公开(公告)号：US09095136B2

公开(公告)日：2015-08-04

申请号：US14360007

申请日：2012-11-23

Applicant: BAYER INTELLECTUAL PROPERTY GMBH

Inventor： Hendrik Helmke ,  Sebastian Hoffmann ,  Carl Friedrich Nising ,  Alexander Sudau ,  Tomoki Tsuchiya ,  Jürgen Benting ,  Peter Dahmen ,  Ulrike Wachendorff-Neumann ,  David Bernier ,  Stephane Brunet ,  Marie-Claire Grosjean-Cournoyer ,  Hélène Lachaise ,  Philippe Rinolfi

IPC: A01N43/50 ,  C07D233/68 ,  C07D405/06

CPC classification number: A01N43/50 ,  A01N43/76 ,  A01N43/78 ,  A01N55/00 ,  C07C49/213 ,  C07C49/255 ,  C07D233/68 ,  C07D263/32 ,  C07D277/24 ,  C07D303/34 ,  C07D405/06 ,  C07F7/0814

Abstract: The present invention relates to novel 2-iodoimidazole derivatives, to processes for preparing these compounds, to compositions comprising these compounds and to their use as biologically active compounds, in particular for controlling harmful microorganisms in crop protection and in the protection of materials and as plant growth regulators.

Abstract translation: 本发明涉及新的2-碘咪唑衍生物，制备这些化合物的方法，包含这些化合物的组合物及其作为生物活性化合物的用途，特别是用于防止作物保护中的有害微生物和保护材料和植物 生长调节剂。

公开(公告)号：US20140336232A1

公开(公告)日：2014-11-13

申请号：US14360007

申请日：2012-11-23

Applicant: BAYER INTELLECTUAL PROPERTY GMBH

Inventor： Hendrik Helmke ,  Sebastian Hoffmann ,  Carl Friedrich Nising ,  Alexander Sudau ,  Tomoki Tsuchiya ,  Jürgen Benting ,  Peter Dahmen ,  Ulrike Wachendorff-Neumann ,  David Bernier ,  Stephane Brunet ,  Marie-Claire Grosjean-Cournoyer ,  Hélène Lachaise ,  Philippe Rinolfi

IPC: A01N43/50 ,  C07D405/06 ,  C07D233/68

CPC classification number: A01N43/50 ,  A01N43/76 ,  A01N43/78 ,  A01N55/00 ,  C07C49/213 ,  C07C49/255 ,  C07D233/68 ,  C07D263/32 ,  C07D277/24 ,  C07D303/34 ,  C07D405/06 ,  C07F7/0814

Abstract: The present invention relates to novel 2-iodoimidazole derivatives, to processes for preparing these compounds, to compositions comprising these compounds and to their use as biologically active compounds, in particular for controlling harmful microorganisms in crop protection and in the protection of materials and as plant growth regulators.

Abstract translation: 本发明涉及新的2-碘咪唑衍生物，制备这些化合物的方法，包含这些化合物的组合物及其作为生物活性化合物的用途，特别是用于防止作物保护中的有害微生物和保护材料和植物 生长调节剂

公开(公告)号：US20140274952A1

公开(公告)日：2014-09-18

申请号：US14360437

申请日：2012-11-23

Applicant: BAYER INTELLECTUAL PROPERTY GMBH

Inventor： Sebastian Hoffmann ,  Hendrik Helmke ,  Gorka Peris ,  Friedrich Carl Nising ,  Tomoki Tsuchiya ,  Alexander Sudau ,  Jürgen Benting ,  David Bernier

IPC: A01N43/78 ,  A01N55/00 ,  A01N43/76 ,  C07C49/213 ,  C07C49/255 ,  C07D303/34

CPC classification number: A01N43/50 ,  A01N43/76 ,  A01N43/78 ,  A01N55/00 ,  C07C49/213 ,  C07C49/255 ,  C07D233/68 ,  C07D263/32 ,  C07D277/24 ,  C07D303/34 ,  C07D405/06 ,  C07F7/0814

Abstract: The present invention relates to novel heterocyclic alkanol derivatives, to processes for these compounds, to compositions comprising these compounds and to their use as biologically active compounds, in particular for controlling harmful microorganisms in crop protection and in the protection of materials and as plant growth regulators.

Abstract translation: 本发明涉及新型杂环烷醇衍生物，这些化合物的方法，包含这些化合物的组合物及其作为生物活性化合物的用途，特别是用于在作物保护和材料保护以及植物生长调节剂中控制有害微生物 。

公开(公告)号：US20140088153A1

公开(公告)日：2014-03-27

申请号：US14005414

申请日：2012-03-12

Applicant: BAYER INTELLECTUAL PROPERTY GMBH

Inventor： Michael Maue ,  Isabelle Adelt ,  Markus Heil ,  Peter Jeschke ,  Tobias Kapferer ,  Friedrich August Muehlthau ,  Alexander Sudau ,  Olga Malsam ,  Peter Loesel ,  Arnd Voerste ,  Ulrich Goergens

IPC: C07D231/14 ,  C07D401/12 ,  C07C237/38 ,  C07D231/18 ,  C07D231/16 ,  A01N43/56

CPC classification number: C07D231/14 ,  A01N43/56 ,  C07C237/38 ,  C07C255/46 ,  C07C2601/02 ,  C07D231/16 ,  C07D231/18 ,  C07D401/12

Abstract: The invention relates to compounds of the general formula (I) in which the radicals A1, A2, A3, A4, L, Q, R1, T and W have the meaning given in the description and to the use of the compounds for controlling animal pests. The invention furthermore relates to processes and intermediates for preparing the compounds of formula (I).

Abstract translation: 本发明涉及通式（I）的化合物，其中基团A1，A2，A3，A4，L，Q，R1，T和W具有说明书中给出的含义以及用于控制动物的化合物的用途 害虫 本发明还涉及制备式（I）化合物的方法和中间体。

公开(公告)号：US09198429B2

公开(公告)日：2015-12-01

申请号：US14360437

申请日：2012-11-23

Applicant: BAYER INTELLECTUAL PROPERTY GMBH

Inventor： Sebastian Hoffmann ,  Hendrik Helmke ,  Gorka Peris ,  Friedrich Carl Nising ,  Tomoki Tsuchiya ,  Alexander Sudau ,  Jürgen Benting ,  David Bernier

IPC: A01N43/76 ,  A01N43/78 ,  A01N55/00 ,  C07D263/32 ,  C07D277/24 ,  C07F7/10 ,  C07F7/08 ,  C07C49/213 ,  C07C49/255 ,  C07D303/34

CPC classification number: A01N43/50 ,  A01N43/76 ,  A01N43/78 ,  A01N55/00 ,  C07C49/213 ,  C07C49/255 ,  C07D233/68 ,  C07D263/32 ,  C07D277/24 ,  C07D303/34 ,  C07D405/06 ,  C07F7/0814

Abstract: The present invention related to novel heterocyclic alkanol derivatives, to processes for preparing these compounds, to compositions comprising these compounds and to their use as biologically active compounds, in particular for controlling harmful microorganisms in crop protection in the protection of materials and as plat growth regulations.

Abstract translation: 本发明涉及新型杂环烷醇衍生物，制备这些化合物的方法，涉及包含这些化合物的组合物及其作为生物活性化合物的用途，特别是用于在作物保护中控制有害微生物以保护材料和作为平板生长规则 。

公开(公告)号：US20140256677A1

公开(公告)日：2014-09-11

申请号：US14349144

申请日：2012-10-04

Applicant: BAYER INTELLECTUAL PROPERTY GMBH

Inventor： Stefan Hillebrand ,  Amos Mattes ,  Alexander Sudau ,  Pierre Wasnaire ,  Jürgen Benting ,  Peter Dahmen ,  Ulrike Wachendorff-Neumann ,  Haruko Sawada ,  Philippe Desbordes ,  Anne-Sophie Rebstock ,  Stéphane Brunet ,  Hélène Lachaise ,  Philippe Rinolfi

IPC: A01N43/90 ,  A01N55/00 ,  A01N53/00

CPC classification number: A01N43/90 ,  A01N53/00 ,  A01N55/00 ,  C07D471/04 ,  C07D487/04 ,  C07D498/04 ,  C07D513/04

Abstract: Heterocyclylpyri(mi)dinylpyrazole of the formula (I) in which R1 to R5, X1, U, Q, W, Y, n, a, b have the meanings given in the description, and agrochemically active salts, to their use and to methods and compositions for controlling phytopathogenic harmful fungi in and/or on plants or in and/or on seed of plants and for reducing mycotoxins in plants and parts of the plants, to processes for preparing such compounds and compositions and treated seed and also to their use for controlling phytopathogenic harmful fungi in agriculture, horticulture, forestry, in animal husbandry, in the protection of materials, in the domestic and hygiene field and for the reduction of mycotoxins in plants and parts of the plants

Abstract translation: 其中R1至R5，X1，U，Q，W，Y，n，a，b具有本说明书中给出的含义的式（I）的二环戊基吡啶（mi）二乙基吡唑，以及农用化学活性盐， 用于控制植物中和/或植物中或植物中和/或植物和/或植物种子和用于减少植物和部分植物中的真菌毒素的植物病原性有害真菌的方法和组合物，用于制备这些化合物和组合物和处理过的种子的方法以及它们 用于控制农业，园艺，林业，畜牧业中的植物病原性有害真菌，保护材料，在家庭和卫生领域以及减少植物和植物部分的真菌毒素

公开(公告)号：US09314026B2

公开(公告)日：2016-04-19

申请号：US14349971

申请日：2012-10-04

Applicant: Bayer Intellectual Property GmbH

Inventor： Alexander Sudau ,  Hendrik Helmke ,  Stefan Hillebrand ,  Amos Mattes ,  Lars Rodefeld ,  Pierre Wasnaire ,  Jürgen Benting ,  Peter Dahmen ,  Ulrike Wachendorff-Neumann ,  Philippe Desbordes ,  Anne-Sophie Rebstock

IPC: A61K31/44 ,  C07D491/02 ,  C07D401/00 ,  A01N43/90 ,  C07D487/04 ,  C07D498/04

CPC classification number: A01N43/90 ,  C07D487/04 ,  C07D498/04

Abstract: Heterocyclylpyri(mi)dinylpyrazole of the formula (I), in which R1 to R5, X1, U, Q, W, a, b and n have the meanings given in the description, and agrochemically active salts, to their use and to methods and compositions for controlling phytopathogenic harmful fungi in and/or on plants or in and/or on seed of plants and for reducing mycotoxins in plants and parts of the plants, to processes for preparing such compounds and compositions and treated seed and also to their use for controlling phytopathogenic harmful fungi in agriculture, horticulture, forestry, in animal husbandry, in the protection of materials, in the domestic and hygiene field and for the reduction of mycotoxins in plants and parts of the plants.

Abstract translation: 其中R1至R5，X1，U，Q，W，a，b和n具有本说明书中给出的含义的式（I）的杂环基吡啶（mi）二乙基吡唑，以及农用化学活性盐，其用途和方法 以及用于在植物中和/或植物中或植物种子和/或植物中植物和/或植物中和/或植物中和/或植物中部分植物病原性有害真菌和用于减少植物和植物部分的真菌毒素的组合物，用于制备这些化合物和组合物以及处理过的种子的方法， 用于控制农业，园艺，林业，畜牧业中的植物病原性有害真菌，保护材料，在国内和卫生领域以及减少植物和植物部分的真菌毒素。

公开(公告)号：US09023844B2

公开(公告)日：2015-05-05

申请号：US14349144

申请日：2012-10-04

Applicant: Bayer Intellectual Property GmbH

Inventor： Stefan Hillebrand ,  Amos Mattes ,  Alexander Sudau ,  Pierre Wasnaire ,  Jürgen Benting ,  Peter Dahmen ,  Ulrike Wachendorff-Neumann ,  Haruko Sawada ,  Philippe Desbordes ,  Anne-Sophie Rebstock ,  Stéphane Brunet ,  Hélène Lachaise ,  Philippe Rinolfi

IPC: C07D471/04 ,  C07D487/04 ,  C07D498/04 ,  A01N43/90 ,  C07D513/04 ,  A01N53/00 ,  A01N55/00

CPC classification number: A01N43/90 ,  A01N53/00 ,  A01N55/00 ,  C07D471/04 ,  C07D487/04 ,  C07D498/04 ,  C07D513/04

Abstract: Heterocyclylpyri(mi)dinylpyrazole of the formula (I) in which R1 to R5, X1, U, Q, W, Y, n, a, b have the meanings given in the description, and agrochemically active salts, to their use and to methods and compositions for controlling phytopathogenic harmful fungi in and/or on plants or in and/or on seed of plants and for reducing mycotoxins in plants and parts of the plants, to processes for preparing such compounds and compositions and treated seed and also to their use for controlling phytopathogenic harmful fungi in agriculture, horticulture, forestry, in animal husbandry, in the protection of materials, in the domestic and hygiene field and for the reduction of mycotoxins in plants and parts of the plants.

Abstract translation: 其中R1至R5，X1，U，Q，W，Y，n，a，b具有本说明书中给出的含义的式（I）的二环戊基吡啶（mi）二乙基吡唑，以及农用化学活性盐， 用于控制植物中和/或植物中或植物中和/或植物和/或植物中植物病原性有害真菌的方法和组合物，以及用于减少植物和植物部分的真菌毒素，制备这些化合物和组合物和处理过的种子的方法以及它们 用于控制农业，园艺，林业，畜牧业中的植物病原性有害真菌，保护材料，在国内和卫生领域以及减少植物和植物部分的真菌毒素。

公开(公告)号：US20140256728A1

公开(公告)日：2014-09-11

申请号：US14355429

申请日：2012-10-29

Applicant: BAYER INTELLECTUAL PROPERTY GMBH

Inventor： Jörg Nico Greul ,  Heiko Rieck ,  Christian Paulitz ,  Matthias Riedrich ,  Ralf Dunkel ,  Arianna Martelletti ,  Alexander Sudau ,  Peter Lösel ,  Olga Malsam ,  Arnd Voerste ,  Hans-Georg Schwarz ,  Ulrich Görgens ,  Kerstin Ilg ,  Michael Maue ,  Pierre-Yves Coqueron ,  Philippe Desbordes ,  Philippe Meresse ,  Stephanie Gary ,  Pierre Cristau ,  David Bernier

IPC: A01N43/40 ,  A01N43/80 ,  A01N43/82 ,  A01N43/647 ,  A01N43/76 ,  A01N43/84 ,  A01N43/56 ,  A01N43/78

CPC classification number: A01N43/40 ,  A01N43/08 ,  A01N43/10 ,  A01N43/18 ,  A01N43/36 ,  A01N43/54 ,  A01N43/56 ,  A01N43/60 ,  A01N43/647 ,  A01N43/707 ,  A01N43/76 ,  A01N43/78 ,  A01N43/80 ,  A01N43/82 ,  A01N43/84 ,  A61K31/443 ,  A61K31/4436 ,  A61K31/4439 ,  A61K31/444 ,  A61K31/4545 ,  A61K31/497 ,  A61K31/5377 ,  C07D213/81 ,  C07D213/82 ,  C07D401/12 ,  C07D401/14 ,  C07D405/12 ,  C07D409/12 ,  C07D411/12 ,  C07D413/12 ,  C07D417/12 ,  C07D417/14

Abstract: The present invention relates to the use of predominantly known pyridyl carboxamide derivatives as nematicides, compositions containing such compounds and methods for the control of nematodes.

Abstract translation: 本发明涉及主要已知的吡啶甲酰胺衍生物作为杀线虫剂的用途，含有这些化合物的组合物和用于控制线虫的方法。

公开(公告)号：US20140364456A1

公开(公告)日：2014-12-11

申请号：US14349971

申请日：2012-10-04

Applicant: Bayer Intellectual Property GmbH

Inventor： Alexander Sudau ,  Hendrik Helmke ,  Stefan Hillebrand ,  Amos Mattes ,  Lars Rodefeld ,  Pierre Wasnaire ,  Jürgen Benting ,  Peter Dahmen ,  Ulrike Wachendorff-Neumann ,  Philippe Desbordes ,  Anne-Sophie Rebstock

IPC: A01N43/90

CPC classification number: A01N43/90 ,  C07D487/04 ,  C07D498/04

Abstract: Heterocyclylpyri(mi)dinylpyrazole of the formula (I), in which R1 to R5, X1, U, Q, W, a, b and n have the meanings given in the description, and agrochemically active salts, to their use and to methods and compositions for controlling phytopathogenic harmful fungi in and/or on plants or in and/or on seed of plants and for reducing mycotoxins in plants and parts of the plants, to processes for preparing such compounds and compositions and treated seed and also to their use for controlling phytopathogenic harmful fungi in agriculture, horticulture, forestry, in animal husbandry, in the protection of materials, in the domestic and hygiene field and for the reduction of mycotoxins in plants and parts of the plants.

Abstract translation: 其中R1至R5，X1，U，Q，W，a，b和n具有本说明书中给出的含义的式（I）的杂环基吡啶（mi）二乙基吡唑，以及农用化学活性盐，其用途和方法 以及用于在植物中和/或植物中或植物种子和/或植物中植物和/或植物中和/或植物中和/或植物中部分植物病原性有害真菌和用于减少植物和植物部分的真菌毒素的组合物，用于制备这些化合物和组合物以及处理过的种子的方法， 用于控制农业，园艺，林业，畜牧业中的植物病原性有害真菌，保护材料，在国内和卫生领域以及减少植物和植物部分的真菌毒素。