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公开(公告)号:US20180141947A1
公开(公告)日:2018-05-24
申请号:US15736510
申请日:2016-06-24
申请人: Meredeth Ann MCGOWAN , Hua ZHOU , Jason D. KATZ , Lihu YANG , Joey L. METHOT , Kathryn Ann LIPFORD , Shimin XU , Ning FU , Guoquan XU , Deqian BIAN , Jianmin FU , Yabin LI , kin Chiu FONG , MERCK SHARP & DOHME CORP.
发明人: Meredith Ann McGowan , Hua Zhou , Jason D. Katz , Lihu Yang , Joey L. Methot , Kathryn Ann Lipford , Shimin Xu , Ning Fu , Guoquan Xu , Deqian Bian , Jianmin Fu , Yabin Li , Kin Chiu Fong
IPC分类号: C07D473/30 , C07D473/34 , C07D519/00 , C07D471/04 , A61P35/00 , A61P19/02 , A61P11/06 , A61P11/00 , A61P37/00 , A61P17/06 , A61P11/08
CPC分类号: C07D473/30 , A61K45/06 , A61P11/00 , A61P11/06 , A61P11/08 , A61P17/06 , A61P19/02 , A61P35/00 , A61P37/00 , C07D471/04 , C07D473/34 , C07D519/00
摘要: The instant invention provides compounds of formula I which are PI3K-delta inhibitors, and as such are useful for the treatment of PI3K-delta-mediated diseases such as inflammation, asthma, COPD and cancer.
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公开(公告)号:US10221178B2
公开(公告)日:2019-03-05
申请号:US15736510
申请日:2016-06-24
发明人: Meredeth Ann McGowan , Hua Zhou , Jason D. Katz , Lihu Yang , Joey L. Methot , Kathryn Ann Lipford , Shimin Xu , Ning Fu , Guoquan Xu , Deqian Bian , Jianmin Fu , Yabin Li , Kin Chiu Fong
IPC分类号: C07D473/30 , C07D473/34 , C07D471/04 , C07D519/00 , A61K45/06 , A61P37/00 , A61P17/06 , A61P11/06 , A61P11/08 , A61P11/00 , A61P35/00
摘要: The instant invention provides compounds of formula I which are PI3K-delta inhibitors, and as such are useful for the treatment of PI3K-delta-mediated diseases such as inflammation, asthma, COPD and cancer.
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