专利检索 ap:("Gerd Schubert" OR "Sven Ring" OR "Guenther Kaufmann" OR "Walter Elger" OR "Birgit Schneider") AND inv:"Birgit Schneider" 第 1 页

1.

发明授权
S-substitute 11&bgr;-benzaldoxime-estra-4, 9-diene-carbonic acid thiolesters, method for the production thereof and pharmaceutical preparations containing these compounds 失效
标题翻译： S-替代物11beta-benzaldoxime-estra-4,9-二烯 - 碳酸硫醇酯，其制备方法和含有这些化合物的药物制剂

公开(公告)号：US06365582B1

公开(公告)日：2002-04-02

申请号：US09622803

申请日：2000-08-22

申请人： Gerd Schubert , Sven Ring , Guenther Kaufmann , Walter Elger , Birgit Schneider

发明人： Gerd Schubert , Sven Ring , Guenther Kaufmann , Walter Elger , Birgit Schneider

IPC分类号： A61K3156

CPC分类号： C07J41/0083 , C07J43/006

摘要： Thiol esters of S-substituted 11&bgr;-benzaldoxime-estra-4,9-dien-carboxylic acids of the formula I their pharmaceutically acceptable salts, a method for their synthesis and pharmaceutical preparations containing these compounds are described. These compounds bind to progesterone receptors and have distinctly reduced anti-glucocorticoid action.

摘要翻译： 描述下式的S-取代的11β-苯甲醛肟 - 雌-4,9-二烯 - 羧酸的硫醇酯，其药学上可接受的盐，它们的合成方法和含有这些化合物的药物制剂。这些化合物结合孕酮受体并具有显着降低的抗糖皮质激素作用。