-
公开(公告)号:US20060025412A1
公开(公告)日:2006-02-02
申请号:US11178823
申请日:2005-10-14
IPC分类号: A61K31/5377 , A61K31/496 , A61K31/454 , A61K31/506 , A61K31/4015 , A61K31/4025
CPC分类号: C07D207/26 , C07D401/06 , C07D401/12 , C07D405/12 , C07D413/06 , C07D417/06
摘要: PDF inhibitors and novel methods for their use are provided.
摘要翻译: 提供PDF抑制剂及其使用的新方法。
-
公开(公告)号:US20070155792A1
公开(公告)日:2007-07-05
申请号:US11683089
申请日:2007-03-07
IPC分类号: A61K31/4439 , A61K31/454 , A61K31/42 , A61K31/4015 , A61K31/4025 , C07D413/02 , C07D405/02 , C07D403/02
CPC分类号: C07D207/26 , C07D401/06 , C07D401/12 , C07D405/12 , C07D413/06 , C07D417/06
摘要: PDF inhibitors and novel methods for their use are provided.
摘要翻译: 提供PDF抑制剂及其使用的新方法。
-
公开(公告)号:US06897233B2
公开(公告)日:2005-05-24
申请号:US10469560
申请日:2002-03-01
IPC分类号: A61K31/4015 , A61P31/00 , A61P31/04 , A61P43/00 , C07D207/26 , C07D207/12 , A61K31/40
CPC分类号: C07D207/26
摘要: PDF inhibitors and novel methods for their use are provided.
摘要翻译: 提供PDF抑制剂及其使用的新方法。
-
公开(公告)号:US07456211B2
公开(公告)日:2008-11-25
申请号:US11683089
申请日:2007-03-07
申请人: Kelly M. Aubart , Jia-Ning Xiang , Siegfried B. Christensen, IV , Xiangmin Liao , Maxwell D. Cummings
发明人: Kelly M. Aubart , Jia-Ning Xiang , Siegfried B. Christensen, IV , Xiangmin Liao , Maxwell D. Cummings
IPC分类号: A61K31/4015 , C07D207/10
CPC分类号: C07D207/26 , C07D401/06 , C07D401/12 , C07D405/12 , C07D413/06 , C07D417/06
摘要: The present invention involves novel anti-bacterial compounds represented by Formula (I), pharmaceutical compositions thereof, their use as PDF inhibitors, and their use in the treatment of bacterial infections.
摘要翻译: 本发明涉及由式(I)表示的新型抗菌化合物,其药物组合物,它们作为PDF抑制剂的用途及其在治疗细菌感染中的用途。
-
5.Levodopa dimethyl-substituted diester prodrugs, compositions, and methods of use 有权
标题翻译: 左旋多巴二甲基取代的二酯前药,组合物和使用方法公开(公告)号:US08324272B2
公开(公告)日:2012-12-04
申请号:US12726978
申请日:2010-03-18
申请人: Jia-Ning Xiang , Cindy X. Zhou , Fenmei Yao , Mark Q. Nguyen
发明人: Jia-Ning Xiang , Cindy X. Zhou , Fenmei Yao , Mark Q. Nguyen
IPC分类号: A61K31/235 , C07C229/36
CPC分类号: C07C229/36
摘要: Levodopa dimethyl-substituted diester prodrugs pharmaceutical, compositions comprising levodopa dimethyl-substituted diester prodrugs, and methods of using such prodrugs and pharmaceutical compositions for treating diseases such as Parkinson's disease are provided.
摘要翻译: 提供左旋多巴二甲基取代的二酯前药药物,包含左旋多巴二甲基取代的二酯前药的组合物,以及使用这些前药和药物组合物治疗疾病如帕金森病的方法。
-
公开(公告)号:US20120190861A1
公开(公告)日:2012-07-26
申请号:US13440936
申请日:2012-04-05
申请人: Jia-Ning Xiang , Mark A. Gallop , Cindy X. Zhou , Mark Nguyen , Xuedong Dai , Jianhua Li , Kenneth C. Cundy , Nelson L. Jumbe
发明人: Jia-Ning Xiang , Mark A. Gallop , Cindy X. Zhou , Mark Nguyen , Xuedong Dai , Jianhua Li , Kenneth C. Cundy , Nelson L. Jumbe
IPC分类号: C07D213/80 , C07C235/48 , C07C229/36
CPC分类号: C07C235/60 , C07C229/34 , C07C229/36 , C07C235/48 , C07C2601/14 , C07D213/79 , C07D213/80 , C07D213/803
摘要: Prodrugs of levodopa, methods of making prodrugs of levodopa, methods of using prodrugs of levodopa, and compositions of prodrugs of levodopa are disclosed.
摘要翻译: 公开了左旋多巴的前药,制备左旋多巴的前药的方法,使用左旋多巴的前药的方法和左旋多巴的前药组合物。
-
7.5-MEMBERED HETEROARYL DERIVATIVES USED AS SPHINGOSINE 1- PHOSPHATE RECEPTOR AGONISTS 审中-公开
标题翻译: 用作SPHINGOSINE 1-磷酸酯受体激动剂的5-MEMBERED HETEROARYL衍生物公开(公告)号:US20120101136A1
公开(公告)日:2012-04-26
申请号:US13379498
申请日:2010-06-24
申请人: Guanghui Deng , Xichen Lin , Feng Ren , Jia-Ning Xiang
发明人: Guanghui Deng , Xichen Lin , Feng Ren , Jia-Ning Xiang
IPC分类号: A61K31/433 , A61K31/425 , C07D285/08 , C07D271/06 , C07D233/61 , A61P9/00 , A61P25/00 , A61P37/00 , A61P29/00 , A61P41/00 , A61P19/02 , A61P1/00 , A61P17/06 , A61P35/00 , A61P35/04 , A61P3/10 , A61K31/4245
CPC分类号: A61K31/422 , A61K31/4245 , A61K31/427 , A61K31/433 , C07D263/32 , C07D271/06 , C07D271/107 , C07D277/30 , C07D285/08 , C07D285/12 , C07D413/04 , C07D413/14 , C07D417/04 , C07D417/14
摘要: 5-membered heteroaryl derivatives of formula (I) or salts thereof, processes for their preparation, pharmaceutical compositions containing them and their uses in the treatment of various disorders mediated by S1P1 receptors are disclosed.
摘要翻译: 公开了式(I)的5元杂芳基衍生物或其盐,其制备方法,含有它们的药物组合物及其在治疗由S1P1受体介导的各种疾病中的用途。
-
公开(公告)号:US07956212B2
公开(公告)日:2011-06-07
申请号:US12364453
申请日:2009-02-02
申请人: Jia-Ning Xiang , Mark A. Gallop , Cindy X. Zhou , Mark Nguyen , Xuedong Dai , Jianhua Li , Kenneth C. Cundy , Nelson L. Jumbe
发明人: Jia-Ning Xiang , Mark A. Gallop , Cindy X. Zhou , Mark Nguyen , Xuedong Dai , Jianhua Li , Kenneth C. Cundy , Nelson L. Jumbe
IPC分类号: C07C229/00
CPC分类号: C07C235/60 , C07C229/34 , C07C229/36 , C07C235/48 , C07C2601/14 , C07D213/79 , C07D213/80 , C07D213/803
摘要: Prodrugs of levodopa, methods of making prodrugs of levodopa, methods of using prodrugs of levodopa, and compositions of prodrugs of levodopa are disclosed.
摘要翻译: 公开了左旋多巴的前药,制备左旋多巴的前药的方法,使用左旋多巴的前药的方法和左旋多巴的前药组合物。
-
9.Levodopa dimethyl-substituted diester prodrugs compositions, and methods of use 失效
标题翻译: 左旋多巴二甲基取代的二酯前药组合物和使用方法公开(公告)号:US20080214663A1
公开(公告)日:2008-09-04
申请号:US12005117
申请日:2007-12-20
申请人: Jia-Ning Xiang , Cindy X. Zhou , Fenmei Yao , Mark Q. Nguyen
发明人: Jia-Ning Xiang , Cindy X. Zhou , Fenmei Yao , Mark Q. Nguyen
IPC分类号: A61K31/192 , C07C69/00 , A61P25/00 , A61P9/00
CPC分类号: C07C229/36
摘要: Levodopa dimethyl-substituted diester prodrugs pharmaceutical, compositions comprising levodopa dimethyl-substituted diester prodrugs, and methods of using such prodrugs and pharmaceutical compositions for treating diseases such as Parkinson's disease are provided.
摘要翻译: 提供左旋多巴二甲基取代的二酯前药药物,包含左旋多巴二甲基取代的二酯前药的组合物,以及使用这些前药和药物组合物治疗疾病如帕金森病的方法。
-
公开(公告)号:US07019003B2
公开(公告)日:2006-03-28
申请号:US10469433
申请日:2002-03-01
IPC分类号: A61K31/535 , C07C271/00
CPC分类号: C07D295/192 , C07C243/32 , C07C243/38 , C07C281/02 , C07C281/06 , C07C2601/08 , C07C2601/14 , C07D295/13 , C07D295/215
摘要: Novel PDF inhibitors and novel methods for their use are provided.
-
-
-
-
-
-
-
-
-