公告)日:2016-08-11

    申请号:US15023128

    申请日:2014-09-18

    Applicant: BASF SE

    Abstract: The present invention relates to N-acylimino compound of formula (I): wherein X is O or S, in particular O; m is an integer selected from 0, 1, 2, 3, 4, 5 or 6; Het is a 5 or 6 membered carbon-bound or nitrogen-bound heterocyclic ring, W1-W2-W3-W4 represents a carbon chain group connected to N and C═N, and thus forming a saturated, unsaturated, or partially unsaturated 5 or 6 membered nitrogen containing heterocycle, wherein W1, W2, W3 and W4 each individually represent CRvRw, R1, R2 may be hydrogen, halogen, etc. R3 may be hydrogen, halogen, CN, C1-C6-alkyl, etc. R4a, R4b if present, may be hydrogen, halogen, C1-C6-alkyl, etc. R5 may be hydrogen, halogen, C1-C6-alkyl, C1-C6-alkenyl, C1-C6-alkinyl, C3-C8-cycloalkyl, S(O)nNR9aR9b, NR9aR9b, C(═O)OR8, C(═O)NR9aR9b, C(═S)NR9aR9b, C(═O)R7a, C(═S)R7a, NR9a—C(═O)R7a, NR9a—C(═S)R7a, NR9a—S(O)nR8a, a moiety Q-phenyl, where the phenyl ring is optionally substituted with one or more, e.g. 1, 2, 3, 4 or 5 identical or different substituents R10, or a moiety Q-Het#, or R3 and R5 together may also form with the carbon atom they are bound to, a 3, 4, 5 or 6 membered saturated partially unsaturated carbocycle or heterocycle. The invention also relates to the use of the N-acylimino heterocyclic compounds, their stereoisomers, their tautomers and their salts, for combating invertebrate pests. Furthermore the invention relates also to methods of combating invertebrate pests, which comprises applying such compounds.

    Abstract translation: 本发明涉及式(I)的N-酰基亚胺基化合物:其中X是O或S,特别是O; m为选自0,1,2,3,4,5或6的整数; Het是5或6元碳键或氮键的杂环,W1-W2-W3-W4表示与N和C = N连接的碳链基团,从而形成饱和的,不饱和的或部分不饱和的5或 6元含氮杂环,其中W1,W2,W3和W4各自独立地表示CRvRw,R1,R2可以是氢,卤素等。R3可以是氢,卤素,CN,C1-C6-烷基等。R4a,R4b R 5可以是氢,卤素,C 1 -C 6 - 烷基,C 1 -C 6 - 烯基,C 1 -C 6 - 炔基,C 3 -C 8 - 环烷基,S( O(n)NR 9a R 9 b,C(= O)OR 8,C(= O)NR 9 a R 9 b,C(= S)NR 9 a R 9 b,C(= O) NR9a-C(= S)R7a,NR9a-S(O)nR8a,部分Q-苯基,其中苯环任选被一个或多个例如 1,2,3或4或5个相同或不同的取代基R10或部分Q-Het#,或R3和R5一起也可以与它们所键合的碳原子一起形成,3,4,5或6元饱和 部分不饱和碳环或杂环。 本发明还涉及N-酰基亚氨基杂环化合物,其立体异构体,其互变异构体及其盐的用途,用于防治无脊椎动物害虫。 此外,本发明还涉及防治无脊椎害虫的方法,其包括施用这样的化合物。

    Substituted Pyrimidinium Compounds and Derivatives for Combating Animal Pests
    9.
    发明申请
    Substituted Pyrimidinium Compounds and Derivatives for Combating Animal Pests 有权
    取代的嘧啶鎓化合物和衍生物用于防治动物害虫

    公开(公告)号:US20160122351A1

    公开(公告)日:2016-05-05

    申请号:US14898892

    申请日:2014-06-17

    Applicant: BASF SE

    CPC classification number: C07D471/16 A01N43/90 C07D471/14

    Abstract: Substituted pyrimidinium compounds of the general formula (I) and their uses for combating animal pestsThe present invention relates to substituted pyrimidinium compounds of formula (I), to the stereoisomers, salts, tautomers and N-oxides thereof and to compositions comprising such compounds. The invention also relates to methods and uses of these substituted pyrimidinium compounds and of compositions thereof, for combating and controlling animal pests. Furthermore the invention relates also to pesticidal methods of applying such substituted pyrimidinium compounds.The substituted pyrimidinium compounds of the present invention are defined by the following general formula (I): wherein X, Y, Z, R1, R2, A, A1 and A2 are defined as in the description.

    Abstract translation: 通式(I)的取代嘧啶化合物及其用于对抗动物害虫的用途本发明涉及式(I)的取代嘧啶鎓化合物,其立体异构体,盐,互变异构体和N-氧化物以及包含这些化合物的组合物。 本发明还涉及这些取代的嘧啶鎓化合物及其组合物用于对抗和控制动物害虫的方法和用途。 此外,本发明还涉及施用这种取代的嘧啶鎓化合物的杀虫方法。 本发明的取代的嘧啶鎓化合物由以下通式(I)定义:其中X,Y,Z,R 1,R 2,A,A 1和A 2如说明书中所定义。

    2-(PYRIDIN-3-YL)-5-HETARYL-THIAZOLE COMPOUNDS CARRYING AN IMINE OR IMINE-DERIVED SUBSTITUENT FOR COMBATING INVERTEBRATE PESTS
    10.
    发明申请
    2-(PYRIDIN-3-YL)-5-HETARYL-THIAZOLE COMPOUNDS CARRYING AN IMINE OR IMINE-DERIVED SUBSTITUENT FOR COMBATING INVERTEBRATE PESTS 审中-公开
    2-(吡啶-3-基)-5-羟基 - 噻唑化合物,其承载用于混合反相物质的烟草或衍生物

    公开(公告)号:US20150368236A1

    公开(公告)日:2015-12-24

    申请号:US14654933

    申请日:2013-12-23

    Applicant: BASF SE

    CPC classification number: C07D417/14 A01N43/78 A01N43/84 C07D413/14

    Abstract: The present invention relates to 2-(pyridin-3-yl)-5-hetaryl-thiazole compounds carrying an imine or imine-derived substituent on the 5-hetaryl ring which are useful for combating or controlling invertebrate pests, in particular arthropod pests and nematodes, and to a method for producing them. The invention also relates to a method for controlling invertebrate pests by using these compounds and to plant propagation material and to an agricultural and a veterinary composition comprising said compounds.

    Abstract translation: 本发明涉及在5-杂芳基环上携带亚胺或亚胺衍生的取代基的2-(吡啶-3-基)-5-辛烷基 - 噻唑化合物,它们可用于防治或控制无脊椎害虫,特别是节肢动物害虫和 线虫,以及生产它们的方法。 本发明还涉及通过使用这些化合物和植物繁殖材料以及包含所述化合物的农业和兽用组合物来控制无脊椎害虫的方法。

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