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公开(公告)号:US20230390249A1
公开(公告)日:2023-12-07
申请号:US18453431
申请日:2023-08-22
Applicant: BRISTOL-MYERS SQUIBB COMPANY
Inventor: Peter Tai Wah Cheng , Robert F. Kaltenbach, III , Jun Li , Jun Shi , Yan Shi , Shiwei Tao , Hao Zhang , Suresh Dhanusu , Kumaravel Selvakumar , Ramesh Babu Reddigunta , Steven J. Walker , Lawrence J. Kennedy , James R. Corte , Tianan Fang , Sutjano Jusuf
IPC: A61K31/4192 , C07D401/14 , C07D249/06 , A61K31/27 , A61K31/454 , C07D401/04
CPC classification number: A61K31/4192 , C07D401/14 , C07D249/06 , A61K31/27 , A61K31/454 , C07D401/04 , A61K31/41
Abstract: The present invention provides compounds of Formula (I):
or stereoisomers, tautomers, pharmaceutically acceptable salts, solvates or prodrugs thereof, wherein all the variables are as defined herein. These compounds are selective LPA receptor inhibitors.-
公开(公告)号:US20170360759A1
公开(公告)日:2017-12-21
申请号:US15628104
申请日:2017-06-20
Applicant: BRISTOL-MYERS SQUIBB COMPANY
Inventor: Peter Tai Wah Cheng , Robert F. Kaltenbach, III , Jun LI , Jun Shi , Yan Shi , Shiwei Tao , Hao Zhang , Suresh Dhanusu , Kumaravel Selvakumar , Ramesh Babu Reddigunta , Steven J. Walker , Lawrence J. Kennedy , James R. Corte , Tianan Fang , Sutjano Jusuf
IPC: A61K31/4192 , A61K31/27 , C07D401/04 , A61K31/454 , C07C62/10 , A61K31/41
CPC classification number: A61K31/4192 , A61K31/27 , A61K31/41 , A61K31/454 , C07C62/10 , C07D249/06 , C07D401/04 , C07D401/14
Abstract: The present invention provides compounds of Formula (I): or stereoisomers, tautomers, pharmaceutically acceptable salts, solvates or prodrugs thereof, wherein all the variables are as defined herein. These compounds are selective LPA receptor inhibitors.
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公开(公告)号:US11007180B2
公开(公告)日:2021-05-18
申请号:US16732387
申请日:2020-01-02
Applicant: BRISTOL-MYERS SQUIBB COMPANY
Inventor: Peter Tai Wah Cheng , Robert F. Kaltenbach, III , Jun Li , Jun Shi , Yan Shi , Shiwei Tao , Hao Zhang , Suresh Dhanusu , Kumaravel Selvakumar , Ramesh Babu Reddigunta , Steven J. Walker , Lawrence J. Kennedy , James R. Corte , Tianan Fang , Sutjano Jusuf
IPC: C07D401/04 , A61K31/4192 , C07D401/14 , C07D249/06 , A61K31/27 , A61K31/454 , A61K31/41 , C07C62/10
Abstract: The present invention provides compounds of Formula (I): or stereoisomers, tautomers, pharmaceutically acceptable salts, solvates or prodrugs thereof, wherein all the variables are as defined herein. These compounds are selective LPA receptor inhibitors.
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公开(公告)号:US10071078B2
公开(公告)日:2018-09-11
申请号:US15628104
申请日:2017-06-20
Applicant: BRISTOL-MYERS SQUIBB COMPANY
Inventor: Peter Tai Wah Cheng , Robert F. Kaltenbach, III , Jun Li , Jun Shi , Yan Shi , Shiwei Tao , Hao Zhang , Suresh Dhanusu , Kumaravel Selvakumar , Ramesh Babu Reddigunta , Steven J. Walker , Lawrence J. Kennedy , James R. Corte , Tianan Fang , Sutjano Jusuf
IPC: C07D401/04 , A61K31/4192 , A61K31/27 , A61K31/454 , C07D401/14 , C07D249/06 , A61K31/41 , C07C62/10
CPC classification number: A61K31/4192 , A61K31/27 , A61K31/41 , A61K31/454 , C07C62/10 , C07D249/06 , C07D401/04 , C07D401/14
Abstract: The present invention provides compounds of Formula (I): or stereoisomers, tautomers, pharmaceutically acceptable salts, solvates or prodrugs thereof, wherein all the variables are as defined herein. These compounds are selective LPA receptor inhibitors.
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公开(公告)号:US20250057815A1
公开(公告)日:2025-02-20
申请号:US18822597
申请日:2024-09-03
Applicant: BRISTOL-MYERS SQUIBB COMPANY
Inventor: Peter Tai Wah Cheng , Robert F. Kaltenbach, III , Jun Li , Jun Shi , Yan Shi , Shiwei Tao , Hao Zhang , Suresh Dhanusu , Kumaravel Selvakumar , Ramesh Babu Reddigunta , Steven J. Walker , Lawrence J. Kennedy , James R. Corte , Tianan Fang , Sutjano Jusuf
IPC: A61K31/4192 , A61K31/27 , A61K31/41 , A61K31/454 , C07C62/10 , C07D249/06 , C07D401/04 , C07D401/14
Abstract: The present invention provides compounds of Formula (I): or stereoisomers, tautomers, pharmaceutically acceptable salts, solvates or prodrugs thereof, wherein all the variables are as defined herein. These compounds are selective LPA receptor inhibitors.
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公开(公告)号:US11261174B2
公开(公告)日:2022-03-01
申请号:US16954221
申请日:2018-12-18
Applicant: BRISTOL-MYERS SQUIBB COMPANY
Inventor: Peter Tai Wah Cheng , Jun Li , Yan Shi , Ying Wang , Hao Zhang , Lawrence J. Kennedy , Steven J. Walker , Ramesh Babu Reddigunta
IPC: C07D231/12 , C07D401/04 , C07D403/04 , A61K31/415 , A61K31/4427 , A61K31/496 , A61P43/00 , A61P17/02 , A61P35/00
Abstract: The present invention provides compounds of Formula (I) or a stereoisomer, tautomer, or pharmaceutically acceptable salt or solvate thereof, wherein all the variables are as defined herein. These compounds are selective LPA receptor inhibitors.
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公开(公告)号:US20210244711A1
公开(公告)日:2021-08-12
申请号:US17221859
申请日:2021-04-05
Applicant: BRISTOL-MYERS SQUIBB COMPANY
Inventor: PETER TAI WAH CHENG , Robert F. Kaltenbach, III , Jun Li , Jun Shi , Yan Shi , Shiwei Tao , Hao Zhang , Suresh Dhanusu , Kumaravel Selvakumar , Ramesh Babu Reddigunta , Steven J. Walker , Lawrence J. Kennedy , James R. Corte , Tianan Fang , Sutjano Jusuf
IPC: A61K31/4192 , C07D401/14 , C07D249/06 , A61K31/27 , A61K31/454 , C07D401/04
Abstract: The present invention provides compounds of Formula (I): or stereoisomers, tautomers, pharmaceutically acceptable salts, solvates or prodrugs thereof, wherein all the variables are as defined herein. These compounds are selective LPA receptor inhibitors.
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公开(公告)号:US20220249443A1
公开(公告)日:2022-08-11
申请号:US17718760
申请日:2022-04-12
Applicant: BRISTOL-MYERS SQUIBB COMPANY
Inventor: Peter Tai Wah Cheng , Robert F. Kaltenbach, III , Jun Li , Jun Shi , Yan Shi , Shiwei Tao , Hao Zhang , Suresh Dhanusu , Kumaravel Selvakumar , Ramesh Babu Reddigunta , Steven J. Walker , Lawrence J. Kennedy , James R. Corte , Tianan Fang , Sutjano Jusuf
IPC: A61K31/4192 , C07D401/14 , C07D249/06 , A61K31/27 , A61K31/454 , C07D401/04
Abstract: The present invention provides compounds of Formula (I): or stereoisomers, tautomers, pharmaceutically acceptable salts, solvates or prodrugs thereof, wherein all the variables are as defined herein. These compounds are selective LPA receptor inhibitors.
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公开(公告)号:US20200308148A1
公开(公告)日:2020-10-01
申请号:US16954221
申请日:2018-12-18
Applicant: BRISTOL-MYERS SQUIBB COMPANY
Inventor: Peter Tai Wah Cheng , Jun Li , Yan Shi , Ying Wang , Hao Zhang , Lawrence J. Kennedy , Steven J. Walker , Ramesh Babu Reddigunta
IPC: C07D403/04 , C07D401/04 , C07D231/12 , A61P35/00 , A61P17/02
Abstract: The present invention provides compounds of Formula (I) or a stereoisomer, tautomer, or pharmaceutically acceptable salt or solvate thereof, wherein all the variables are as defined herein. These compounds are selective LPA receptor inhibitors.
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公开(公告)号:US10576062B2
公开(公告)日:2020-03-03
申请号:US16038739
申请日:2018-07-18
Applicant: Bristol-Myers Squibb Company
Inventor: Peter Tai Wah Cheng , Robert F. Kaltenbach, III , Jun Li , Jun Shi , Yan Shi , Shiwei Tao , Hao Zhang , Suresh Dhanusu , Kumaravel Selvakumar , Ramesh Babu Reddigunta , Steven J. Walker , Lawrence J. Kennedy , James R. Corte , Tianan Fang , Sutjano Jusuf
IPC: C07D401/14 , C07D249/06 , A61K31/27 , A61K31/4192 , A61K31/454 , C07D401/04 , A61K31/41 , C07C62/10
Abstract: The present invention provides compounds of Formula (I): or stereoisomers, tautomers, pharmaceutically acceptable salts, solvates or prodrugs thereof, wherein all the variables are as defined herein. These compounds are selective LPA receptor inhibitors.
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