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公开(公告)号:US20140045778A1
公开(公告)日:2014-02-13
申请号:US13733369
申请日:2013-01-03
发明人: Kimihiko GOTO , Ryo HORIKOSHI , Mariko TSUCHIDA , Kazuhiko OYAMA , Satoshi OMURA , Hiroshi TOMODA , Toshiaki SUNAZUKA
IPC分类号: A01N43/90
CPC分类号: A01N43/90
摘要: Disclosed is a composition for use as a pest control agent, comprising a compound represented by formula (I) or an agriculturally and horticulturally acceptable salt thereof as active ingredient and an agriculturally and horticulturally acceptable carrier:
摘要翻译: 公开了一种用作害虫控制剂的组合物,其包含式(I)表示的化合物或其农业和园艺可接受的盐作为活性成分和农业和园艺可接受的载体:
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公开(公告)号:US20170215422A1
公开(公告)日:2017-08-03
申请号:US15488944
申请日:2017-04-17
发明人: Masaaki MITOMI , Masayo SAKAI , Ryo HORIKOSHI , Yasumichi ONOZAKI , Satoshi NAKAMURA , Satoshi OMURA , Toshiaki SUNAZUKA , Tomoyasu HIROSE , Kazuro SHIOMI , Rokuro MASUMA
IPC分类号: A01N43/72 , C07C235/12 , C07C231/12 , C07C271/22 , C07D273/08 , C07C269/06 , C07B51/00 , C07K11/02 , C07D273/00
CPC分类号: A01N43/72 , C07B51/00 , C07C231/12 , C07C235/12 , C07C269/06 , C07C271/22 , C07D273/00 , C07D273/08 , C07K11/02
摘要: An objective of the present invention is to provide novel cyclic depsipeptide derivatives and harmful organism control agents including the same as each other. Specifically, the present invention provides compounds represented by formula (1) or stereoisomers thereof, harmful organism control agents containing them, and a process for producing them.
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公开(公告)号:US20210147448A1
公开(公告)日:2021-05-20
申请号:US17050747
申请日:2019-04-26
发明人: Toshio KANAI , Sachiko KOIKE , Takayuki FUKAYA , Shunichiro UESUGI , Shingo MIZUSHIMA , Hitoshi SUDA , Yuki MIZUKAMI , Yohei IKUMA , Toshiaki SUNAZUKA , Yoshihiko NOGUCHI
摘要: Provided is a novel compound that has an excellent β-lactamase inhibitory effect. More specifically, provided is a compound represented by formula (1a), (1b) or (11) having an excellent β-lactamase inhibitory effect or a pharmaceutically acceptable salt thereof. By using this compound either in combination with a β-lactam drug or alone, a useful preventive or therapeutic agent for bacterial infections is provided. Also provided are useful preventive or therapeutic agents for treating various diseases with the combined use of the aforesaid compound and β-lactam drugs.
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公开(公告)号:US20230287009A1
公开(公告)日:2023-09-14
申请号:US18309641
申请日:2023-04-28
发明人: Toshio KANAI , Sachiko KOIKE , Takayuki FUKAYA , Shunichiro UESUGI , Shingo MIZUSHIMA , Hitoshi SUDA , Yuki MIZUKAMI , Yohei IKUMA , Toshiaki SUNAZUKA , Yoshihiko NOGUCHI
IPC分类号: C07F5/02 , A61K45/06 , A61P31/04 , A61K31/407 , A61K31/69
CPC分类号: C07F5/025 , A61K45/06 , A61P31/04 , A61K31/407 , A61K31/69
摘要: Provided is a novel compound that has an excellent β-lactamase inhibitory effect. More specifically, provided is a compound represented by formula (1a), (1b) or (11) having an excellent β-lactamase inhibitory effect or a pharmaceutically acceptable salt thereof. By using this compound either in combination with a β-lactam drug or alone, a useful preventive or therapeutic agent for bacterial infections is provided. Also provided are useful preventive or therapeutic agents for treating various diseases with the combined use of the aforesaid compound and β-lactam drugs.
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公开(公告)号:US20210130315A1
公开(公告)日:2021-05-06
申请号:US16762068
申请日:2018-11-06
发明人: Dirk HEIMBACH , Satoshi OMURA , Toshiaki SUNAZUKA , Tomoyasu HIROSE , Yoshihiko NOGUCHI , Johannes KÖBBERLING , Zhijie WU , Shuibiao FU , Wei WU , Jinfeng QIU , Liu HE , Xudong WEI
IPC分类号: C07D325/00 , A61K38/15
摘要: The present invention relates to a method for the synthesis of cyclic depsipeptides, in particular emodepside, from the open form.
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