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1.发明授权4-(azacycloalkyl)benzene-1,3-diol compounds as tyrosinase inhibitors, process for the preparation thereof and use thereof in human medicine and in cosmetics 有权4-（氮杂环烷基）苯-1,3-二醇化合物作为酪氨酸酶抑制剂，其制备方法及其在人类药物和化妆品中的应用公开(公告)号：US08299259B2
公开(公告)日：2012-10-30
申请号：US13131363
申请日：2009-12-02
IPC分类号： C07D211/06 , C07D295/00
CPC分类号： C07D401/12 , A61K9/06 , C07D205/04 , C07D207/08 , C07D207/16 , C07D211/22 , C07D211/26 , C07D211/60
摘要： 4-(azacycloalkyl)benzene-1,3-diol compounds are described corresponding to general formula (I) below: Also described, are compositions including the same, processes for preparation thereof and uses thereof in pharmaceutical or cosmetic compositions to treat pigmentary disorders.
摘要翻译： 4-（氮杂环烷基）苯-1,3-二醇化合物对应于下列通式（I）描述：还描述了包含它们的组合物，其制备方法及其在药物或化妆品组合物中用于治疗色素障碍的用途。
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2.发明申请4-(AZACYCLOALKYL)BENZENE-1,3-DIOL COMPOUNDS AS TYROSINASE INHIBITORS, PROCESS FOR THE PREPARATION THEREOF AND USE THEREOF IN HUMAN MEDICINE AND IN COSMETICS 有权4-（齐克洛尔基）苯甲腈-1,3-二醇化合物作为酪氨酸酶抑制剂，其制备方法及其在人体药物和化妆品中的应用公开(公告)号：US20130023516A1
公开(公告)日：2013-01-24
申请号：US13611546
申请日：2012-09-12
IPC分类号： A61K31/397 , A61P17/02 , A61P17/00 , A61K31/40 , A61K31/451
CPC分类号： C07D401/12 , A61K9/06 , C07D205/04 , C07D207/08 , C07D207/16 , C07D211/22 , C07D211/26 , C07D211/60
摘要： 4-(azacycloalkyl)benzene-1,3-diol compounds are described corresponding to general formula (I) below: Also described, are compositions including the same, processes for preparation thereof and uses thereof in pharmaceutical or cosmetic compositions to treat pigmentary disorders.
摘要翻译： 4-（氮杂环烷基）苯-1,3-二醇化合物对应于下列通式（I）描述：还描述了包含它们的组合物，其制备方法及其在药物或化妆品组合物中用于治疗色素障碍的用途。
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3.发明授权4-(azacycloalkyl)benzene-1,3-diol compounds as tyrosinase inhibitors, process for the preparation thereof and use thereof in human medicine and in cosmetics 有权4-（氮杂环烷基）苯-1,3-二醇化合物作为酪氨酸酶抑制剂，其制备方法及其在人类药物和化妆品中的应用公开(公告)号：US08697726B2
公开(公告)日：2014-04-15
申请号：US13611546
申请日：2012-09-12
IPC分类号： A61K31/445
CPC分类号： C07D401/12 , A61K9/06 , C07D205/04 , C07D207/08 , C07D207/16 , C07D211/22 , C07D211/26 , C07D211/60
摘要： 4-(azacycloalkyl)benzene-1,3-diol compounds are described corresponding to general formula (I) below: Also described, are compositions including the same, processes for preparation thereof and uses thereof in pharmaceutical or cosmetic compositions to treat pigmentary disorders.
摘要翻译： 4-（氮杂环烷基）苯-1,3-二醇化合物对应于下列通式（I）描述：还描述了包含它们的组合物，其制备方法及其在药物或化妆品组合物中用于治疗色素障碍的用途。
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4.发明申请NOVEL 4-(AZACYCLOALKYL)BENZENE-1,3-DIOL COMPOUNDS AS TYROSINASE INHIBITORS, PROCESS FOR THE PREPARATION THEREOF AND USE THEREOF IN HUMAN MEDICINE AND IN COSMETICS 有权新型4-（氮杂环丁基）苯甲-1,3-二醇化合物作为酪氨酸酶抑制剂，其制备方法及其在人体药物和化妆品中的应用公开(公告)号：US20110311466A1
公开(公告)日：2011-12-22
申请号：US13131363
申请日：2009-12-02
IPC分类号： A61K31/397 , C07D207/08 , C07D211/60 , A61K31/40 , A61Q19/02 , A61P17/00 , A61P17/02 , A61P37/08 , A61K8/49 , C07D205/04 , A61K31/451
CPC分类号： C07D401/12 , A61K9/06 , C07D205/04 , C07D207/08 , C07D207/16 , C07D211/22 , C07D211/26 , C07D211/60
摘要： 4-(azacycloalkyl)benzene-1,3-diol compounds are described corresponding to general formula (I) below: Also described, are compositions including the same, processes for preparation thereof and uses thereof in pharmaceutical or cosmetic compositions to treat pigmentary disorders.
摘要翻译： 4-（氮杂环烷基）苯-1,3-二醇化合物对应于下列通式（I）描述：还描述了包含它们的组合物，其制备方法及其在药物或化妆品组合物中用于治疗色素障碍的用途。
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5.发明申请NOVEL 4-HETEROARYLIMIDAZOLE-2-THIONE TYROSINASE INHIBITORS AND PHARMACEUTICAL/COSMETIC APPLICATIONS THEREOF 失效新型4-杂环二咪唑-2-硫酸酯酶抑制剂及其药物/化妆品应用公开(公告)号：US20100144813A1
公开(公告)日：2010-06-10
申请号：US12631309
申请日：2009-12-04
IPC分类号： A61K31/4178 , C07D233/10 , A61P17/02 , A61P37/08
CPC分类号： C07D405/04 , C07D409/04 , C07D417/04
摘要： Novel 4-heteroarylimidazole-2-thione tyrosinase inhibiting compounds corresponding to the following general formula (I): formulated into pharmaceutical or cosmetic compositions are useful for the treatment or prevention of pigmentary disorders, or for preventing and/or treating signs of skin aging, and/or for body or hair hygiene.
摘要翻译： 对应于以下通式（I）的新型4-杂芳基咪唑-2-硫酮酪氨酸酶抑制化合物：配制成药物或化妆品组合物可用于治疗或预防色素障碍，或用于预防和/或治疗皮肤老化迹象， 和/或用于身体或头发卫生。
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6.发明授权4-heteroarylimidazole-2-thione tyrosinase inhibitors and pharmaceutical/cosmetic applications thereof 失效4-杂芳基咪唑-2-硫酮酪氨酸酶抑制剂及其药物/化妆品应用公开(公告)号：US07989483B2
公开(公告)日：2011-08-02
申请号：US12631309
申请日：2009-12-04
IPC分类号： A61K31/4178 , C07D233/20
CPC分类号： C07D405/04 , C07D409/04 , C07D417/04
摘要： Novel 4-heteroarylimidazole-2-thione tyrosinase inhibiting compounds corresponding to the following general formula (I): formulated into pharmaceutical or cosmetic compositions are useful for the treatment or prevention of pigmentary disorders, or for preventing and/or treating signs of skin aging, and/or for body or hair hygiene.
摘要翻译： 对应于以下通式（I）的新型4-杂芳基咪唑-2-硫酮酪氨酸酶抑制化合物：配制成药物或化妆品组合物可用于治疗或预防色素障碍，或用于预防和/或治疗皮肤老化迹象， 和/或用于身体或头发卫生。
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