专利检索 ap:("MIMETOGEN PHARMACEUTICALS, INC.") AND inv:"Martin Bohlin" 第 1 页

1.

发明授权
Solution phase synthesis of beta-turn peptidomimetic cyclic salts 有权

公开(公告)号：US11753441B2

公开(公告)日：2023-09-12

申请号：US17337383

申请日：2021-06-02

申请人： MIMETOGEN PHARMACEUTICALS, INC.

发明人： Sébastien Rocchi , Chantal Devin , Wei Tian , Martin Bohlin

IPC分类号： C07K1/02 , C07K5/10 , C07K5/113 , C07K1/30

CPC分类号： C07K5/1021 , C07K1/02 , C07K1/306 , C07K5/10 , C07K5/1027 , C07B2200/13

摘要： The present disclosure relates to methods of preparing and crystallizing β-turn cyclic peptidomimetic salts of formula I:

where R1, R2, R3, R4, R5, R6, R7, R8, R10, X, Y and n are as defined in the specification.

The present disclosure provides a more efficient route for preparing a crystalline form of a β-turn cyclic peptidomimetic compounds and salts thereof.

2.

发明申请
SOLUTION PHASE SYNTHESIS OF BETA-TURN PEPTIDOMIMETIC CYCLIC SALTS 有权

公开(公告)号：US20210300966A1

公开(公告)日：2021-09-30

申请号：US17337383

申请日：2021-06-02

申请人： MIMETOGEN PHARMACEUTICALS, INC.

发明人： Sébastien Rocchi , Chantal Devin , Wei Tian , Martin Bohlin

IPC分类号： C07K5/113 , C07K1/30 , C07K1/02 , C07K5/10

摘要： The present disclosure relates to methods of preparing and crystallizing β-turn cyclic peptidomimetic salts of formula I: where R1, R2, R3, R4, R5, R6, R7, R8, R10, X, Y and n are as defined in the specification.
The present disclosure provides a more efficient route for preparing a crystalline form of a β-turn cyclic peptidomimetic compounds and salts thereof.

3.

发明申请
SOLUTION PHASE SYNTHESIS AND CRYSTALLIZATION OF BETA-TURN PEPTIDOMIMETIC CYCLIC SALTS 审中-公开

公开(公告)号：US20190194251A1

公开(公告)日：2019-06-27

申请号：US16184485

申请日：2018-11-08

申请人： MIMETOGEN PHARMACEUTICALS, INC.

发明人： Sébastien Rocchi , Chantal Devin , Wei Tian , Martin Bohlin

IPC分类号： C07K5/113 , C07K5/10 , C07K1/02 , C07K1/30

CPC分类号： C07K5/1021 , C07B2200/13 , C07K1/02 , C07K1/306 , C07K5/1027

摘要： The present disclosure relates to methods of preparing and crystallizing β-turn cyclic peptidomimetic salts of formula I: where R1, R2, R3, R4, R5, R6, R7, R8, R10, X, Y and n are as defined in the specification.The present disclosure provides a more efficient route for preparing a crystalline form of β-turn cyclic peptidomimetic compounds and salts thereof.

4.

发明授权
Solution phase synthesis and crystallization of beta-turn peptidomimetic cyclic salts 有权

公开(公告)号：US10125165B2

公开(公告)日：2018-11-13

申请号：US15205909

申请日：2016-07-08

申请人： Mimetogen Pharmaceuticals, Inc.

发明人： Sébastien Rocchi , Chantal Devin , Wei Tian , Martin Bohlin

IPC分类号： A61K38/12 , C07K5/00 , C07K7/00 , C07K16/00 , C07K17/00 , C07K5/113 , C07K1/30 , C07K1/02 , C07K5/10

摘要： The present disclosure relates to methods of preparing and crystallizing β-turn cyclic peptidomimetic salts of formula I: where R1, R2, R3, R4, R5, R6, R7, R8, R10, X, Y and n are as defined in the specification. The present disclosure provides a more efficient route for preparing a crystalline form of β-turn cyclic peptidomimetic compounds and salts thereof.

5.

发明申请
SOLUTION PHASE SYNTHESIS AND CRYSTALLIZATION OF BETA-TURN PEPTIDOMIMETIC CYCLIC SALTS 审中-公开
标题翻译：解决方案相位合成和结晶形式的BETA-TURN PEPTIDOMMIC循环盐

公开(公告)号：US20170008923A1

公开(公告)日：2017-01-12

申请号：US15205909

申请日：2016-07-08

申请人： Mimetogen Pharmaceuticals, Inc.

发明人： Sébastien Rocchi , Chantal Devin , Wei Tian , Martin Bohlin

IPC分类号： C07K5/113

CPC分类号： C07K5/1021 , C07B2200/13 , C07K1/02 , C07K1/306 , C07K5/1027

摘要： The present disclosure relates to methods of preparing and crystallizing β-turn cyclic peptidomimetic salts of formula I: where R1, R2, R3, R4, R5, R6, R7, R8, R10, X, Y and n are as defined in the specification. The present disclosure provides a more efficient route for preparing a crystalline form of β-turn cyclic peptidomimetic compounds and salts thereof.

摘要翻译： 本公开内容提供了制备β-袢环肽模拟化合物及其盐的结晶形式的更有效的途径。

6.

发明公开
SOLUTION PHASE SYNTHESIS OF BETA-TURN PEPTIDOMIMETIC CYCLIC SALTS 审中-公开

公开(公告)号：US20230357318A1

公开(公告)日：2023-11-09

申请号：US18354076

申请日：2023-07-18

申请人： MIMETOGEN PHARMACEUTICALS, INC.

发明人： Sébastien Rocchi , Chantal Devin , Wei Tian , Martin Bohlin

IPC分类号： C07K5/113 , C07K1/30 , C07K1/02 , C07K5/10

CPC分类号： C07K5/1021 , C07K1/306 , C07K1/02 , C07K5/1027 , C07K5/10 , C07B2200/13

摘要： The present disclosure relates to methods of preparing and crystallizing β-turn cyclic peptidomimetic salts of formula I:

where R1, R2, R3, R4, R5, R6, R7, R8, R10, X, Y and n are as defined in the specification.

The present disclosure provides a more efficient route for preparing a crystalline form of a β-turn cyclic peptidomimetic compounds and salts thereof.

7.

发明授权
Solution phase synthesis and crystallization of beta-turn peptidomimetic cyclic salts 有权

公开(公告)号：US11078234B2

公开(公告)日：2021-08-03

申请号：US16184485

申请日：2018-11-08

申请人： MIMETOGEN PHARMACEUTICALS, INC.

发明人： Sébastien Rocchi , Chantal Devin , Wei Tian , Martin Bohlin

IPC分类号： C07K1/02 , C07K1/30 , C07K5/10 , C07K5/113

摘要： The present disclosure relates to methods of preparing and crystallizing β-turn cyclic peptidomimetic salts of formula I: where R1, R2, R3, R4, R5, R6, R7, R8, R10, X, Y and n are as defined in the specification. The present disclosure provides a more efficient route for preparing a crystalline form of β-turn cyclic peptidomimetic compounds and salts thereof.