Benzylthio pyridazinone derivatives, preparation thereof, and
insecticidal acaricidal, fungicidal compositions
    8.
    发明授权
    Benzylthio pyridazinone derivatives, preparation thereof, and insecticidal acaricidal, fungicidal compositions 失效
    苄硫基哒嗪酮衍生物,其制备和杀虫杀螨,杀真菌组合物

    公开(公告)号:US4877787A

    公开(公告)日:1989-10-31

    申请号:US27191

    申请日:1987-03-17

    摘要: Novel 3(2H)-pyridazinone derivatives having the formula I: ##STR1## wherein, R is a straight or branched C.sub.2 to C.sub.6 alkyl, R.sup.1 and R.sup.2 are each independently hydrogen or a lower alkyl, R.sup.4 is a halogen, R.sup.3 is a halogen, an alkyl, a cycloalkyl, an alkoxy, a haloalkyl, a haloalkoxy, --CN, --NO.sub.2, a phenyl, a benzyloxy, a benzyl, a phenoxy, a phenylthio, a pyridyloxy, a quinoxalyloxy, a lower alkenyloxy, a lower alkylthio, a lower haloalkylthio, --Si(CH.sub.3).sub.3, --OH, --N(CH.sub.3).sub.2, --SCN, --COOCH.sub.3 or --OCH(CH.sub.3)COOC.sub.2 H.sub.5, and n is an integer of 1 to 5, said R.sup.3 being the same or different when n is an integer of 2 to 5. A process for preparation of said derivatives is also provided. These derivatives are useful as an active ingredient of insecticidal, acaricidal, nematicidal and/or fungicidal compositions for agricultural and horticultural uses as well as of expellent compositions for ticks parasitic on animals.

    摘要翻译: 具有式I的新型3(2H) - 哒嗪酮衍生物:其中R是直链或支链C 2至C 6烷基,R 1和R 2各自独立地是氢或低级烷基,R 4是卤素,R 3 是卤素,烷基,环烷基,烷氧基,卤代烷基,卤代烷氧基,-CN,-NO 2,苯基,苄氧基,苄基,苯氧基,苯硫基,吡啶氧基,喹喔啉氧基,低级烯氧基, 低级烷硫基,低级卤代烷硫基,-Si(CH3)3,-OH,-N(CH3)2,-SCN,-COOCH3或-OCH(CH3)COOC2H5,n为1〜5的整数,R3 当n为2〜5的整数时,其相同或不同。还提供了制备所述衍生物的方法。 这些衍生物可用作农业和园艺用途的杀虫,杀螨,杀线虫和/或杀真菌组合物的活性成分,以及用于动物寄生的蜱的驱虫剂组合物。

    3(2H)-pyridazinone derivatives, and their uses in insecticidal
compositions
    9.
    发明授权
    3(2H)-pyridazinone derivatives, and their uses in insecticidal compositions 失效
    3(2H) - 哒嗪酮衍生物及其在杀虫组合物中的用途

    公开(公告)号:US4910201A

    公开(公告)日:1990-03-20

    申请号:US075725

    申请日:1987-07-20

    摘要: Novel 3(2H)-pyridazinone derivatives of the formula (I): ##STR1## wherein, X represents a halogen, an alkyl, a haloalkyl, a haloalkoxy atoms, NO.sub.2, an alkoxy or ##STR2## (wherein, R represents an alkyl); n is 1 to 4;A represents hydrogen, a halogen, an alkyl or an alkoxy;B represents CX.sub.1 (wherein, X.sub.1 represents H or a halogen) or N;R.sup.1 and R.sup.2 represent each independently H or an alkyl;E represents H, a halogen, an alkoxy or --OH; andQ represents: ##STR3## (wherein, Y represents a halogen, an alkyl, an alkoxy, a haloalkyl, a haloalkoxy, CN, ##STR4## (wherein, Z represents a halogen, an alkyl, an alkoxy or a haloalkyl atoms, and l is 0, 1 to 5, said Z being the same or different when l is 2 to 5); and m is 1 to 5, said Y being the same or different when n is 2 to 4. A process for preparation of said derivatives is also provided. These derivatives are useful as an active ingredient of insecticidal composition.

    摘要翻译: 式(I)的新型3(2H) - 哒嗪酮衍生物:其中X表示卤素,烷基,卤代烷基,卤代烷氧基,NO 2,烷氧基或(其中,R 表示烷基); n为1〜4; A表示氢,卤素,烷基或烷氧基; B表示CX1(其中,X1表示H或卤素)或N; R 1和R 2各自独立地表示氢或烷基; E表示H,卤素,烷氧基或-OH; 和Q表示:其中Y表示卤素,烷基,烷氧基,卤代烷基,卤代烷氧基,CN,其中Z表示 卤素,烷基,烷氧基或卤代烷基,l为0,1至5,当l为2至5时所述Z相同或不同); m为1至5,所述Y为相同或 n为2〜4时不同。还提供了制备所述衍生物的方法,这些衍生物可用作杀虫组合物的活性成分。