-
公开(公告)号:US20230046680A1
公开(公告)日:2023-02-16
申请号:US17603548
申请日:2020-04-08
发明人: Andreas TURBERG , Iring HEISLER , Joachim TELSER , Alexander ARLT , Peter JESCHKE , Hans-Georg SCHWARZ , Martin FUESSLEIN , Yolanda CANCHO GRANDE , Kerstin ILG , Ulrich EBBINGHAUS-KINTSCHER , Peter LOESEL , Marc LINKA , Arunas Jonas DAMIJONAITIS , Ingo LIMBERG
IPC分类号: C07D413/14 , C07D417/14 , A01N43/78 , A01N43/76 , A01N43/653 , A01N43/90 , C07D471/04 , C07D403/14
摘要: The present invention relates to novel heteroaryl-substituted aminoalkyl azole compounds of the general formula (I), in which the structural elements Y, Q1, Q2, R1, R2, R3 and R4 have the meaning given in the description, to formulations and compositions comprising such compounds and for their use in the control of animal pests including arthropods and insects in plant protection and to their use for control of ectoparasites on animals.
-
公开(公告)号:US20220274971A1
公开(公告)日:2022-09-01
申请号:US17630742
申请日:2020-07-27
发明人: Bernd ALIG , Walter HUEBSCH , Nils GRIEBENOW , Hans-Georg SCHWARZ , Wei ZHUANG , Daniel KULKE , Claudia BOEHM , Iring HEISLER , Isa Jana Irina JANSSEN , Kirsten BOERNGEN
IPC分类号: C07D413/14 , C07D405/12
摘要: The present invention covers new isoquinoline compounds of general formula (I): in which A, R1, R2, R3, R4, R5, R6, and Q are as defined herein, methods of preparing said compounds, intermediate compounds useful for preparing said compounds, pharmaceutical compositions and combinations comprising said compounds and the use of said compounds for manufacturing pharmaceutical compositions for the treatment, control and/or prevention of diseases, in particular of helminth infections, as a sole agent or in combination with other active ingredients.
-
公开(公告)号:US20200024264A1
公开(公告)日:2020-01-23
申请号:US16348797
申请日:2017-11-06
发明人: Walter HÜBSCH , Johannes KÖBBERLING , Adeline KÖHLER , Hans-Georg SCHWARZ , Daniel KULKE , Claudia WELZ , Thomas ILG , Kirsten BÖRNGEN , Wei ZHUANG , Nils GRIEBENOW , Claudia BÖHM , Niels LINDNER , Maike HINK , Ulrich GÖRGENS
IPC分类号: C07D405/14 , A61P33/10 , C07D405/12 , C07D413/14
摘要: The present invention covers new quinoline compounds of general formula (I) in which A, R1, R2, R3, R4, R5, R6, and Q are as defined herein, methods of preparing said compounds, intermediate compounds useful for preparing said compounds, pharmaceutical compositions and combinations comprising said compounds and the use of said compounds for manufacturing pharmaceutical compositions for the treatment, control and/or prevention of diseases, in particular of helminth infections, as a sole agent or in combination with other active ingredients.
-
公开(公告)号:US20230023326A1
公开(公告)日:2023-01-26
申请号:US17766151
申请日:2020-10-08
发明人: Andreas TURBERG , Iring HEISLER , Joachim TELSER , Alexander ARLT , Peter JESCHKE , Hans-Georg SCHWARZ , Martin FUESSLEIN , Yolanda CANCHO-GRANDE , Peter LOESEL , Ulrich EBBINGHAUS-KINTSCHER , Bing Ashley Liang ODOWD , Arunas DAMIJONAITIS , Steffen MUELLER , Jiakang MA
IPC分类号: C07D417/04 , C07D403/04 , C07D413/04
摘要: The present invention relates to novel heteroaryl-substituted pyrazine derivatives of the general formula (I), in which the structural elements R1, R2, R3, R4, R5 and R6 have the meaning given in the description, to formulations and compositions comprising such compounds and for their use in the control of animal pests including arthropods and insects in plant protection and to their use for control of ectoparasites on animals.
-
公开(公告)号:US20190071447A1
公开(公告)日:2019-03-07
申请号:US16093565
申请日:2017-04-10
发明人: Adeline KÖHLER , Claudia WELZ , Kirsten BÖRNGEN , Daniel KULKE , Thomas ILG , Johannes KÖBBERLING , Walter HÜBSCH , Hans-Georg SCHWARZ , Ulrich GÖRGENS , Ulrich EBBINGHAUS-KINTSCHER , Maike HINK , Dirk NENNSTIEL , Klaus RAMING , Martin ADAMCZEWSKI , Claudia BÖHM
IPC分类号: C07D487/04 , A61P33/10
摘要: The present invention covers Pyrazolopyrimidine compounds of general formula (I), in which n, o, X, Y, R, Q, R1, R2, R3 and R4 are as defined herein, methods of preparing said compounds, intermediate compounds useful for preparing said compounds, pharmaceutical compositions and combinations comprising said compounds and the use of said compounds for manufacturing pharmaceutical compositions for the treatment, control and/or prevention of diseases, in particular of helminth infections, as a sole agent or in combination with other active ingredients.
-
公开(公告)号:US20170144988A1
公开(公告)日:2017-05-25
申请号:US15325665
申请日:2015-07-13
发明人: Werner HALLENBACH , Hans-Georg SCHWARZ , Ulrich GOERGENS , Kerstin ILG , Andreas TURBERG , Sebastian HORSTMANN , Adeline KOEHLER
IPC分类号: C07D401/04 , A01N43/647
CPC分类号: C07D401/04 , A01N43/647
摘要: The invention relates to novel aryltriazolylpyridines of the general formula (I). Also described are processes for preparing the compounds of the formula (I). The compounds according to the invention are especially suitable for controlling insects and arachnids in agriculture, and ectoparasites in veterinary medicine.
-
公开(公告)号:US20160326140A1
公开(公告)日:2016-11-10
申请号:US15109630
申请日:2014-12-30
发明人: Hans-Georg SCHWARZ , Michael MAUE , Kerstin ILG , Ulrich GÖRGENS , Andreas TURBERG , Sebastian HORSTMANN , Johannes KÖBBERLING , Niels LINDNER
IPC分类号: C07D403/04 , A01N43/56 , C07D409/14 , A01N43/90 , C07D413/14 , A01N43/76 , C07D407/14 , C07D487/04 , C07D401/14 , C07D403/14
CPC分类号: C07D403/04 , A01N43/56 , A01N43/76 , A01N43/90 , C07D231/38 , C07D401/14 , C07D403/14 , C07D407/14 , C07D409/14 , C07D413/14 , C07D487/04
摘要: The invention comprises, inter alia, pyrazolylheteroarylamides of the general formula (I) in which the A1-A4, T, W, Q, R1 and Z1-Z3 radicals are each as defined in the description. Also described are processes for preparing the compounds of the formula (I). The inventive compounds are especially suitable for controlling insects, arachnids and nematodes in agriculture and ectoparasites in veterinary medicine.
摘要翻译: 其中A1-A4,T,W,Q,R1和Z1-Z3基团各自如说明书中所定义。 还描述了制备式(I)化合物的方法。 本发明化合物特别适用于控制农药中的昆虫,蜘蛛和线虫,并在兽医学中控制外寄生虫。
-
公开(公告)号:US20160007604A1
公开(公告)日:2016-01-14
申请号:US14772471
申请日:2014-02-27
发明人: Michael MAUE , Anne DECOR , Thomas BRETSCHNEIDER , Julia Johanna HAHN , Werner HALLENBACH , Reiner FISCHER , Hans-Georg SCHWARZ , Ulrich GÖRGENS , Kerstin ILG , Klaus RAMING , Johannes KÖBBERLING , Walter HÜBSCH , Andreas TURBERG
IPC分类号: A01N43/56 , C07D231/12
CPC分类号: A01N43/56 , A01N43/647 , A01N43/653 , C07D231/12 , C07D401/14 , C07D403/04 , C07D403/14
摘要: The invention relates inter alia to halogen-substituted compounds of the general formula (II) in which the radicals A1-A4, T, n, W, Q, R1 and Z1-Z3 have the meanings given in the description. Also described are processes for preparing the compounds of the formula (II). The compounds according to the invention are particularly suitable for controlling insects, arachnids and nematodes in agriculture and ectoparasites in veterinary medicine.
摘要翻译: 本发明尤其涉及通式(II)的卤素取代的化合物,其中基团A1-A4,T,n,W,Q,R1和Z1-Z3具有在说明书中给出的含义。 还描述了制备式(II)化合物的方法。 根据本发明的化合物特别适用于在兽医学中控制农业和外寄生虫中的昆虫,蜘蛛和线虫。
-
公开(公告)号:US20230242513A1
公开(公告)日:2023-08-03
申请号:US18002928
申请日:2021-06-23
发明人: Iring HEISLER , Andreas TURBERG , Joachim TELSER , Alexander ARLT , Peter JESCHKE , Hans-Georg SCHWARZ , Martin FUESSLEIN , Yolanda CANCHO-GRANDE , Peter LOESEL , Ulrich EBBINGHAUS-KINTSCHER , Bing Ashley Liang O'DOWD , Melanie ARMENAT
IPC分类号: C07D403/04 , C07D403/14 , C07D413/14 , A01N43/647 , A01N43/653 , A01N43/84 , A01P7/04 , A61K31/497 , A61K31/5377 , A61P33/14 , A01N47/02
CPC分类号: C07D403/04 , C07D403/14 , C07D413/14 , A01N43/647 , A01N43/653 , A01N43/84 , A01P7/04 , A61K31/497 , A61K31/5377 , A61P33/14 , A01N47/02
摘要: The present invention relates to novel heteroaryl-substituted pyrazine derivatives of the general formula (I), in which the structural elements R1, R2, R3, R4, R5 and R6 have the meaning given in the description, to formulations and compositions comprising such compounds and for their use in the control of animal pests including arthropods and insects in plant protection and to their use for control of ectoparasites on animals.
-
公开(公告)号:US20230141809A1
公开(公告)日:2023-05-11
申请号:US18063766
申请日:2022-12-09
发明人: Walter HUEBSCH , Nils GRIEBENOW , Hans-Georg SCHWARZ , Daniel KULKE , Claudia BOEHM , Kirsten BOERNGEN , Bernd ALIG , Wei ZHUANG , Iring HEISLER , Thomas ILG , Johannes KOEBBERLING , Adeline KOEHLER , Niels LINDNER , Ulrich GOERGENS , Claudia WELZ , Maike HINK
IPC分类号: C07D405/14 , C07D405/12 , A61P33/10
CPC分类号: C07D405/14 , C07D405/12 , A61P33/10
摘要: The present invention covers new quinoline compounds of general formula (I):
in which A, R1, R2, R3, R4, R5, R6, and Q are as defined herein, methods of preparing said compounds, intermediate compounds useful for preparing said compounds, pharmaceutical compositions and combinations comprising said compounds and the use of said compounds for manufacturing pharmaceutical compositions for the treatment, control and/or prevention of diseases, in particular of helminth infections, as a sole agent or in combination with other active ingredients.
-
-
-
-
-
-
-
-
-