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公开(公告)号:US20120220577A1
公开(公告)日:2012-08-30
申请号:US13375954
申请日:2010-06-04
申请人: Markus Henrich , Angela Hansen , Jens Nagel , Valerjans Kauss , Jevgenijs Rozhkovs , Ginta Grunsteine , Dina Trifanova
发明人: Markus Henrich , Angela Hansen , Jens Nagel , Valerjans Kauss , Jevgenijs Rozhkovs , Ginta Grunsteine , Dina Trifanova
IPC分类号: A61K31/19 , C07C271/22 , A61K31/27 , C07D211/60 , A61K31/445 , C07D207/08 , A61K31/40 , C07D215/14 , A61K31/47 , C07D265/36 , A61K31/538 , C07D265/30 , A61K31/5375 , C07D257/04 , A61K31/41 , A61P29/00 , A61P25/02 , C07C63/34
CPC分类号: C07C311/51 , C07C49/84 , C07C65/24 , C07C235/20 , C07C235/22 , C07C235/24 , C07C237/42 , C07C255/16 , C07C255/44 , C07C255/60 , C07C271/20 , C07C2601/02 , C07C2602/08 , C07C2602/10 , C07D207/16 , C07D207/273 , C07D209/42 , C07D211/60 , C07D213/36 , C07D213/50 , C07D213/74 , C07D215/06 , C07D215/48 , C07D217/02 , C07D217/26 , C07D233/90 , C07D257/04 , C07D257/06 , C07D265/36 , C07D277/42 , C07D295/185 , C07D307/85 , C07D403/04 , C07D513/04
摘要: The invention relates to naphthalene derivatives as well as their pharmaceutically acceptable salts. The invention further relates to a process for the preparation of such compounds. The compounds of the invention are glycine B antagonists and are therefore useful for the control and prevention of various disorders, including neurological disorders.
摘要翻译: 本发明涉及萘衍生物及其药学上可接受的盐。 本发明还涉及制备这些化合物的方法。 本发明的化合物是甘氨酸B拮抗剂,因此可用于控制和预防各种疾病,包括神经障碍。