公开(公告)号：US4661477A

公开(公告)日：1987-04-28

申请号：US426949

申请日：1982-09-29

申请人： Katalin Gorog nee Privitzer ,  Laszlo Bodnar ,  Erzsebet Dudar ,  Maria Kocsis nee Bagi ,  Sandor Gaal ,  Marta Tasnadi ,  Eva Egyhazi nee Csizmadia ,  Valeria M. Varga ,  Istvan Kajati ,  Gyorgy Kis ,  Janos Molnar ,  Bertalan Toth ,  Ilona Cserhati nee Botka ,  Tibor Kaptas ,  Sandor Csete

发明人： Katalin Gorog nee Privitzer ,  Laszlo Bodnar ,  Erzsebet Dudar ,  Maria Kocsis nee Bagi ,  Sandor Gaal ,  Marta Tasnadi ,  Eva Egyhazi nee Csizmadia ,  Valeria M. Varga ,  Istvan Kajati ,  Gyorgy Kis ,  Janos Molnar ,  Bertalan Toth ,  Ilona Cserhati nee Botka ,  Tibor Kaptas ,  Sandor Csete

IPC分类号： A01N57/10 ,  A01N33/12 ,  A01N57/12 ,  A01N57/14 ,  A01P3/00 ,  C07F9/09 ,  C07F9/141 ,  C07F9/142 ,  C07F9/38 ,  C07F9/40 ,  A01N57/26

CPC分类号： C07F9/142 ,  A01N57/12 ,  A01N57/14 ,  C07F9/141

摘要： The invention relates to new compounds of the general formula I ##STR1## wherein R.sub.1 is a straight or branched chained alkyl having 1 to 13 carbon atoms, optionally substituted with halogen, alkoxyalkyl containing 1 to 5 carbon atoms in the alkoxy and 1 to 4 carbon atoms in the alkyl moiety or phenyl;R.sub.2 is alkyl having 6 to 20 carbon atoms; alkoxyalkyl, phenoxyalkyl, furfuryl, cyclopropyl-alkyl, cyclopentyl, cycloheptyl, thiazolyl, triazolyl, thiazolinyl, pyridinyl, picolyl, benzimidazolyl, piperonyl, pirimidinyl, chlorobenzothiazolyl, benzyl, phenyl substituted with chloro and/or amino, or amino and alkyl, or amino and nitro groups, alkenyl, alkinyl, aminoalkyl, dialkylamino-alkyl, alkylaminoalkyl, alkylphosphonateammoniumalkyl, 3,5-dichlorophenyl-hidantoinyl, or thiadiazolyl optionally substituted with alkyl;R.sub.3 is hydrogen, phenyl, benzyl, alkenyl, alkyl, hydroxy, alkoxy or alkoxyalkyl; orR.sub.2 and R.sub.3 together stand for a 3,5-dichlorophenyl-hidantoinyl group;R.sub.4 is hydrogen or alkyl optionally substituted with hydroxyl.The new phosphoric acid monoester salts of the general formula I show fungicidal activity. The fungicidal compositions containing said compounds as active ingredients are also within the scope of the invention. According to a further aspect of the invention there is provided a process for the preparation of the new compounds.

摘要翻译： 本发明涉及通式I（I）的新化合物，其中R 1是具有1至13个碳原子的直链或支链链烷基，任选被卤素取代，烷氧基中含有1至5个碳原子的烷氧基烷基和1 至烷基部分中的4个碳原子或苯基; R2是具有6至20个碳原子的烷基; 烷氧基烷基，苯氧基烷基，糠基，环丙基 - 烷基，环戊基，环庚基，噻唑基，三唑基，噻唑啉基，吡啶基，吡啶甲基，苯并咪唑基，胡椒基，吡啶基，氯代苯并噻唑基，苄基，被氯和/或氨基取代的苯基，或氨基和烷基或氨基 硝基，烯基，炔基，氨基烷基，二烷基氨基 - 烷基，烷基氨基烷基，烷基膦酸铵烷基，3,5-二氯苯基 - 乙二酰基或任选被烷基取代的噻二唑基; R3是氢，苯基，苄基，烯基，烷基，羟基，烷氧基或烷氧基烷基; 或R 2和R 3一起代表3,5-二氯苯基 - 乙酰乙酰基; R4是氢或任选被羟基取代的烷基。 通式I的新型磷酸单酯盐显示出杀真菌活性。 含有所述化合物作为活性成分的杀真菌组合物也在本发明的范围内。 根据本发明的另一方面，提供了一种制备新化合物的方法。

公开(公告)号：US4675431A

公开(公告)日：1987-06-23

申请号：US888267

申请日：1986-07-18

申请人： Katalin Gorog nee Privitzer ,  Laszlo Bodnar ,  Erzsebet Dudar ,  Maria Kocsis nee Bagi ,  Sandor Gaal ,  Marta Tasnadi ,  Eva Egyhazi nee Csizmadia ,  Valeria M. Varga ,  Istvan Kajati ,  Gvorgy Kis ,  Janos Molnar ,  Bertalan Toth ,  Ilona Cserhati nee Botka ,  Tibor Kaptas ,  Sandor Csete

发明人： Katalin Gorog nee Privitzer ,  Laszlo Bodnar ,  Erzsebet Dudar ,  Maria Kocsis nee Bagi ,  Sandor Gaal ,  Marta Tasnadi ,  Eva Egyhazi nee Csizmadia ,  Valeria M. Varga ,  Istvan Kajati ,  Gvorgy Kis ,  Janos Molnar ,  Bertalan Toth ,  Ilona Cserhati nee Botka ,  Tibor Kaptas ,  Sandor Csete

IPC分类号： A01N57/10 ,  A01N33/12 ,  A01N57/12 ,  A01N57/14 ,  A01P3/00 ,  C07F9/09 ,  C07F9/141 ,  C07F9/142 ,  C07F9/38 ,  C07F9/40

CPC分类号： C07F9/142 ,  A01N57/12 ,  A01N57/14 ,  C07F9/141

摘要： The invention relates to new compounds of the general formula I ##STR1## wherein R.sub.1 is a straight or branched chained alkyl having 1 to 13 carbon atoms, optionally substituted with halogen, alkoxyalkyl containing 1 to 5 carbon atoms in the alkoxy and 1 to 4 carbon atoms in the alkyl moiety or phenyl;R.sub.2 is alkyl having 6 to 20 carbon atoms; alkoxyalkyl, phenoxyalkyl, furfuryl, cyclopropyl-alkyl, cyclopentyl, cycloheptyl, thiazolyl, triazolyl, thiazolinyl, pyridinyl, picolyl, benzimidazolyl, piperonyl, pirimidinyl, chlorobenzothiazolyl, benzyl, phenyl substituted with chloro and/or amino, or amino and alkyl, or amino and nitro groups, alkenyl, alkinyl, aminoalkyl, dialkylamino-alkyl, alkylaminoalkyl, alkylphosphonateammoniumalkyl, 3,5-dichlorophenyl-hidantoinyl, or thiadiazolyl optionally substituted with alkyl;R.sub.3 is hydrogen, phenyl, benzyl, alkenyl, alkyl, hydroxy, alkoxy or alkoxyalkyl; orR.sub.2 and R.sub.3 together stand for a 3,5-dichlorophenyl-hidantoinyl group;R.sub.4 is hydrogen or alkyl optionally substituted with hydroxyl.The new phosphoric acid monoester salts of the general formula I show fungicidal activity. The fungicidal compositions containing said compounds as active ingredients are also within the scope of the invention. According to a further aspect of the invention there is provided a process for the preparation of the new compounds.

摘要翻译： 本发明涉及通式I（I）的新化合物，其中R 1是具有1至13个碳原子的直链或支链链烷基，任选被卤素取代，烷氧基中含有1至5个碳原子的烷氧基烷基和1 至烷基部分中的4个碳原子或苯基; R2是具有6至20个碳原子的烷基; 烷氧基烷基，苯氧基烷基，糠基，环丙基 - 烷基，环戊基，环庚基，噻唑基，三唑基，噻唑啉基，吡啶基，吡啶甲基，苯并咪唑基，胡椒基，吡啶基，氯代苯并噻唑基，苄基，被氯和/或氨基取代的苯基，或氨基和烷基或氨基 硝基，烯基，炔基，氨基烷基，二烷基氨基 - 烷基，烷基氨基烷基，烷基膦酸铵烷基，3,5-二氯苯基 - 乙二酰基或任选被烷基取代的噻二唑基; R3是氢，苯基，苄基，烯基，烷基，羟基，烷氧基或烷氧基烷基; 或R 2和R 3一起代表3,5-二氯苯基 - 乙酰乙酰基; R4是氢或任选被羟基取代的烷基。 通式I的新型磷酸单酯盐显示出杀真菌活性。 含有所述化合物作为活性成分的杀真菌组合物也在本发明的范围内。 根据本发明的另一方面，提供了一种制备新化合物的方法。