公开(公告)号：US4874861A

公开(公告)日：1989-10-17

申请号：US127518

申请日：1987-11-30

申请人： Tomoyuki Ogura ,  Yasuo Kawamura ,  Shigeru Ishii ,  Masatoshi Baba ,  Masakazu Taniguchi ,  Masayoshi Hirose ,  Kiminori Hirata ,  Yoshinori Ochiai

发明人： Tomoyuki Ogura ,  Yasuo Kawamura ,  Shigeru Ishii ,  Masatoshi Baba ,  Masakazu Taniguchi ,  Masayoshi Hirose ,  Kiminori Hirata ,  Yoshinori Ochiai

IPC分类号： A01N43/58 ,  A01N55/00 ,  C07D237/14 ,  C07D237/16 ,  C07D237/18 ,  C07D401/12 ,  C07D403/12 ,  C07F7/08

CPC分类号： C07D401/12 ,  A01N43/58 ,  A01N55/00 ,  C07D237/14 ,  C07D237/16 ,  C07D237/18 ,  C07D403/12 ,  C07F7/0812

摘要： Novel 3(2H)-pyridazinone derivatives having the general formula (I): ##STR1## wherein, R denotes a straight or branched C.sub.1 to C.sub.6 alkyl; A denotes a straight or branched C.sub.1 to C.sub.6 alkyl or a halogen; X denotes oxygen or sulfur atom; Q denotes a group; ##STR2## when A is a straight or branched C.sub.1 to C.sub.6 alkyl, and Q denotes a group: ##STR3## when A is a halogen atom; R.sup.1 and R.sup.2 denote each independently hydrogen, a lower alkyl, a lower haloalkyl, or 4-tert-butylphenyl; B denotes --CR.sup.6 .dbd.CR.sup.7 --, --CR.sup.6 R.sup.7 O--, or ##STR4## (wherein, R.sup.6 and R.sup.7 denote various specific organic radicals. A process for preparation of said derivatives is also provided. These derivatives are useful as an active ingredient of insecticidal, acaricidal, nematicidal and/or fungicidal compositions for agricultural and horticultural uses as well as of expellent compositions for ticks parasitic on animals.

摘要翻译： 具有通式（I）的新型3（2H） - 哒嗪酮衍生物：其中R表示直链或支链C 1至C 6烷基; A表示直链或支链C1至C6烷基或卤素; X表示氧或硫原子; Q表示一组; 当A为直链或支链C 1至C 6烷基时，并且Q表示基团：当A为卤素原子时： R 1和R 2各自独立地表示氢，低级烷基，低级卤代烷基或4-叔丁基苯基; B表示-CR6 = CR7-，-CR6R7O-或（其中，R6和R7表示各种特定的有机基团，也提供了所述衍生物的制备方法，这些衍生物可用作杀虫， 用于农业和园艺用途的杀螨，杀线虫和/或杀真菌组合物以及寄生在动物上的蜱的驱虫剂组合物。

公开(公告)号：US4571397A

公开(公告)日：1986-02-18

申请号：US467259

申请日：1983-02-17

申请人： Masakazu Taniguchi ,  Masatoshi Baba ,  Yoshinori Ochiai ,  Masayoshi Hirose ,  Kiminori Hirata

发明人： Masakazu Taniguchi ,  Masatoshi Baba ,  Yoshinori Ochiai ,  Masayoshi Hirose ,  Kiminori Hirata

IPC分类号： C07D237/16 ,  A01N20060101 ,  A01N43/58 ,  A01N55/00 ,  C07D20060101 ,  C07F7/08 ,  C07D237/06 ,  A61K31/50

CPC分类号： A01N55/00 ,  A01N43/58 ,  C07D237/16 ,  C07F7/0812

摘要： Novel 5-substituted -3(2H)-pyridazinone derivatives and preparation thereof are provided.The derivatives have the formula: ##STR1## wherein, R denotes an alkyl, R.sup.1 and R.sup.2 denote each independently hydrogen or a lower alkyl, X denotes hydrogen, a lower alkyl, a halogen, a lower alkoxy, a lower haloalkyl, a lower haloalkoxy, a cycloalkyl, trimethylsilyl (-Si(CH.sub.3).sub.3), ##STR2## (wherein Y denotes hydrogen, a halogen, a lower alkyl, a lower alkoxy, a lower haloalkyl, a lower haloalkoxy or a cycloalkyl, and m is an integer of 1 to 5), n is an integer of 1 to 5, and Z denotes a halogen; said X being the same or different when n is 2 or more, and the alkyls and the alkyl moieties contained in the groups being straight or branched.

摘要翻译： 提供新的5-取代-3（2H） - 哒嗪酮衍生物及其制备。 衍生物具有下式：其中R表示烷基，R 1和R 2各自独立地表示氢或低级烷基，X表示氢，低级烷基，卤素，低级烷氧基，低级卤代烷基， 低级卤代烷氧基，环烷基，三甲基甲硅烷基（-Si（CH 3）3），其中Y表示氢，卤素，低级烷基，低级烷氧基，低级卤代烷基，低级卤代烷氧基或环烷基，m 为1〜5的整数），n为1〜5的整数，Z为卤素。 当n为2或更多时，所述X相同或不同，并且所述基团中所含的烷基和烷基部分是直链或支链的。

公开(公告)号：US4877787A

公开(公告)日：1989-10-31

申请号：US27191

申请日：1987-03-17

申请人： Masakazu Taniguchi ,  Masayoshi Hirose ,  Masatoshi Baba ,  Kiminori Hirata ,  Yoshinori Ochiai

发明人： Masakazu Taniguchi ,  Masayoshi Hirose ,  Masatoshi Baba ,  Kiminori Hirata ,  Yoshinori Ochiai

IPC分类号： A01N43/58 ,  A01P7/02 ,  A01P7/04 ,  C07D237/18 ,  C07D401/12 ,  C07D403/12 ,  C07F7/08

CPC分类号： C07D401/12 ,  A01N43/58 ,  C07D237/18 ,  C07D403/12 ,  C07F7/0812

摘要： Novel 3(2H)-pyridazinone derivatives having the formula I: ##STR1## wherein, R is a straight or branched C.sub.2 to C.sub.6 alkyl, R.sup.1 and R.sup.2 are each independently hydrogen or a lower alkyl, R.sup.4 is a halogen, R.sup.3 is a halogen, an alkyl, a cycloalkyl, an alkoxy, a haloalkyl, a haloalkoxy, --CN, --NO.sub.2, a phenyl, a benzyloxy, a benzyl, a phenoxy, a phenylthio, a pyridyloxy, a quinoxalyloxy, a lower alkenyloxy, a lower alkylthio, a lower haloalkylthio, --Si(CH.sub.3).sub.3, --OH, --N(CH.sub.3).sub.2, --SCN, --COOCH.sub.3 or --OCH(CH.sub.3)COOC.sub.2 H.sub.5, and n is an integer of 1 to 5, said R.sup.3 being the same or different when n is an integer of 2 to 5. A process for preparation of said derivatives is also provided. These derivatives are useful as an active ingredient of insecticidal, acaricidal, nematicidal and/or fungicidal compositions for agricultural and horticultural uses as well as of expellent compositions for ticks parasitic on animals.

摘要翻译： 具有式I的新型3（2H） - 哒嗪酮衍生物：其中R是直链或支链C 2至C 6烷基，R 1和R 2各自独立地是氢或低级烷基，R 4是卤素，R 3 是卤素，烷基，环烷基，烷氧基，卤代烷基，卤代烷氧基，-CN，-NO 2，苯基，苄氧基，苄基，苯氧基，苯硫基，吡啶氧基，喹喔啉氧基，低级烯氧基， 低级烷硫基，低级卤代烷硫基，-Si（CH3）3，-OH，-N（CH3）2，-SCN，-COOCH3或-OCH（CH3）COOC2H5，n为1〜5的整数，R3 当n为2〜5的整数时，其相同或不同。还提供了制备所述衍生物的方法。 这些衍生物可用作农业和园艺用途的杀虫，杀螨，杀线虫和/或杀真菌组合物的活性成分，以及用于动物寄生的蜱的驱虫剂组合物。

公开(公告)号：US5026850A

公开(公告)日：1991-06-25

申请号：US362348

申请日：1989-06-06

申请人： Masakazu Taniguchi ,  Masatoshi Baba ,  Yoshinori Ochiai ,  Masayoshi Hirose ,  Kiminori Hirata

发明人： Masakazu Taniguchi ,  Masatoshi Baba ,  Yoshinori Ochiai ,  Masayoshi Hirose ,  Kiminori Hirata

IPC分类号： A01N43/58 ,  A01P7/02 ,  A01P7/04 ,  C07D237/18 ,  C07D401/12 ,  C07D403/12 ,  C07F7/08

CPC分类号： C07D401/12 ,  A01N43/58 ,  C07D237/18 ,  C07D403/12 ,  C07F7/0812

摘要： Compounds of the formula: ##STR1## wherein R is a member selected from the group consisting of lower alkyls having from 2 to 4 carbon atoms; and chlorine and bromine. The compounds are useful as active ingredients in, e.g., insecticidal, acaricidal, nematicidal, fungicidal and expellant compositions.

公开(公告)号：US4837217A

公开(公告)日：1989-06-06

申请号：US850533

申请日：1986-04-11

申请人： Tomoyuki Ogura ,  Yasuo Kawamura ,  Masatoshi Baba ,  Shigeru Ishii ,  Kiminori Hirata ,  Masaki Kudo ,  Yoshinori Ochiai ,  Masayoshi Hirose

发明人： Tomoyuki Ogura ,  Yasuo Kawamura ,  Masatoshi Baba ,  Shigeru Ishii ,  Kiminori Hirata ,  Masaki Kudo ,  Yoshinori Ochiai ,  Masayoshi Hirose

IPC分类号： A01N43/58 ,  C07D237/16 ,  C07D237/18 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12

CPC分类号： C07D401/12 ,  A01N43/58 ,  C07D237/16 ,  C07D237/18 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12

摘要： A 3(2H)-pyridazinone derivative of the general formula (I): ##STR1## wherein R is a straight or branched C.sub.2 -C.sub.6 alkyl,A is a straight or branched C.sub.1 -C.sub.6 alkyl or a halogen atom,X is --O-- or --S--,R.sup.1 and R.sup.2 are each independently hydrogen atom or C.sub.1 -C.sub.3 alkyl,B is --CH.dbd.CH--, --N.dbd.CH--, --N.dbd.N--, --S--, --O-- or ##STR2## wherein R.sup.3 is hydrogen or C.sub.1 -C.sub.3 alkyl, Y is a halogen atom, a straight or branched C.sub.1 -C.sub.6 alkyl, a C.sub.3 -C.sub.6 cycloalkyl or cycloalkoxy, and other substituents,n is 0 or an integer of 1 to 3, and when n is 2 or 3, Y may be same or different, with the proviso that when B is --CH.dbd.CH--, n is an integer of 1 to 3 and at least one of Y is --O--W, as this term is defined in the specification.A process for the preparation of said derivatives is also provided. These derivatives are useful as an active ingredient of insecticidal, acaricidal, nematicidal and/or fungicidal compositions for agricultural and horticultural uses as well as of expellent compositions for ticks parasitic on animals.

摘要翻译： 通式（I）的3（2H） - 哒嗪酮衍生物：其中R是直链或支链C 2 -C 6烷基，A是直链或支链C 1 -C 6烷基或卤素原子，X是-O - 或-S-，R1和R2各自独立地为氢原子或C1-C3烷基，B为-CH = CH-，-N = CH-，-N = N-，-S-，-O-或

公开(公告)号：US4908379A

公开(公告)日：1990-03-13

申请号：US185992

申请日：1988-04-25

申请人： Yasuyuki Nakajima ,  Takahiro Makabe ,  Kazunari Nakayama ,  Tatsuo Numata ,  Kiminori Hirata ,  Masaki Kudo ,  Yoshinori Ochiai ,  Masayoshi Hirose

发明人： Yasuyuki Nakajima ,  Takahiro Makabe ,  Kazunari Nakayama ,  Tatsuo Numata ,  Kiminori Hirata ,  Masaki Kudo ,  Yoshinori Ochiai ,  Masayoshi Hirose

IPC分类号： A01N43/40 ,  A01N43/54 ,  A01N43/64 ,  A01N43/707 ,  A01N43/90 ,  C07D239/52 ,  C07D239/54 ,  C07D239/553 ,  C07D239/56 ,  C07D239/58 ,  C07D239/60 ,  C07D251/20 ,  C07D251/38 ,  C07D253/075 ,  C07D401/12 ,  C07D471/04 ,  C07D487/04 ,  C07D498/04 ,  C07D513/04

CPC分类号： C07D239/553 ,  A01N43/40 ,  A01N43/54 ,  A01N43/64 ,  A01N43/707 ,  A01N43/90 ,  C07D239/52 ,  C07D239/56 ,  C07D239/60 ,  C07D251/20 ,  C07D251/38 ,  C07D253/075 ,  C07D401/12 ,  C07D471/04 ,  C07D487/04 ,  C07D513/04

摘要： A nitrogen-containing heterocyclic compound of the following formula: ##STR1## wherein D represents --N.dbd. or ##STR2## E represents .dbd.N--, ##STR3## G represents --N.dbd., ##STR4## with proviso that when G represents --N.dbd. or ##STR5## the bond of G and E is double bond; and G represents ##STR6## the bond thereof is a single bond, but the case that D represents ##STR7## E represents ##STR8## and G represents --N.dbd. is omitted (R.sup.1, R.sup.2, R.sup.9, R.sup.10, X, Y, A and Q are specified in the specification), as well as compositions for controlling and/or preventing pests and blights, said compositions containing one or two or more of said compounds as an active ingredient.

公开(公告)号：US4906627A

公开(公告)日：1990-03-06

申请号：US191260

申请日：1988-05-06

申请人： Yasuyuki Nakajima ,  Yasuo Kawamura ,  Tomoyuki Ogura ,  Takahiro Makabe ,  Kiminori Hirata ,  Masaki Kudo ,  Yoshinori Ochiai ,  Masayoshi Hirose

发明人： Yasuyuki Nakajima ,  Yasuo Kawamura ,  Tomoyuki Ogura ,  Takahiro Makabe ,  Kiminori Hirata ,  Masaki Kudo ,  Yoshinori Ochiai ,  Masayoshi Hirose

IPC分类号： C07D237/14 ,  A01N25/30 ,  A01N43/58 ,  A01N43/60 ,  A01P7/02 ,  C07D237/16 ,  C07D237/18 ,  C07D401/12 ,  C07D403/12

CPC分类号： C07D401/12 ,  A01N43/58 ,  A01N43/60 ,  C07D237/16 ,  C07D237/18 ,  C07D403/12

摘要： Compounds of the following formula: ##STR1## wherein Z.sup.3 represents halogen atom, straight or branched chain alkyl group having 1 to 10 carbon atoms, alkoxy group having 1 to 10 carbon atoms, alkylcarbonyl having 2 to 10 carbon atoms, alkoxyalkyl group having 2 to 4 carbon atoms, ##STR2## W represents halogen atom, alkyl group having 1 to 4 carbon atoms, alkoxy group having 1 to 4 carbon atoms, haloalkyl group having 1 to 4 carbon atoms, or nitro group, m is 0 or an integer of 1 to 2, and when m is 2, W may be same or different, and compositions for controlling insects, acari and nemati which contain such compound.

摘要翻译： 下式的化合物：其中Z 3表示卤素原子，碳原子数1〜10的直链或支链烷基，碳原子数1〜10的烷氧基，碳原子数2〜10的烷基羰基，烷氧基烷基，具有2〜 4个碳原子，W表示卤原子，碳原子数1〜4的烷基，碳原子数1〜4的烷氧基，碳原子数1〜4的卤代烷基或硝基，m表示 0或1〜2的整数，当m为2时，W可以相同也可以不同，也可以是用于控制含有该化合物的昆虫，螨和螨的组合物。

公开(公告)号：US4425343A

公开(公告)日：1984-01-10

申请号：US267077

申请日：1981-05-26

申请人： Gojyo Sakata ,  Kenji Makino ,  Yasuo Kawamura ,  Jun Sato ,  Kiyomi Ozawa ,  Masayoshi Hirose ,  Kiminori Hirata

发明人： Gojyo Sakata ,  Kenji Makino ,  Yasuo Kawamura ,  Jun Sato ,  Kiyomi Ozawa ,  Masayoshi Hirose ,  Kiminori Hirata

IPC分类号： A01N47/34 ,  C07D215/22 ,  C07D215/227 ,  C07D215/36 ,  C07D241/44 ,  A61K31/47 ,  A61K31/495

CPC分类号： C07D215/227 ,  A01N47/34 ,  C07D215/36 ,  C07D241/44

摘要： This invention relates to a heterocyclic ether or thioether linkage containing urea compounds of the following formula I: ##STR1## wherein B denotes an oxygen atom or a sulfur atom, A denotes CH or a nitrogen atom, X.sup.1 and X.sup.2 denote independently of each other hydrogen atom, halogen atom, trifluoromethyl group or nitro group, Y and Z denote independently of each other hydrogen atom or halogen atom, and P and Q denote independently of each other hydrogen atom, halogen atom, alkoxyl group or alkyl group, a process for producing the same and an insecticide containing the same.

摘要翻译： 本发明涉及含有下式I的脲化合物的杂环醚或硫醚键：其中B表示氧原子或硫原子，A表示CH或氮原子，X1和X2独立地表示 氢原子，卤原子，三氟甲基或硝基，Y和Z彼此独立地表示氢原子或卤素原子，P和Q彼此独立地表示氢原子，卤素原子，烷氧基或烷基， 其制造方法和含有该杀虫剂的杀虫剂。

公开(公告)号：US4255447A

公开(公告)日：1981-03-10

申请号：US65340

申请日：1979-08-09

申请人： Kiyomi Ozawa ,  Shigeru Ishii ,  Mamoru Hayashi ,  Masayoshi Hirose ,  Kiminori Hirata

发明人： Kiyomi Ozawa ,  Shigeru Ishii ,  Mamoru Hayashi ,  Masayoshi Hirose ,  Kiminori Hirata

IPC分类号： C07C253/00 ,  A01N53/00 ,  A01N53/08 ,  C07C67/00 ,  C07C255/39 ,  C07C121/75

CPC分类号： A01N53/00

摘要： Phenylcyclopropane carboxylic acid derivatives having the formula (I) ##STR1## wherein X represents a C.sub.2 -C.sub.10 straight or branched alkyl group, are novel compounds having excellent acaricidal effect.

摘要翻译： 具有式（I）的苯基环丙烷羧酸衍生物（I）其中X表示C2-C10直链或支链烷基，是具有优异杀螨效果的新型化合物。

公开(公告)号：US4462994A

公开(公告)日：1984-07-31

申请号：US376639

申请日：1982-05-10

申请人： Gojyo Sakata ,  Tatsuo Numata ,  Kazuya Kusano ,  Masayoshi Hirose ,  Kiminori Hirata

发明人： Gojyo Sakata ,  Tatsuo Numata ,  Kazuya Kusano ,  Masayoshi Hirose ,  Kiminori Hirata

IPC分类号： A01N57/16 ,  C07F9/60 ,  C07F9/6509 ,  C07F9/18

CPC分类号： C07F9/60 ,  A01N57/16 ,  C07F9/650994

摘要： Novel N-containing heterocyclic ring-substituted O-arylphosphate derivatives, the preparation thereof and insecticides acaricides and nematicides containing said derivatives are provided. The O-arylphosphate derivatives have the general formula: ##STR1## wherein A is --CH or nitrogen, X is hydrogen, a halogen or trifluoromethyl; Y is oxygen, S(O)n (wherein n is an integer of from 0 to 2) or NR.sup.2 (wherein R.sup.2 is hydrogen or a lower alkyl); Z is oxygen or sulfur; R and R.sup.1 independently are a lower alkoxy or lower alkylthiol; and B is hydrogen, a halogen or a lower alkyl. The O-arylphosphate derivatives have an excellent insecticidal acaricidal and nematocidal action.

摘要翻译： 提供新型含氮杂环环取代的O-芳基磷酸酯衍生物，其制备方法和杀虫剂杀螨剂和含有所述衍生物的杀线虫剂。 O-芳基磷酸酯衍生物具有以下通式：其中A是-CH或氮，X是氢，卤素或三氟甲基; Y是氧，S（O）n（其中n是0-2的整数）或NR2（其中R2是氢或低级烷基）; Z是氧或硫; R和R 1独立地是低级烷氧基或低级烷基硫醇; 和B是氢，卤素或低级烷基。 O-芳基磷酸酯衍生物具有优良的杀虫杀螨和杀线虫作用。