公开(公告)号：US5252596A

公开(公告)日：1993-10-12

申请号：US903940

申请日：1992-06-26

申请人： Tokio Obata ,  Katsutoshi Fujii ,  Akira Ooka ,  Shoji Shikita

发明人： Tokio Obata ,  Katsutoshi Fujii ,  Akira Ooka ,  Shoji Shikita

IPC分类号： A01N43/56 ,  C07D231/54 ,  A61K43/56

CPC分类号： C07D231/54

摘要： Disclosed are a novel phenoxyalkylamine compound represented by the following formula: ##STR1## wherein R.sup.1 represents a lower alkyl group or a lower haloalkyl group; R.sup.2 represents hydrogen atom or a lower alkyl group; R.sup.3 represents hydrogen atom, a lower alkyl group or a halogen atom; R.sup.4 represents a lower alkenyl group or --S--O--R.sup.6 where A represents a lower alkylene group and R.sup.6 represents a lower alkyl group, a lower alkenyl group or a lower alkynyl group; R.sup.5 represents hydrogen atom, a lower alkyl group or a halogen atom,a method for preparing the same and a chemical for controlling noxious organisms which contains the same as an active ingredient.

公开(公告)号：US5039692A

公开(公告)日：1991-08-13

申请号：US539965

申请日：1990-06-15

申请人： Tokio Obata ,  Katsutoshi Fujii ,  Toshinobu Tanaka ,  Akira Ooka ,  Shoji Shikita

发明人： Tokio Obata ,  Katsutoshi Fujii ,  Toshinobu Tanaka ,  Akira Ooka ,  Shoji Shikita

IPC分类号： C07D233/64 ,  A01N43/56 ,  C07D231/14 ,  C07D231/16 ,  C07D233/68

CPC分类号： C07D231/16 ,  C07D231/14

摘要： There are disclosed a phenoxyalkylamine derivative represented by the formula: ##STR1## wherein A.sup.1 represents an alkylene group having 2 to 5 carbon atoms, R.sup.1 and R.sup.2 each represent hydrogen atom or a lower alkyl group having 1 to 5 carbon atoms, R.sup.3, R.sup.4 and R.sup.5 each represent hydrogen atom, an alkyl group having 1 to 5 carbon atoms or a halogen atom, R.sup.6 represents hydrogen atom, an alkyl group having 1 to 5 carbon atoms, an alkenyl group having 3 to 5 carbon atoms or a group --A.sup.2 --X--R.sup.7, A.sup.2 represents an alkylene group having 1 to 5 carbon atoms, X represents oxygen atom or sulfur atom, R.sup.7 represents a lower alkyl group having 1 to 5 carbon atoms, an alkenyl group having 3 to 5 carbon atoms, an alkynyl group having 3 to 5 carbon atoms or a substituted or unsubstituted aralkyl group,and an insecticide, an acaricide and a fungicide for agriculture and horticulture, which comprises a carrier and the above phenoxyalkylamine derivative represented as the active ingredient.

公开(公告)号：US5498612A

公开(公告)日：1996-03-12

申请号：US380717

申请日：1995-01-30

申请人： Tokio Obata ,  Katsutoshi Fujii ,  Akira Ooka ,  Yoshinori Yamanaka

发明人： Tokio Obata ,  Katsutoshi Fujii ,  Akira Ooka ,  Yoshinori Yamanaka

IPC分类号： A01N43/54 ,  A01N47/06 ,  A01N55/00 ,  C07D239/42 ,  C07D401/12 ,  C07D405/12 ,  C07F7/18 ,  C07D239/30

CPC分类号： C07D239/42 ,  A01N43/54 ,  A01N47/06 ,  A01N55/00 ,  C07D401/12 ,  C07D405/12 ,  C07F7/1856

摘要： Disclosed are a 4-phenethylaminopyrimidine compound represented by the formula (I): ##STR1## wherein R.sup.1 represents halogen, hydroxyl, acyloxy, alkoxy, haloalkoxy, alkylthio, benzyloxycarbonyloxy, alkyloxycarbonyloxy, alkylsulfonyloxy, tri(alkyl)silyloxy or alkyloxycarbonylalkyloxy;R.sup.2 represents hydrogen, alkyl, alkoxy, halogen, haloalkyl, haloalkoxy, unsubstituted or substituted benzoyl, hydroxyl, haloalkylcarbonyl, alkylsulfonyloxy, haloalkylsulfonyloxy, alkylsulfonyl, alkylsulfinyl, haloalkylsulfinyl, tri(alkyl)silylalkoxy, alkylthio, unsubstituted or substituted pyridyloxy, unsubstituted or substituted phenoxy, alkenyloxy, haloalkenyloxy, unsubstituted or substituted benzyl, 2-phenyl-2-1,3-dioxolanyl, alkoxyiminobenzyl, nitro, haloalkylthio or alkynyloxy; n is an integer of 1 to 5 and * represents an asymmetric carbon atom.a process for preparing the same and an agricultural and horticultural chemical for controlling noxious organisms which contains the same as an active ingredient.

摘要翻译： 公开了由式（I）表示的4-苯乙基氨基嘧啶化合物：其中R 1表示卤素，羟基，酰氧基，烷氧基，卤代烷氧基，烷硫基，苄氧羰基氧基，烷氧基羰氧基，烷基磺酰氧基，三（烷基）甲硅烷氧基或烷氧基羰基烷氧基。 R 2表示氢，烷基，烷氧基，卤素，卤代烷基，卤代烷氧基，未取代或取代的苯甲酰基，羟基，卤代烷基羰基，烷基磺酰氧基，卤代烷基磺酰氧基，烷基磺酰基，烷基亚磺酰基，卤代烷基亚磺酰基，三（烷基）甲硅烷基烷氧基，烷硫基，未取代或取代的吡啶氧基，未取代或取代的苯氧基 ，烯氧基，卤代烯氧基，未取代或取代的苄基，2-苯基-2,3-二氧戊环，烷氧基亚氨基苄基，硝基，卤代烷硫基或炔氧基; n为1〜5的整数，*表示不对称碳原子。 其制备方法以及用于控制含有与活性成分相同的有害生物的农业和园艺化学品。

公开(公告)号：US5380744A

公开(公告)日：1995-01-10

申请号：US221496

申请日：1994-04-01

申请人： Tokio Obata ,  Akira Ooka ,  Katsutoshi Fujii ,  Shin Suizu

发明人： Tokio Obata ,  Akira Ooka ,  Katsutoshi Fujii ,  Shin Suizu

IPC分类号： A01N43/56 ,  A01N47/12 ,  C07C233/18 ,  C07C233/60 ,  C07C233/69 ,  C07C235/48 ,  C07D231/14 ,  C07D231/16 ,  C07D231/20 ,  C07D231/54 ,  A01N43/40 ,  C07D401/12

CPC分类号： C07D231/20 ,  A01N43/56 ,  A01N47/12 ,  C07C233/18 ,  C07C233/60 ,  C07C233/69 ,  C07C235/48 ,  C07D231/14 ,  C07D231/16 ,  C07D231/54 ,  C07C2101/02 ,  C07C2101/04

摘要： Disclosed are a phenoxyalkylamine compound represented by the formula (I): ##STR1## wherein R.sup.1 is C.sub.1-8 alkyl group, C.sub.3-8 cycloalkyl group, a hydrogen atom, a phenyl group, or C.sub.1-4 haloalkyl group; R.sup.2 is a halogen atom, a hydrogen atom, C.sub.1-4 alkyl group, C.sub.1-4 alkoxy group or a nitro group; R.sup.1 and R.sup.2 may be linked with each other and condensed to a pyrazole ring to form a saturated 4- to 8-membered ring; R.sup.3 is C.sub.1-15 alkyl group, C.sub.3-8 cycloalkyl group, a phenyl group, C.sub.1-4 haloalkyl group, C.sub.2-8 alkoxyalkyl group, C.sub.3-6 alkenyl group, a pyridyl group, a benzyl group, C.sub.3-8 alkoxycarbonylalkyl group, a pyrazole group, or C.sub.1-4 alkoxy group; R.sup.4 is C.sub.1-4 alkyl group, a hydrogen atom or a halogen atom; R.sup.5 is C.sub.1-20 alkyl group, a hydrogen atom, C.sub.3-6 alkenyl group, a benzyl group, a phenoxy group, a halogen atom, a cyanomethyl group or --A--O--R.sup.7 where A is C.sub.1-4 alkylene group and R.sup.7 is C.sub.1-6 alkyl group, C.sub.3-6 alkenyl group, C.sub.3-6 alkynyl group or C.sub.2-5 acyl group; and R.sup.6 is a hydrogen atom, C.sub.1-4 alkyl group or a halogen atom,a process for preparing the same and a chemical for controlling noxious organisms containing the same as an effective ingredient.

摘要翻译： 公开了由式（I）表示的苯氧基烷基胺化合物：其中R 1是C 1-8烷基，C 3-8环烷基，氢原子，苯基或C 1-4卤代烷基; R2是卤素原子，氢原子，C1-4烷基，C1-4烷氧基或硝基; R 1和R 2可以彼此连接并稠合成吡唑环以形成饱和的4-至8-元环; R3是C1-15烷基，C3-8环烷基，苯基，C1-4卤代烷基，C2-8烷氧基烷基，C3-6烯基，吡啶基，苄基，C3-8烷氧基羰基烷基， 吡唑基或C 1-4烷氧基; R4是C1-4烷基，氢原子或卤素原子; R5是C1-20烷基，氢原子，C3-6烯基，苄基，苯氧基，卤素原子，氰基甲基或-AO-R7，其中A是C1-4亚烷基，R7是C1 C6烷基，C3-6烯基，C3-6炔基或C2-5酰基; R6为氢原子，C1-4烷基或卤素原子，其制备方法以及控制含有有机成分的有害生物的化学物质。