公开(公告)号：US5192778A

公开(公告)日：1993-03-09

申请号：US677030

申请日：1991-03-29

申请人： Kenji Kodaka ,  Katsutoshi Kinoshita ,  Michihiko Nakaya ,  Koichi Ebihara ,  Shirou Shiraishi ,  Eiichi Yamada ,  Satoshi Numata

发明人： Kenji Kodaka ,  Katsutoshi Kinoshita ,  Michihiko Nakaya ,  Koichi Ebihara ,  Shirou Shiraishi ,  Eiichi Yamada ,  Satoshi Numata

IPC分类号： C07D401/06 ,  C07D405/14 ,  C07D417/06 ,  C07D417/14

CPC分类号： C07D401/06 ,  C07D405/14 ,  C07D417/06 ,  C07D417/14

摘要： Novel dialkoxymethylimidazolidine derivatives of the formula (1) ##STR1## are described. Also, a preparation process of the derivatives and insecticidal compositions comprising the same are set forth. In addition, novel intermediate compounds of the formula (2) useful in preparing the derivatives of the formula(1) are also described along with their preparation process ##STR2##

公开(公告)号：US5264584A

公开(公告)日：1993-11-23

申请号：US944687

申请日：1992-09-14

申请人： Kenji Kodaka ,  Katsutoshi Kinoshita ,  Michihiko Nakaya ,  Koichi Ebihara ,  Shirou Shiraishi ,  Eiichi Yamada ,  Satoshi Numata

发明人： Kenji Kodaka ,  Katsutoshi Kinoshita ,  Michihiko Nakaya ,  Koichi Ebihara ,  Shirou Shiraishi ,  Eiichi Yamada ,  Satoshi Numata

IPC分类号： C07D401/06 ,  C07D405/14 ,  C07D417/06 ,  C07D417/14 ,  C07D233/52

CPC分类号： C07D401/06 ,  C07D405/14 ,  C07D417/06 ,  C07D417/14

摘要： Novel dialkoxymethylimidazolidine derivatives of the formula (1) ##STR1## are described. Also, a preparation process of the derivatives and insecticidal compositions comprising the same are set forth. In addition, novel intermediate compounds of the formula (2) useful in preparing the derivatives of the formula (1) are also described along with their preparation process ##STR2##

摘要翻译： 描述了式（1）的新型二烷氧基甲基咪唑烷衍生物（1）。 另外，提出了包含它们的衍生物和杀虫组合物的制备方法。 此外，还描述了可用于制备式（1）的衍生物的式（2）的新型中间体化合物及其制备方法。

公开(公告)号：US5219868A

公开(公告)日：1993-06-15

申请号：US802092

申请日：1991-12-04

申请人： Kenji Kodaka ,  Katsutoshi Kinoshita ,  Michihiko Nakaya ,  Koichi Ebihara ,  Shirou Shiraishi ,  Eiichi Yamada ,  Satoshi Numata

发明人： Kenji Kodaka ,  Katsutoshi Kinoshita ,  Michihiko Nakaya ,  Koichi Ebihara ,  Shirou Shiraishi ,  Eiichi Yamada ,  Satoshi Numata

IPC分类号： A01N43/50 ,  C07D233/52 ,  C07D233/88 ,  C07D401/06

CPC分类号： C07D401/06 ,  C07D233/88

摘要： Herein disclosed are novel imidazolidine derivatives of the formula (I) and intermediates of the formula (II) ##STR1## wherein each R represents a hydrogen atom, an alkyl group having from 1 to 6 carbon atoms, a halogen atom, an alkoxy group having from 1 to 6 carbon atoms, a methylenedioxy group, an alkylthio group having from 1 to 4 carbon atoms, a haloalkyl group having from 1 to 2 carbon atoms, a haloalkoxy group having from 1 to 4 carbon atoms, an alkylcarbonyl group having from 1 to 6 carbon atoms, an alkoxycarbonyl.group having from 1 to 6 carbon atoms, a hydroxy group, a cyano group, a nitro group, an alkylamino group having from 1 to 8 carbon atoms, a phenyl group, a phenoxy group, a benzyl group or a halopyridylmethyloxy group, and n is an integer of from 1 to 3, ##STR2## wherein R and n have, respectively, the same meanings as defined above. Processes for preparing the compounds of the formulas (I) and (II) are also described. Moreover, insecticidal compositions comprising an effective amount of the derivative (I) are described.

公开(公告)号：US5614527A

公开(公告)日：1997-03-25

申请号：US447962

申请日：1995-05-23

申请人： Katsutoshi Kinoshita ,  Takeo Wakita ,  Kenji Kodaka ,  Hirozumi Matsuno ,  Kenichi Satoh ,  Shirou Shiraishi ,  Kazutomi Ohnuma ,  Eiichi Yamada ,  Naoko Yasui ,  Nobuyuki Kawahara ,  Koichi Ebihara ,  Michihiko Nakaya

发明人： Katsutoshi Kinoshita ,  Takeo Wakita ,  Kenji Kodaka ,  Hirozumi Matsuno ,  Kenichi Satoh ,  Shirou Shiraishi ,  Kazutomi Ohnuma ,  Eiichi Yamada ,  Naoko Yasui ,  Nobuyuki Kawahara ,  Koichi Ebihara ,  Michihiko Nakaya

IPC分类号： A01N43/50 ,  A01N43/54 ,  A01N51/00 ,  C07D405/06 ,  C07D251/08

CPC分类号： C07D405/06 ,  A01N51/00

摘要： A tetrahydrofuran-compound is disclosed herein which is represented by the formula (1) ##STR1## wherein each of X.sub.1 and X.sub.2 is a hydrogen atom or a methyl group, Y is a hydrogen atom or a carbonyl group substituted by a lower alkyl group (Y') having 1 to 4 carbon atoms, i.e., an acyl group (--COY'), andn is 2 or 3,and an insecticide containing the tetrahydrofuran-compound as an effective component.

摘要翻译： 本文公开的四氢呋喃化合物，其由式（1）表示：其中X1和X2各自为氢原子或甲基，Y为氢原子或被低级 具有1至4个碳原子的烷基（Y'），即酰基（-COY'），n为2或3，以及含有四氢呋喃化合物作为有效成分的杀虫剂。

公开(公告)号：US5434181A

公开(公告)日：1995-07-18

申请号：US326260

申请日：1994-10-20

申请人： Kenji Kodaka ,  Katsutoshi Kinoshita ,  Takeo Wakita ,  Shirou Shiraishi ,  Kazutomi Ohnuma ,  Eiichi Yamada ,  Naoko Yasui ,  Michihiko Nakaya ,  Hirozumi Matsuno ,  Nobuyuki Kawahara ,  Koichi Ebihara

发明人： Kenji Kodaka ,  Katsutoshi Kinoshita ,  Takeo Wakita ,  Shirou Shiraishi ,  Kazutomi Ohnuma ,  Eiichi Yamada ,  Naoko Yasui ,  Michihiko Nakaya ,  Hirozumi Matsuno ,  Nobuyuki Kawahara ,  Koichi Ebihara

IPC分类号： A01N43/08 ,  A01N43/36 ,  A01N47/12 ,  A01N47/40 ,  A01N51/00 ,  A01N53/00 ,  C07D307/14 ,  C07D405/06 ,  C07D307/16

CPC分类号： C07D405/06 ,  A01N43/08 ,  A01N43/36 ,  A01N47/40 ,  A01N51/00 ,  A01N53/00 ,  C07D307/14

摘要： The present invention relates to novel (tetrahydro-3-furanyl)methylamino derivatives of the following formula (1): ##STR1## wherein the variables are defined in the specification, which are useful as insecticides.

摘要翻译： 本发明涉及下式（1）的新的（四氢-3-呋喃基）甲基氨基衍生物：其中变量在本说明书中定义，其可用作杀虫剂。

公开(公告)号：US5532365A

公开(公告)日：1996-07-02

申请号：US417111

申请日：1995-04-05

申请人： Kenji Kodaka ,  Katsutoshi Kinoshita ,  Takeo Wakita ,  Shirou Shiraishi ,  Kazutomi Ohnuma ,  Eiichi Yamada ,  Naoko Yasui ,  Michihiko Nakaya ,  Hirozumi Matsuno ,  Nobuyuki Kawahara ,  Koichi Ebihara

发明人： Kenji Kodaka ,  Katsutoshi Kinoshita ,  Takeo Wakita ,  Shirou Shiraishi ,  Kazutomi Ohnuma ,  Eiichi Yamada ,  Naoko Yasui ,  Michihiko Nakaya ,  Hirozumi Matsuno ,  Nobuyuki Kawahara ,  Koichi Ebihara

IPC分类号： A01N43/08 ,  A01N43/36 ,  A01N47/12 ,  A01N47/40 ,  A01N51/00 ,  A01N53/00 ,  C07D307/14 ,  C07D405/06 ,  C07D251/08

CPC分类号： C07D405/06 ,  A01N43/08 ,  A01N43/36 ,  A01N47/40 ,  A01N51/00 ,  A01N53/00 ,  C07D307/14

摘要： The present invention relates to novel (tetrahydro-3-furanyl)methylamino derivatives of the following formula (1): ##STR1## wherein the variables are defined in the specification, which are useful as insecticides.

摘要翻译： 本发明涉及下式（1）的新的（四氢-3-呋喃基）甲基氨基衍生物：其中变量在本说明书中定义，其可用作杀虫剂。

公开(公告)号：US5310920A

公开(公告)日：1994-05-10

申请号：US991051

申请日：1992-12-15

申请人： Kenji Kodaka ,  Michihiko Nakaya ,  Katsutoshi Kinoshita ,  Koichi Ebihara ,  Hirozumi Matsuno ,  Shirou Shiraishi ,  Kazutomi Ohnuma ,  Ei-ich Yamada

发明人： Kenji Kodaka ,  Michihiko Nakaya ,  Katsutoshi Kinoshita ,  Koichi Ebihara ,  Hirozumi Matsuno ,  Shirou Shiraishi ,  Kazutomi Ohnuma ,  Ei-ich Yamada

IPC分类号： A01N51/00 ,  C07D233/52 ,  C07D401/06 ,  C07D401/14 ,  C07D405/06 ,  C07D405/14 ,  C07D417/06 ,  A61K31/44

CPC分类号： C07D401/06 ,  A01N51/00 ,  C07D233/52 ,  C07D401/14 ,  C07D405/06 ,  C07D405/14 ,  C07D417/06

摘要： The present invention relates to novel N-vinylimidazolidine derivatives of the following formula (1), a process for producing them, an insecticide containing the derivatives as an effective ingredient, and novelintermediates. The derivatives (1) are useful as agricultural chemicals (particularly, as insecticides) in the fields of agriculture, and the intermediates are useful in various industrial fields, especially as intermediates for agricultural chemicals. ##STR1## where R.sup.1, R.sup.2, Z are as defined in the specification.

摘要翻译： 本发明涉及下述式（1）的新型N-乙烯基咪唑烷衍生物，其制造方法，含有该衍生物作为有效成分的杀虫剂和新型中间体。 衍生物（1）可用作农业领域的农药（特别是杀虫剂），中间体可用于各种工业领域，特别是作为农药的中间体。 （1）其中R1，R2，Z如说明书中所定义。

公开(公告)号：US5021412A

公开(公告)日：1991-06-04

申请号：US328398

申请日：1989-03-24

申请人： Michihiko Nakaya ,  Yukiharu Fukushi ,  Kenji Kodaka ,  Masayuki Ooka ,  Shirou Shiraishi ,  Masahiko Nakamura ,  Satoshi Numata

发明人： Michihiko Nakaya ,  Yukiharu Fukushi ,  Kenji Kodaka ,  Masayuki Ooka ,  Shirou Shiraishi ,  Masahiko Nakamura ,  Satoshi Numata

IPC分类号： A01N43/88 ,  A01N47/02 ,  C07D285/34 ,  C07D417/12

CPC分类号： C07D417/12 ,  A01N43/88 ,  A01N47/02 ,  C07D285/34

摘要： Novel tetrahydro-1,3,5-thiadiazin-4-ones of the following general formula (I) or their salts which are useful as an insecticidal and acaricidal agent. ##STR1## In the formula, each of R.sup.1 and R.sup.2 represents a halogen atom or a C.sub.1 -C.sub.4 alkyl group; R.sup.3 represents a halogen atom, a C.sub.1 -C.sub.4 alkyl group, a C.sub.3 -C.sub.6 cycloalkyl group, a C.sub.1 -C.sub.4 alkoxy group, an acetyl group, a phenoxy group, a halo-substituted phenoxy group, a benzyl group, a benzyloxy group, a phenylcarbonyl group, a C.sub.1 -C.sub.4 haloalkyloxy group, a C.sub.1 -C.sub.4 haloalkyloxymethyl group, a C.sub.2 -C.sub.4 haloalkenyloxy group, a C.sub.1 -C.sub.4 haloalkylthio group, a C.sub.1 -C.sub.4 haloalkylthiomethyl group, a C.sub.2 -C.sub.4 haloalkenylthio group, a C.sub.1 -C.sub.8 haloalkyl group, a C.sub.2 -C.sub.8 haloalkenyl group, a C.sub.1 -C.sub.8 alkyloxycarbonyl group, a substituted phenoxycarbonyl group, or a substituted pyridyloxy group; m represents 0, 1, 2 or 3; and n represents 0, 1, 2 or 3.These novel thiadiazines are produced by reacting a compound of general formula (II) ##STR2## wherein R.sup.1 and m are as defined above, with a compound of general formula (III) ##STR3## wherein R.sup.2, R.sup.3 and n are as defined above.

摘要翻译： 具有以下通式（I）的四氢-1,3,5-噻二嗪-4-酮或它们的盐可用作杀虫剂和杀螨剂。 （I）式中，R 1和R 2各自表示卤原子或C 1〜C 4烷基; R3表示卤素原子，C1-C4烷基，C3-C6环烷基，C1-C4烷氧基，乙酰基，苯氧基，卤素取代的苯氧基，苄基，苄氧基， 苯基羰基，C 1 -C 4卤代烷氧基，C 1 -C 4卤代烷氧基甲基，C 2 -C 4卤代烯氧基，C 1 -C 4卤代烷硫基，C 1 -C 4卤代烷硫基甲基，C 2 -C 4卤代链烯基硫基，C 1 -C 8 卤代烷基，C 2 -C 8卤代烯基，C 1 -C 8烷氧基羰基，取代的苯氧基羰基或取代的吡啶氧基; m表示0,1,2或3; 并且n表示0,1,2或3.这些新的噻二嗪通过使通式（II）的化合物（II）（其中R 1和m如上定义）与通式（III）的化合物反应制备， （III）其中R2，R3和n如上所定义。