公开(公告)号：US4931455A

公开(公告)日：1990-06-05

申请号：US289626

申请日：1988-12-22

申请人： Hirosuke Yoshioka ,  Tokio Obata ,  Katsutoshi Fujii ,  Haruo Yoshiya ,  Kiyoshi Tsutsumiuchi ,  Shoji Shikita

发明人： Hirosuke Yoshioka ,  Tokio Obata ,  Katsutoshi Fujii ,  Haruo Yoshiya ,  Kiyoshi Tsutsumiuchi ,  Shoji Shikita

IPC分类号： A01N43/54 ,  A01N47/06 ,  A01N47/12 ,  A01N47/16 ,  A01N47/20 ,  A01N47/28 ,  A01N49/00 ,  A01N53/00 ,  C07D239/42 ,  C07D403/12 ,  C07D405/12 ,  C07D413/12

CPC分类号： C07D239/42 ,  A01N43/54 ,  A01N47/06 ,  A01N47/12 ,  A01N47/16 ,  A01N47/20 ,  A01N47/28 ,  A01N49/00 ,  A01N53/00 ,  C07D403/12 ,  C07D405/12 ,  C07D413/12

摘要： There are described an alkylaminopyrimidine derivative represented by the formula: ##STR1## wherein R.sub.1 represents a hydrogen atom, a halogen atom, a lower alkyl group, a cycloalkyl group having 3 to 6 carbon atoms, a halogenated lower alkyl group or a substituted or unsubstituted phenyl group; R.sub.2 represents a halogen atom; R.sub.3 represents a hydrogen atom, a lower alkyl group or a cycloalkyl group having 3 to 6 carbon atoms; and R.sub.4 represents a straight or branched alkyl group having 1 to 20 carbon atoms which may have substituents,or an acid addition salt thereof, a process for preparing the same and an insecticide, an acaricide or a fungicide containing the compound as an active ingredient.

公开(公告)号：US4895849A

公开(公告)日：1990-01-23

申请号：US105403

申请日：1987-10-05

申请人： Hirosuke Yoshioka ,  Tokio Obata ,  Katsutoshi Fujii ,  Kiyoshi Tsutsumiuchi ,  Haruo Yoshiya

发明人： Hirosuke Yoshioka ,  Tokio Obata ,  Katsutoshi Fujii ,  Kiyoshi Tsutsumiuchi ,  Haruo Yoshiya

IPC分类号： A01N43/54 ,  A01N43/58 ,  A01N43/66 ,  A01N43/78 ,  A01N49/00 ,  A01N55/00 ,  C07D239/42 ,  C07D239/56 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D417/12 ,  C07F7/08

CPC分类号： C07D239/42 ,  A01N43/54 ,  A01N43/58 ,  A01N43/66 ,  A01N43/78 ,  A01N49/00 ,  A01N55/00 ,  C07D239/56 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D417/12 ,  C07F7/0812

摘要： There are disclosed a compound represented by the formula: ##STR1## wherein R.sub.1 represents a hydrogen atom or a lower alkyl group; R.sub.2 and R.sub.3 each independently represent a halogen atom or a lower alkyl group; R.sub.4 represents a hydrogen atom, a halogen atom or a lower alkyl group; n represents an integer of 1 or 2; Q represents a phenyl group or a heterocyclic group; a substituted or unsubstituted alkyl group; an allyl group; a geranyl group; a farnesyl group; a cycloalkylmethyl group; a substituted ethyl group; a glycidyl group; an acetonyl group; a substituted dioxoranyl group; a 2,2-diethoxyethyl group, a 1-ethoxycarbonylethyl group, a trimethylsilylmethyl group or a 1-pyridylethyl group; A represents a lower alkylene group; and B represents a direct bond, an oxygen atom, a sulfur atom, a straight or branched lower alkylene group or a lower alkyleneoxy group;or an acid addition salt thereof, a process for producing the same, and an insecticide, an acaricide and a fungicide containing the derivative as the active ingredient.

摘要翻译： 公开了下式表示的化合物：其中R 1表示氢原子或低级烷基; R2和R3各自独立地表示卤素原子或低级烷基; R4表示氢原子，卤素原子或低级烷基; n表示1或2的整数; Q表示苯基或杂环基; 取代或未取代的烷基; 烯丙基; 香叶基 法呢基 环烷基甲基; 取代的乙基; 缩水甘油基; 丙酮基; 取代的二氧杂环戊烷基; 2,2-二乙氧基乙基，1-乙氧基羰基乙基，三甲基甲硅烷基甲基或1-吡啶基乙基; A表示低级亚烷基; B表示直接键，氧原子，硫原子，直链或支链低级亚烷基或低级亚烷基氧基; 或其酸加成盐，其制备方法，以及含有该衍生物作为活性成分的杀虫剂，杀螨剂和杀真菌剂。

公开(公告)号：US4985426A

公开(公告)日：1991-01-15

申请号：US435937

申请日：1989-11-13

申请人： Hirosuke Yoshioka ,  Tokio Obata ,  Katsutoshi Fujii ,  Kiyoshi Tsutsumiuchi ,  Haruo Yoshiya

发明人： Hirosuke Yoshioka ,  Tokio Obata ,  Katsutoshi Fujii ,  Kiyoshi Tsutsumiuchi ,  Haruo Yoshiya

IPC分类号： A01N43/54 ,  A01N43/58 ,  A01N43/66 ,  A01N43/78 ,  A01N49/00 ,  A01N55/00 ,  C07D239/42 ,  C07D239/56 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D417/12 ,  C07F7/08

CPC分类号： C07D239/42 ,  A01N43/54 ,  A01N43/58 ,  A01N43/66 ,  A01N43/78 ,  A01N49/00 ,  A01N55/00 ,  C07D239/56 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D417/12 ,  C07F7/0812

摘要： There is disclosed a compound represented by the formula: ##STR1## wherein R.sub.1 represents a hydrogen atom or a lower alkyl group; R.sub.2 and R.sub.3 each independently represent a halogen atom or a lower alkyl group; R.sub.4 represents a hydrogen atom, a halogen atom or a lower alkyl group; n represents an integer of 1 or 2; Q represents a phenyl group or a heterocyclic group; a substituted or unsubstituted alkyl group; an allyl group, a geranyl group; a farnesyl group; a cycloalkylmethyl group; a substituted ethyl group; a glycidyl group; an acetonyl group; a substituted dioxoranyl group; a 2,2-diethoxyethyl group, a 1-ethoxycarbonylethyl group, a trimethylsilylmethyl group or a 1-pyridylethyl group; A represents a lower alkylene group; and B represents a direct bond, an oxygen atom, a sulfur atom, a straight or branched lower alkylene group or a lower alkyleneoxy group;or an acid addition salt thereof, a process for producing the same, and an insecticide, an acaricide and a fungicide containing the derivative as the active ingredient.

公开(公告)号：US5081144A

公开(公告)日：1992-01-14

申请号：US503684

申请日：1990-04-02

申请人： Tokio Obata ,  Katsutoshi Fujii ,  Yasuhisa Fukuda ,  Kiyoshi Tsutsumiuchi

发明人： Tokio Obata ,  Katsutoshi Fujii ,  Yasuhisa Fukuda ,  Kiyoshi Tsutsumiuchi

IPC分类号： C07D231/22

CPC分类号： C07D231/22

摘要： A compound represented by the formula: ##STR1## wherein R.sub.1 represents hydrogen atom, a halogen atom or an alkyl group having 1 to 5 carbon atoms; R.sub.2 represents hydrogen atom or an alkyl group having 1 to 5 carbon atoms; R.sub.3 represents an alkyl group having 1 to 8 carbon atoms, an alkenyl group having 3 to 5 carbon atoms, an alkynyl group having 3 to 5 carbon atoms or an aralkyl group which may be also substituted; R.sub.4 represents hydrogen atom or an alkyl group having 1 to 5 carbon atoms; n represents an integer of 4 and when R.sub.2 is an alkyl group, n represents an integer of 1 to 3; A represents an alkylene group having 1 to 5 carbon atoms; and X represents an oxygen atom or a sulfur atom and an insecticide, acaricide or fungicide comprising a compound of the formula (I) as the active ingredient.

公开(公告)号：US5280025A

公开(公告)日：1994-01-18

申请号：US977753

申请日：1992-11-17

申请人： Tokio Obata ,  Katsutoshi Fujii ,  Kiyoshi Tsutsumiuchi ,  Yasushi Nakamoto

发明人： Tokio Obata ,  Katsutoshi Fujii ,  Kiyoshi Tsutsumiuchi ,  Yasushi Nakamoto

IPC分类号： A01N43/54 ,  C07D239/42

CPC分类号： C07D239/42 ,  A01N43/54

摘要： Disclosed are an aralkylaminopyrimidine compound represented by the following formula: ##STR1## wherein R.sup.1 represents a halogen atom, a lower acyloxy group, a hydroxyl group, a lower alkoxy group or a lower alkylthio group; R.sup.2 represents a lower alkyl group, a hydrogen atom or a cycloalkyl group; R.sup.3 may be the same or different and represents a lower haloalkoxy group, a hydrogen atom, a lower alkyl group, a lower alkoxy group, a halogen atom, a lower alkylthio group, a nitro group, a lower haloalkyl group, a lower alkylsulfinyl group, a lower alkylsulfonyl group, a lower haloalkylthio group or a hydroxyl group; a carbon atom to which * is attached represents an asymmetric carbon atom provided that the case where R.sup.2 is a hydrogen atom is excluded; and n represents an integer of 1 to 5.a method for preparing the same and a chemical for controlling noxious organisms which contains the same as an active ingredient.

摘要翻译： 公开了由下式表示的芳烷基氨基嘧啶化合物：（*化学结构*）（I）其中R1表示卤素原子，低级酰氧基，羟基，低级烷氧基或低级烷硫基; R2表示低级烷基，氢原子或环烷基; R3可以相同或不同，表示低级卤代烷氧基，氢原子，低级烷基，低级烷氧基，卤素原子，低级烷硫基，硝基，低级卤代烷基，低级烷基亚磺酰基 ，低级烷基磺酰基，低级卤代烷硫基或羟基; 只要不排除R2为氢原子的情况，则与其相连的碳原子表示不对称碳原子; n表示1〜5的整数。其制备方法和用于控制含有活性成分的有害生物的化学物质。

公开(公告)号：US5221685A

公开(公告)日：1993-06-22

申请号：US828110

申请日：1992-01-30

申请人： Tokio Obata ,  Katsutoshi Fujii ,  Yasuhisa Fukuda ,  Kiyoshi Tsutsumiuchi ,  Yoshinori Yamanaka

发明人： Tokio Obata ,  Katsutoshi Fujii ,  Yasuhisa Fukuda ,  Kiyoshi Tsutsumiuchi ,  Yoshinori Yamanaka

IPC分类号： C07D277/46 ,  C07D277/48 ,  C07D417/12

CPC分类号： C07D417/12 ,  C07D277/46 ,  C07D277/48

摘要： Disclosed are a thiazoline compound represented by the following formula (I): ##STR1## wherein R represents hydrogen atom or a lower alkyl group, X represents oxygen atom or sulfur atom, and Q represents Ar (where Ar represents a substituted or unsubstituted phenyl group or a substituted or unsubstituted naphthyl group) or ##STR2## (where Y represents a halogen atom, a lower alkyl group, a lower alkoxy group, a lower haloalkyl group, a lower haloalkoxy group, nitro group, acetyl group or cyano group and n represents an integer of 0 to 5),a process for preparing the same and a chemical for controlling noxious organisms containing the same as an active ingredient.

公开(公告)号：US5124333A

公开(公告)日：1992-06-23

申请号：US558798

申请日：1990-07-26

申请人： Tokio Obata ,  Katsutoshi Fujii ,  Isamu Narita ,  Shoji Shikita

发明人： Tokio Obata ,  Katsutoshi Fujii ,  Isamu Narita ,  Shoji Shikita

IPC分类号： A01N43/54 ,  A01N43/90 ,  A01N47/38 ,  C07D239/42 ,  C07D239/70 ,  C07D239/94 ,  C07D403/12 ,  C07D491/048 ,  C07D495/04

CPC分类号： C07D239/42 ,  A01N43/54 ,  A01N43/90 ,  A01N47/38 ,  C07D239/70 ,  C07D239/94 ,  C07D403/12 ,  C07D495/04

摘要： An aminopyrimidine compound of the formula: ##STR1## wherein R.sup.1 represents a hydrogen atom, an alkyl group, a cycloalkyl group or a halogen atom;R.sup.2 and R.sup.3 each represent an alkyl group or a halogen atom, or R.sup.2 and R.sup.3 represent a saturated or unsaturated 5- or 6-membered ring;R.sup.4 represents a hydrogen atom or --CONR.sup.6 R.sup.7, where R.sup.6 and R.sup.7 represent an unsaturated 5-membered ring; andR.sup.5 represents ##STR2## where m represents an integer of 1 to 10; m' represents an integer of 1 to 15;n represents an integer of 0, 1 or 2;R.sup.8 represents a hydrogen atom, an alkyl group or a cycloalkyl group;R.sup.9 represents an alkyl group, an alkenyl group, an alkynyl group, a substituted or unsubstituted phenyl group, a substituted or unsubstituted aralkyl group or an alkyl group,and acid addition salts thereof. Such compound is useful for combatting insects, acarids, nematodes and fungus.

公开(公告)号：US5073558A

公开(公告)日：1991-12-17

申请号：US427818

申请日：1989-10-26

申请人： Tokio Obata ,  Katsutoshi Fujii ,  Isamu Narita ,  Shoji Shikita

发明人： Tokio Obata ,  Katsutoshi Fujii ,  Isamu Narita ,  Shoji Shikita

IPC分类号： A01N47/36 ,  A01N47/38 ,  C07D239/42 ,  C07D239/94 ,  C07D403/12 ,  C07D405/12 ,  C07D405/14 ,  C07D413/12 ,  C07D417/12 ,  C07D491/04 ,  C07D491/048 ,  C07D495/04 ,  C07D521/00

CPC分类号： C07D239/42 ,  A01N47/36 ,  A01N47/38 ,  C07D231/12 ,  C07D233/56 ,  C07D249/08 ,  C07D403/12 ,  C07D417/12 ,  C07D491/04 ,  C07D495/04

摘要： Disclosed are an aminopyrimidine compound or an acid addition salt thereof represented by the formula: ##STR1## wherein R1, R2, R3, R4, R5 and Y have the same meanings defined in the specification;a process for preparing the compound and insecticide or bactericide containing the compound.

公开(公告)号：US5252596A

公开(公告)日：1993-10-12

申请号：US903940

申请日：1992-06-26

申请人： Tokio Obata ,  Katsutoshi Fujii ,  Akira Ooka ,  Shoji Shikita

发明人： Tokio Obata ,  Katsutoshi Fujii ,  Akira Ooka ,  Shoji Shikita

IPC分类号： A01N43/56 ,  C07D231/54 ,  A61K43/56

CPC分类号： C07D231/54

摘要： Disclosed are a novel phenoxyalkylamine compound represented by the following formula: ##STR1## wherein R.sup.1 represents a lower alkyl group or a lower haloalkyl group; R.sup.2 represents hydrogen atom or a lower alkyl group; R.sup.3 represents hydrogen atom, a lower alkyl group or a halogen atom; R.sup.4 represents a lower alkenyl group or --S--O--R.sup.6 where A represents a lower alkylene group and R.sup.6 represents a lower alkyl group, a lower alkenyl group or a lower alkynyl group; R.sup.5 represents hydrogen atom, a lower alkyl group or a halogen atom,a method for preparing the same and a chemical for controlling noxious organisms which contains the same as an active ingredient.

公开(公告)号：US5039692A

公开(公告)日：1991-08-13

申请号：US539965

申请日：1990-06-15

申请人： Tokio Obata ,  Katsutoshi Fujii ,  Toshinobu Tanaka ,  Akira Ooka ,  Shoji Shikita

发明人： Tokio Obata ,  Katsutoshi Fujii ,  Toshinobu Tanaka ,  Akira Ooka ,  Shoji Shikita

IPC分类号： C07D233/64 ,  A01N43/56 ,  C07D231/14 ,  C07D231/16 ,  C07D233/68

CPC分类号： C07D231/16 ,  C07D231/14

摘要： There are disclosed a phenoxyalkylamine derivative represented by the formula: ##STR1## wherein A.sup.1 represents an alkylene group having 2 to 5 carbon atoms, R.sup.1 and R.sup.2 each represent hydrogen atom or a lower alkyl group having 1 to 5 carbon atoms, R.sup.3, R.sup.4 and R.sup.5 each represent hydrogen atom, an alkyl group having 1 to 5 carbon atoms or a halogen atom, R.sup.6 represents hydrogen atom, an alkyl group having 1 to 5 carbon atoms, an alkenyl group having 3 to 5 carbon atoms or a group --A.sup.2 --X--R.sup.7, A.sup.2 represents an alkylene group having 1 to 5 carbon atoms, X represents oxygen atom or sulfur atom, R.sup.7 represents a lower alkyl group having 1 to 5 carbon atoms, an alkenyl group having 3 to 5 carbon atoms, an alkynyl group having 3 to 5 carbon atoms or a substituted or unsubstituted aralkyl group,and an insecticide, an acaricide and a fungicide for agriculture and horticulture, which comprises a carrier and the above phenoxyalkylamine derivative represented as the active ingredient.