公开(公告)号：US11825838B2

公开(公告)日：2023-11-28

申请号：US16498674

申请日：2018-03-26

Applicant: Bayer CropScience Aktiengesellschaft

Inventor： Tobias Harschneck ,  Alexander Arlt ,  Robert Velten ,  Michael Maue ,  Kerstin Ilg ,  Werner Hallenbach ,  Ulrich Goergens ,  Sebastian Horstmann ,  Peter Loesel ,  Andreas Turberg

IPC: C07D417/04 ,  C07D409/04 ,  C07D403/04 ,  A01N43/56 ,  A01N43/78 ,  A01N33/26

CPC classification number: A01N33/26 ,  A01N43/56 ,  A01N43/78 ,  C07D403/04 ,  C07D409/04 ,  C07D417/04

Abstract: The invention relates, inter alia, to compounds of general formula (I). The invention also relates to methods for synthesizing the compounds of formula (I). The compounds according to the invention are in particular suitable for controlling insects, arachnids and nematodes in agricultural applications and for controlling ectoparasites in veterinary medicine.

公开(公告)号：US11072609B2

公开(公告)日：2021-07-27

申请号：US16481124

申请日：2018-02-05

Applicant: Bayer Aktiengesellschaft ,  Bayer CropScience Aktiengesellschaft

Inventor： Marc Mosrin ,  Ruediger Fischer ,  Dominik Hager ,  Laura Hoffmeister ,  Nina Kausch-Busies ,  David Wilcke ,  Matthieu Willot ,  Kerstin Ilg

IPC: C07D471/04

Abstract: The present invention relates to a method for preparing halogenated imidazopyridine derivatives of the formula (II) proceeding from compounds of the formula (I) via intermediates of the formula (IVa) or (IVb) in which the radicals Q, Z, R1, R3, R4, Rc, A1 and A2 have the definitions stated. The invention further relates to such halogenated imidazopyridine derivatives, and also intermediates and the reaction products of compounds of the formula (II) to give compounds of the formula (III) in which the specified structural elements have the definitions stated.

公开(公告)号：US11058115B2

公开(公告)日：2021-07-13

申请号：US16476358

申请日：2018-01-03

Applicant: Bayer Aktiengesellschaft ,  Bayer CropScience Aktiengesellschaft

Inventor： David Wilcke ,  Ruediger Fischer ,  Dominik Hager ,  Laura Hoffmeister ,  Nina Kausch-Busies ,  Marc Mosrin ,  Matthieu Willot ,  Kerstin Ilg ,  Ulrich Goergens ,  Andreas Turberg

IPC: C07D487/04 ,  A01N43/90 ,  C07D471/04

Abstract: The invention relates to novel compounds of the formula (I) in which X, R1, R2, R3 and n have the definitions given above, to the use thereof as acaricides and/or insecticides for control of animal pests and to processes and intermediates for preparation thereof.

公开(公告)号：US10986840B2

公开(公告)日：2021-04-27

申请号：US16590006

申请日：2019-10-01

Applicant: Bayer CropScience Aktiengesellschaft

Inventor： Ruediger Fischer ,  David Wilcke ,  Nina Kausch-Busies ,  Dominik Hager ,  Kerstin Ilg ,  Laura Hoffmeister ,  Matthieu Willot ,  Daniela Portz ,  Ulrich Goergens ,  Andreas Turberg

IPC: C07D235/18 ,  C07D401/04 ,  C07D403/10 ,  C07D409/10 ,  A01N43/90 ,  C07D401/14 ,  C07D471/04 ,  C07D487/04 ,  C07D498/04 ,  A01N43/56 ,  C07D409/14 ,  A01N43/54 ,  A01N43/52 ,  C07D401/12 ,  C07D491/056

Abstract: The invention relates to novel compounds of the formula (I) in welcher R1, R2, R3, A1, X and n have the meanings given above, to their use as acaricides and/or insecticides for controlling animal pests and to processes and intermediates for their preparation.

公开(公告)号：US10765116B2

公开(公告)日：2020-09-08

申请号：US16463327

申请日：2017-11-22

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT ,  BAYER AKTIENGESELLSCHAFT

Inventor： Nina Kausch-Busies ,  Rüdiger Fischer ,  Laura Hoffmeister ,  David Wilcke ,  Dominik Hager ,  Matthieu Willot ,  Marc Mosrin ,  Kerstin Ilg ,  Ulrich Görgens ,  Andreas Turberg

IPC: C07D471/04 ,  A01N43/90 ,  C07D519/00

Abstract: The invention relates to compounds of the formula (Ia) or (Ib), in which Aa, Ab, Ac, Ad, R1, R10 R11, R12, R13, R14, R15, R16, R17, Q, R4, R5, R6 and have the meanings indicated in the claims, and to agrochemical formulations containing the compounds according to formula (Ia) or (Ib) for use as acaricides and/or insecticides for combating animal pests, primarily arthropods and in particular insects and arachnids. 2-[3-(alkylsulfonyl)-2H-indazol-2-yl]-3H-imidazo[4,5-b]pyridine derivatives and similar compounds are particularly preferable.

公开(公告)号：US10544124B2

公开(公告)日：2020-01-28

申请号：US16076786

申请日：2017-02-06

Applicant: Bayer CropScience Aktiengesellschaft

Inventor： Johannes-Rudolf Jansen ,  Markus Heil ,  Reiner Fischer ,  David Wilcke ,  Matthieu Willot ,  Kerstin Ilg ,  Sascha Eilmus ,  Peter Lösel ,  Wolfram Andersch

IPC: C07D401/12 ,  C07D403/12 ,  C07D413/14 ,  C07D403/14 ,  C07D407/14 ,  C07D409/14 ,  A01N43/50 ,  A01N43/54 ,  A01N43/647 ,  A01N43/80 ,  A01N43/84 ,  C07D401/14 ,  C07D405/14

Abstract: The present invention relates to compounds of the general formula (I) in which Q, V, T, W, X, Y and A have the meanings given in the description—and to their use for controlling animal pests.

公开(公告)号：US10364243B2

公开(公告)日：2019-07-30

申请号：US15119124

申请日：2015-02-05

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Rüdiger Fischer ,  Bernd Alig ,  Kerstin Ilg ,  Olga Malsam ,  Ulrich Görgens ,  Andreas Turberg ,  Jun Li ,  Sergey Zhersh ,  Alexander Arlt

IPC: C07D471/04 ,  A01N43/90 ,  C07D213/73 ,  C07D213/74 ,  C07D473/40 ,  C07D498/04 ,  C07D487/04

Abstract: The invention relates to novel compounds of the formula (I) in which the R1, R2a, R2b, R3, A1, A2, A3, A4, A5 and n radicals are each as defined above, to the use thereof as acaricides and/or insecticides for controlling animal pests and to processes and intermediates for preparation thereof.

公开(公告)号：US10239859B2

公开(公告)日：2019-03-26

申请号：US15742369

申请日：2016-07-04

Applicant: Bayer CropScience Aktiengesellschaft

Inventor： Peter Jeschke ,  Oliver Gutbrod ,  Reiner Fischer ,  Elke Hellwege ,  Peter Loesel ,  Olga Malsam ,  Sascha Eilmus ,  Kerstin Ilg ,  Daniela Portz ,  Ulrich Goergens ,  Anton Lishchynskyi

IPC: C07D401/04 ,  C07D213/74 ,  C07D417/04 ,  A01N43/40 ,  C07D401/14

Abstract: The present application relates to novel heterocyclic compounds, to processes and intermediates for the preparation thereof, and their use for controlling animal pests.

公开(公告)号：US09981940B2

公开(公告)日：2018-05-29

申请号：US14899259

申请日：2014-06-16

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Bernd Alig ,  Silvia Cerezo-Galvez ,  Reiner Fischer ,  Adeline Koehler ,  Julia Johanna Hahn ,  Angela Becker ,  Kerstin Ilg ,  Arnd Voerste ,  Daniela Portz

IPC: C07D207/273 ,  C07D207/38 ,  C07D207/408 ,  C07D249/12 ,  C07D257/04 ,  C07D271/113 ,  C07D277/40 ,  C07D277/42 ,  C07D233/70 ,  C07D401/04 ,  C07D405/04 ,  A01N25/00 ,  A01N43/36 ,  A01N43/50 ,  A01N43/653 ,  A01N43/713 ,  A01N43/78 ,  A01N43/82

CPC classification number: C07D401/04 ,  A01N25/00 ,  A01N43/36 ,  A01N43/50 ,  A01N43/653 ,  A01N43/713 ,  A01N43/78 ,  A01N43/82 ,  C07D207/273 ,  C07D207/38 ,  C07D207/408 ,  C07D233/70 ,  C07D249/12 ,  C07D257/04 ,  C07D271/113 ,  C07D277/40 ,  C07D277/42 ,  C07D405/04

Abstract: The present invention relates to aryl sulphide and aryl sulphoxide derivatives, to the use thereof as acaricides and insecticides for controlling animal pests and to processes and intermediates for preparation thereof. The aryl sulphide and aryl sulphoxide derivatives have the general structure (I) in which the respective radicals are as defined in the description.

公开(公告)号：US09936700B2

公开(公告)日：2018-04-10

申请号：US15029533

申请日：2014-10-20

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Bernd Alig ,  Joerg Greul ,  Ruediger Fischer ,  Hans-Georg Schwarz ,  Niklas Tim Bretschneider ,  Uta Bretschneider ,  Reiner Fischer ,  Daniela Portz ,  Olga Malsam ,  Peter Loesel ,  Kerstin Ilg ,  Angela Becker ,  Ulrich Goergens ,  Stefan Herrmann ,  Claudia Welz

IPC: A01N43/60 ,  C07D401/04 ,  C07D403/04 ,  C07D409/04 ,  C07D241/40 ,  C07D491/04 ,  A01N43/90 ,  C07D213/50 ,  C07D491/056

CPC classification number: A01N43/60 ,  A01N43/90 ,  C07D213/50 ,  C07D241/40 ,  C07D401/04 ,  C07D403/04 ,  C07D409/04 ,  C07D491/04 ,  C07D491/056

Abstract: The invention relates to novel compounds of the formula (I) in which R1, R2, R3, R4, R5, R6, Y1 and Y2 have the meanings given above, to a plurality of processes and intermediates for their preparation and to their use as acaricides and/or insecticides for controlling animal pests. The compounds of the formula (I) are also suitable as nematicides for plant-damaging pests and/or anthelminthics for endoparasites in humans and animals.