公开(公告)号：US20060241128A1

公开(公告)日：2006-10-26

申请号：US10532719

申请日：2003-11-04

申请人： Jordi Tormo I Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Tormo I Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04

CPC分类号： C07C69/65 ,  A01N43/90 ,  C07D487/04

摘要： Substituted 6-(2-halogenphenyl)-triazolopyrimidines of formula I in which R1 denote alkyl, alkenyl, alkynyl, alkadienyl, haloalkyl, haloalkenyl, cycloalkyl, phenyl, naphthyl, or a 5- or 6-membered saturated, unsaturated, or aromatic heterocycle, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, wherein R1 and R2 radicals may be substituted as defined in the description, R2 denote hydrogen, or a group mentioned for R1; or R1 and R2 together with the interjacent nitrogen atom represent a 5- or 6-membered heterocycle, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which ring may be substituted as defined in the description; Hal is halogen; L1, L3 independently denote hydrogen, halogen, or alkyl; L2 is hydrogen, halogen, haloalkyl, or NH2, NHRb, or N(Rb)2, wherein Rb is as defined in the description, wherein at least one from L1, L2, and L3 is not hydrogen; X is halogen, cyano, alkyl, alkoxy, haloalkoxy or alkenyloxy. processes for their preparation, compositions containing them and to their use for combating phytopathogenic fungi.

摘要翻译： 其中R 1表示烷基，烯基，炔基，链二烯基，卤代烷基，卤代烯基，环烷基，苯基，萘基或5-或6-元的取代的6-（2-卤代苯基） - 三唑并嘧啶， 含有1至4个氮原子或1至3个氮原子和1个硫或氧原子的饱和，不饱和或芳族杂环，其中R 1和R 2可以是 如说明书中所定义，R 2表示氢或R 1所提及的基团; 或R 1和R 2连同中间的氮原子代表含有1-4个氮原子或一至三个氮原子的一个或多个六元杂环，一个 硫或氧原子，该环可以如说明书中所定义取代; 卤素是卤素; L 1，L 3独立地表示氢，卤素或烷基; L 2是氢，卤素，卤代烷基或NH 2，NHR b或/或N（R b） 其中R b如描述中所定义，其中至少一个L 1，L 2， ，而L 3不是氢; X是卤素，氰基，烷基，烷氧基，卤代烷氧基或烯氧基。 其制备方法，含有它们的组合物及其用于对抗植物病原真菌的用途。

公开(公告)号：US20060100220A1

公开(公告)日：2006-05-11

申请号：US10532769

申请日：2003-11-14

申请人： Jordi Tormo I Blasco ,  Thomas Grote ,  Eberhard Ammermann ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

发明人： Jordi Tormo I Blasco ,  Thomas Grote ,  Eberhard Ammermann ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

IPC分类号： A01N43/90 ,  A01N43/80 ,  A01N43/50

CPC分类号： A01N43/90 ,  A01N2300/00

摘要： Fungicidal mixtures, comprising A) the triazolopyrimidine of the formula I and B) imidazole derivatives of the formula II where X1 and X2 are halogen and phenyl which may be substituted by halogen or alkyl or X1 and X2 together with the bridging C═C double bond form a difluoromethylenedioxyphenyl group; X3 is cyano or halogen, and X4 is dialkylamino or isoxazol-4-yl which may carry two alkyl radicals, in a synergistically effective amount, methods for controlling harmful fungi using mixtures of the compounds I and II, compositions comprising these compounds and the use of the compounds I and II for preparing such mixtures are described.

摘要翻译： 杀真菌混合物，其包含A）式I的三唑并嘧啶和B）式II的咪唑衍生物，其中X 1和X 2是卤素和可以被 卤素或烷基或X 1和X 2连同桥连CC双键形成二氟亚甲二氧基苯基; X 3是氰基或卤素，X 4是可以以协同有效量存在两个烷基的二烷基氨基或异恶唑-4-基，用于控制有害真菌的方法 描述了使用化合物I和II的混合物，包含这些化合物的组合物和化合物I和II用于制备这些混合物的用途。

公开(公告)号：US20070191397A1

公开(公告)日：2007-08-16

申请号：US11579084

申请日：2004-05-17

申请人： Jordi Tormo i Blasco ,  Thomas Grote ,  Eberhard Ammermann ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

发明人： Jordi Tormo i Blasco ,  Thomas Grote ,  Eberhard Ammermann ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

IPC分类号： A01N43/90 ,  A01N37/18

CPC分类号： A01N43/90 ,  A01N37/52 ,  A01N2300/00

摘要： The invention relates to fungicidal mixtures containing: A) triazolopyrimidine of formula (I) and B) oxime derivatives of formula (II), wherein the index and substitutents have the following meaning: X=C1-halogen alkyl or C1-halogen alkoxy; R=halogen, alkyl, halogen alkyl, alkoxy or halogen alkoxy; n=0, 1, 2 or 3 in a synergistically effective amount. The invention also relates to a method for controlling harmful fungi with mixtures of compounds (I) and (II), to the agents containing said mixtures and to the utilization of compounds (I) and (II) for the production of said mixtures.

摘要翻译： 本发明涉及杀真菌混合物，其包含：A）式（I）的三氮代嘧啶和B）式（II）的肟衍生物，其中指数和取代基具有以下含义：X = C 1 - 卤素 烷基或C 1 - 卤代烷氧基; R =卤素，烷基，卤素烷基，烷氧基或卤素烷氧基; n = 0,1,2或3，具有协同有效量。 本发明还涉及一种利用化合物（I）和（II）的混合物将有害真菌控制在含有所述混合物的试剂中，以及利用化合物（I）和（II）来生产所述混合物的方法。

公开(公告)号：US20050176736A1

公开(公告)日：2005-08-11

申请号：US10508409

申请日：2003-03-19

申请人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl ,  Ulrich Schofl

发明人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl ,  Ulrich Schofl

IPC分类号： A01N43/90 ,  C07C255/57 ,  C07D487/04 ,  A61K31/519

CPC分类号： C07D487/04 ,  A01N43/90 ,  C07C255/57

摘要： The invention relates to triazolopyrimidines of formula (I), in which the substituents are defined as follows: L1 represents cyano, S(═O)nA1 or C(═O)A2, wherein A1 stands for hydrogen, hydroxy, alkyl, alkylamino or dialkylamino; A2 stands for C1-C8 alkoxy, C1-C6 haloalkoxy or one of the groups named in A1; and n stands for 0, 1 or 2; L2, L3 represent hydrogen or halogen; L4, L5 represent hydrogen, halogen or alkyl; X represents halogen, cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; R1 represents alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl or cycloalkynyl, phenyl, naphthyl, or a five to ten-membered saturated, partially unsaturated or aromatic heterocyclus containing between one and four heteroatoms from the group containing O, N or S; R2 represents hydrogen or R1; R1 and R2 can form, together with the nitrogen atom to which they are bonded, a five or six-membered ring, which can be interrupted and/or substituted by an atom from the group O, N and S; whereby R1 and/or R2 can be substituted in accordance with the description. The invention also relates to methods and intermediate products for producing said compounds, to agents containing the latter and to the use of said compounds for combating harmful fungi.

摘要翻译： 本发明涉及式（I）的三唑并嘧啶，其中取代基定义如下：L 1表示氰基，S（-O）n A 1 或其中A 1代表氢，羟基，烷基，烷基氨基或二烷基氨基;或C（= O） A 2代表C 1 -C 8烷氧基，C 1 -C 6烷基，C 1 -C 6 - >卤代烷氧基或在A 中命名的基团之一; 而n代表0,1或2; L 2，L 3表示氢或卤素; L 4，L 5代表氢，卤素或烷基; X表示卤素，氰基，烷基，卤代烷基，烷氧基或卤代烷氧基; R 1表示烷基，卤代烷基，环烷基，卤代环烷基，烯基，链烯基，卤代烯基，环烯基，炔基，卤代炔基或环炔基，苯基，萘基或五至十元饱和，部分不饱和或芳族杂环 含有一个至四个来自含有O，N或S的基团的杂原子; R 2表示氢或R 1; R 1和R 2可以与它们所键合的氮原子一起形成五元或六元环，其可被中断和/或被 来自O，N和S族的原子; 其中R 1和/或R 2可以根据描述被取代。 本发明还涉及用于生产所述化合物的方法和中间产物，含有后者的试剂和所述化合物用于防治有害真菌的用途。

公开(公告)号：US20080221177A1

公开(公告)日：2008-09-11

申请号：US12101175

申请日：2008-04-11

申请人： Wassilios GRAMMENOS ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Jordi Tormo i Blasco ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Norbert Gotz ,  Siegfried Strathmann ,  Ulrich Schofl ,  Maria Scherer ,  Reinhard Stierl

发明人： Wassilios GRAMMENOS ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Jordi Tormo i Blasco ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Norbert Gotz ,  Siegfried Strathmann ,  Ulrich Schofl ,  Maria Scherer ,  Reinhard Stierl

IPC分类号： A01N43/40 ,  A01P3/00

CPC分类号： C04B35/632 ,  C07D213/42 ,  C07D215/12 ,  C07D401/12 ,  C07D409/12

摘要： Sulfonamides of the formula I where the substituents are as follows: R1 is hydrogen, alkyl, alkoxy, alkenyl or alkynyl; and R2, R3, R4, R5 are hydrogen, halogen, alkyl, alkoxy or halomethyl; R2 and R3 together may also form a phenyl, cyclopentyl or cyclohexyl ring, it being possible for these rings to carry two groups R2′ and R3′, R2′, R3′ are hydrogen, halogen, alkyl, alkoxy or halomethyl; in case a), if R2, R3, R4 and R5 are hydrogen: X is phenyl substituted by a group C(R6)═NOR7, where R6 is alkyl and R7 is alkyl, benzyl, alkenyl, haloalkyl, haloalkenyl, alkynyl or haloalkynyl; and in case b), if at least one of the groups R2, R3, R4 and R5 is not hydrogen: X is phenyl, naphthyl or a five- or six-membered saturated, or partially unsaturated or aromatic heterocycle which is attached via a carbon atom and contains one to four heteroatoms from the group consisting of O, N and S, where X may be substituted according to the description; Processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

摘要翻译： 式I的磺酰胺，其中取代基如下：R 1是氢，烷基，烷氧基，烯基或炔基; R 2，R 3，R 4，R 5是氢，卤素，烷基，烷氧基或卤代甲基 ; R 2和R 3一起也可以形成苯基，环戊基或环己基环，这些环可以携带两个基团R 2， '和R 3'，R 2'，R 3'是氢，卤素，烷基，烷氧基或卤代甲基; 在a）情况下，如果R 2，R 3，R 4和R 5是氢：X是 被C（R 6） - - NOR 7取代的苯基，其中R 6是烷基，R 7是 烷基，苄基，烯基，卤代烷基，卤代烯基，炔基或卤代炔基; 并且在情况b）中，如果R 2，R 3，R 4和R 5中的至少一个， SUP>不是氢：X是苯基，萘基或五或六元饱和或部分不饱和或芳族杂环，其通过碳原子连接并含有一至四个由O，N和S组成的组的杂原子 ，其中X可以根据描述被替代; 制备这些化合物的方法，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20080139387A1

公开(公告)日：2008-06-12

申请号：US10585981

申请日：2005-01-15

申请人： Jordi Tormo i Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

发明人： Jordi Tormo i Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

IPC分类号： A01N25/34 ,  A01N43/84 ,  A01P3/00

CPC分类号： A01N43/90 ,  A01N43/84 ,  A01N2300/00

摘要： The invention relates to fungicidal mixtures for the control of fungal pests harmful to plants, comprising the active components 1) the triazolopyrimidine derivative of formula (1), and 2) tridemorph of formula (II), in which n=10, 11, 12 (60-70%) or 14, in a synergistically-effective amount, method for the control of fungal pests using mixtures of compound (I) with the compounds (II), the use of compound (I) with the compounds (II) for the production of such mixtures and means comprising said mixtures.

摘要翻译： 本发明涉及用于控制对植物有害的真菌害虫的杀真菌混合物，其包含活性组分1）式（1）的三唑并嘧啶衍生物和2）式（II）的三美丹，其中n = 10,11,12 （I）与化合物（II）的混合物，使用化合物（I）与化合物（II）的混合物来控制真菌害虫的方法（60-70％）或14， 用于生产这样的混合物和包含所述混合物的装置。

公开(公告)号：US20080139386A1

公开(公告)日：2008-06-12

申请号：US10585741

申请日：2005-01-13

申请人： Jordi Tormo i Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

发明人： Jordi Tormo i Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

IPC分类号： A01N25/34 ,  A01N43/54 ,  A01P3/00

CPC分类号： A01N43/90 ,  A01N47/32 ,  A01N2300/00

摘要： Fungicidal mixtures for controlling harmful fungi, which mixtures comprise, as active components,1) the triazolopyrimidine derivative of the formula I and2) pencycuron of the formula II in a synergistically effective amount, methods for controlling rice pathogens using mixtures of the compound I with the compounds II and the use of the compound I with the compounds II for preparing such mixtures, and also compositions comprising these mixtures.

摘要翻译： 用于控制有害真菌的杀真菌混合物，其混合物包含作为活性组分的1）式I的三氮代嘧啶衍生物和2）协同有效量的式II的焦虑霉素，使用化合物I与 化合物II和化合物I与化合物II用于制备这种混合物的用途，以及包含这些混合物的组合物。

公开(公告)号：US20070191396A1

公开(公告)日：2007-08-16

申请号：US10591342

申请日：2005-03-17

申请人： Jordi Tormo i Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl ,  Markus Gewehr

发明人： Jordi Tormo i Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl ,  Markus Gewehr

IPC分类号： A01N43/90 ,  A01N37/52 ,  A01N37/34

CPC分类号： A01N43/90 ,  A01N2300/00

摘要： The invention relates to fungicidal mixtures, containing the following in a synergistically effective quantity as active components: 1) the triazolopyrimidine derivative of formula (I); and 2) a phenylamidine derivative of formula (II), in which the variables are defined as follows: R1, R4, R5 represent alkyl, alkenyl or alkynyl; R2, R3 represent cyano, alkyl, alkenyl, alkynyl, alkoxy, alkoxyalkyl, benzyloxy or alkylcarbonyl; m represents 0 or 1; A represents a direct bond, —O—, —S—, NRd, CHRe or —O—CHRe; R6 represents phenyl or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle, containing between one and four heteroatoms from the group comprising O, N or S, whereby the groups can be substituted according to the description. The invention also relates to a method for controlling pathogenic fungi using mixtures of compounds (I) and (II), to the use of compounds (I) and (II) for producing mixtures of this type and to agents that contain said mixtures.

摘要翻译： 本发明涉及杀真菌混合物，其具有协同有效量作为活性成分：1）式（I）的三唑并嘧啶衍生物; 和2）式（II）的苯基脒衍生物，其中变量定义如下：R 1，R 4，R 5， 代表烷基，烯基或炔基; R 2，R 3代表氰基，烷基，烯基，炔基，烷氧基，烷氧基烷基，苄氧基或烷基羰基; m表示0或1; A表示直接键，-O-，-S-，NR d，CHR e或-O-CHR e; R 6表示苯基或五元或六元饱和，部分不饱和或芳族杂环，其含有一个至四个来自O，N或S的基团的杂原子，其中基团可以根据 的描述。 本发明还涉及使用化合物（I）和（II）的混合物来控制致病真菌的方法，用于制备这种类型的混合物和含有所述混合物的试剂的化合物（I）和（II）。

公开(公告)号：US20070135453A1

公开(公告)日：2007-06-14

申请号：US10579395

申请日：2004-12-14

申请人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04

CPC分类号： C07D487/04 ,  A01N43/90

摘要： The present invention relates to 6-(2,4,6-trihalophenyl)triazolopyrimidines of the formula I in which the substituents are as defined below: R1 is alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl or a five- or six-member saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R2 is hydrogen or one of the groups mentioned under R1, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and may contain one to three further heteroatoms from the group consisting of O, N and S as ring members; R1 and/or R2 may be substituted as defined in the description; L1, L2, L3 are chlorine or fluorine, where at least one group is chlorine; X is cyano, alkyl, alkoxy, alkenyloxy, haloalkoxy or haloalkenyloxy; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

摘要翻译： 本发明涉及式I的6-（2,4,6-三卤代苯基）三唑并嘧啶，其中取代基如下：R 1是烷基，卤代烷基，环烷基，卤代环烷基，烯基， 卤代烯基，环烯基，卤代环烯基，炔基，卤代炔基或苯基，萘基或五或六元饱和的部分不饱和或芳族杂环，其含有一至四个由O，N和S组成的组的杂原子，R 2 R 1是氢或R 1，R 2和R 2中所提及的基团之一，与它们的氮原子一起 还可以形成通过N连接的五元或六元杂环基或杂芳基，并且可以含有一个至三个其它由O，N和S组成的组的杂原子作为环成员; R 1和/或R 2可以如说明书中所定义的取代; L 1，L 2，L 3 3是氯或氟，其中至少一个基团是氯; X是氰基，烷基，烷氧基，烯氧基，卤代烷氧基或卤代烯氧基; 制备这些化合物的方法，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20060063786A1

公开(公告)日：2006-03-23

申请号：US10532841

申请日：2003-11-14

申请人： Jordi Tormo I Blasco ,  Thomas Grote ,  Eberhard Ammermann ,  Reinhard Stierl ,  Siegfried Strathman ,  Ulrich Schofl

发明人： Jordi Tormo I Blasco ,  Thomas Grote ,  Eberhard Ammermann ,  Reinhard Stierl ,  Siegfried Strathman ,  Ulrich Schofl

IPC分类号： A01N43/90 ,  A01N37/18

CPC分类号： A01N43/90 ,  A01N37/50 ,  A01N2300/00

摘要： Fungicidal mixtures for controlling rice pathogens, comprising, as active components, 1) the compound of the formula I, and 2) the compound of the formula II, in a synergistically effective amount, methods for controlling harmful fungi using mixtures of the compound I with the compound II, the use of the compounds I and II for preparing such mixtures and compositions comprising these mixtures are described.

摘要翻译： 用于防治水稻病原体的杀真菌混合物，包括作为活性成分