N-substituted phenylcarbamic acid derivatives, a process for production
thereof, agricultural and horticultural fungicides, intermediates of
the derivatives and a process for production thereof
    1.
    发明授权
    N-substituted phenylcarbamic acid derivatives, a process for production thereof, agricultural and horticultural fungicides, intermediates of the derivatives and a process for production thereof 失效
    N-取代苯基氨基甲酸衍生物,其制备方法,农业和园艺杀真菌剂,衍生物的中间体及其制备方法

    公开(公告)号:US5712399A

    公开(公告)日:1998-01-27

    申请号:US816969

    申请日:1997-03-13

    摘要: An N-substituted phenylcarbamic acid derivative represented by the general formula (I): ##STR1## �wherein R.sup.1 is H, a (C.sub.1-6)alkyl group, a halo(C.sub.1-6)alkyl group, a (C.sub.1-6)alkoxy(C.sub.1-6)alkyl group, a (C.sub.2-6)alkenyl group, a (C.sub.2-6)alkynyl group or a halo(C.sub.1-6)alkoxy(C.sub.1-6)alkyl group, R.sup.2 is H, a (C.sub.1-6)alkyl group, a halo(C.sub.1-6)alkyl group, a (C.sub.1-6)alkoxy(C.sub.1-6)alkyl group, a (C.sub.2-6)alkenyl group, a (C.sub.2-6)alkynyl group, a halo(C.sub.1-6)alkoxy(C.sub.1-6)alkyl group or a cyano(C.sub.1-6)alkyl group, R.sup.3 is a (C.sub.1-6)alkyl group or a halo(C.sub.1-6)alkyl group, each of R.sup.4 and R.sup.5 is a specific group, and Y is O or S! which is very effective in controlling powdery mildew, scab, late blight and gray mold; a process for producing said derivative; an agricultural and horticultural fungicide containing said derivative as an active ingredient; an intermediate of said derivative; and a process for producing the intermediate.

    摘要翻译: 由通式(I)表示的N-取代的苯基氨基甲酸衍生物:其中R1是H,(C1-6)烷基,卤代(C1-6)烷基,(C1 -6)烷氧基(C 1-6)烷基,(C 2-6)烯基,(C 2-6)炔基或卤代(C 1-6)烷氧基(C 1-6)烷基,R 2为H, (C 1-6)烷基,卤代(C 1-6)烷基,(C 1-6)烷氧基(C 1-6)烷基,(C 2-6)烯基,(C 2-6)炔基 基团,卤代(C 1-6)烷氧基(C 1-6)烷基或氰基(C 1-6)烷基,R 3为(C 1-6)烷基或卤代(C 1-6)烷基, R4和R5是一个特定的组,Y是O或S],这对控制白粉病,痂病,晚疫病和灰霉病非常有效; 一种制备所述衍生物的方法; 含有所述衍生物作为活性成分的农业和园艺杀真菌剂; 所述衍生物的中间体; 和中间体的制造方法。

    N-substituted phenylcarbamic acid derivatives, a process for production
thereof, agricultural and horticultural fungicides, intermediates of
the derivatives and a process for production thereof
    2.
    发明授权
    N-substituted phenylcarbamic acid derivatives, a process for production thereof, agricultural and horticultural fungicides, intermediates of the derivatives and a process for production thereof 失效
    N-取代苯基氨基甲酸衍生物,其制备方法,农业和园艺杀真菌剂,衍生物的中间体及其制备方法

    公开(公告)号:US5650434A

    公开(公告)日:1997-07-22

    申请号:US529048

    申请日:1995-09-15

    摘要: An N-substituted phenylcarbamic acid derivative represented by the general formula (I): ##STR1## [wherein R.sup.1 is H, a (C.sub.1-6)alkyl group, a halo(C.sub.1-6)alkyl group, a (C.sub.1-6)alkoxy(C.sub.1-6)alkyl group, a (C.sub.2-6)alkenyl group, a (C.sub.2-6)alkynyl group or a halo(C.sub.1-6)alkoxy(C.sub.1-6)alkyl group, R.sup.2 is H, a (C.sub.1-6)alkyl group, a halo(C.sub.1-6)alkyl group, a (C.sub.1-6)alkoxy(C.sub.1-6)alkyl group, a (C.sub.2-6)alkenyl group, a (C.sub.2-6)alkynyl group, a halo(C.sub.1-6)alkoxy(C.sub.1-6)alkyl group or a cyano(C.sub.1-6)alkyl group, R.sup.3 is a (C.sub.1-6)alkyl group or a halo(C.sub.1-6)alkyl group, each of R.sup.4 and R.sup.5 is a specific group, and Y is O or S] which is very effective in controlling powdery mildew, scab, late blight and gray mold; a process for producing said derivative; an agricultural and horticultural fungicide containing said derivative as an active ingredient; an intermediate of said derivative; and a process for producing the intermediate.

    摘要翻译: 由通式(I)表示的N-取代的苯基氨基甲酸衍生物:其中R1是H,(C1-6)烷基,卤代(C1-6)烷基,(C1 -6)烷氧基(C 1-6)烷基,(C 2-6)烯基,(C 2-6)炔基或卤代(C 1-6)烷氧基(C 1-6)烷基,R 2为H, (C 1-6)烷基,卤代(C 1-6)烷基,(C 1-6)烷氧基(C 1-6)烷基,(C 2-6)烯基,(C 2-6)炔基 基团,卤代(C 1-6)烷氧基(C 1-6)烷基或氰基(C 1-6)烷基,R 3为(C 1-6)烷基或卤代(C 1-6)烷基, R4和R5是一个特定的组,Y是O或S],这对控制白粉病,痂病,晚疫病和灰霉病非常有效; 一种制备所述衍生物的方法; 含有所述衍生物作为活性成分的农业和园艺杀真菌剂; 所述衍生物的中间体; 和中间体的制造方法。

    1,2,3-Thiadiazole derivatives or salts thereof and agrohorticultural disease controller
    4.
    发明授权
    1,2,3-Thiadiazole derivatives or salts thereof and agrohorticultural disease controller 失效
    1,2,3-噻二唑衍生物或其盐和农业园艺病控制剂

    公开(公告)号:US06337341B1

    公开(公告)日:2002-01-08

    申请号:US09665591

    申请日:2000-09-19

    IPC分类号: A01N4382

    摘要: A 1,2,3-thiadiazole derivative represented by general formula (I) or a salt thereof: wherein R1 is H, (halo) C1-C4 alkyl, 5- or 6-membered heterocycle containing 1 to 3 same or different O, N or S or the like, A is a group of the following formulas: wherein R2 and R3 are H, halogen, cyano, formyl, alkylthio, alkoxycarbonyl, substituted or unsubstituted phenyl, or the like, or R2 and R3, taken conjointly, may form a 3- to 7-membered ring including a C2-C6 alkylene group which may be intercepted by —O—, —S(O)n— (n is 0-2), —CO— or —NR8— (R8 is H, halogen or the like), B is cyano or an unsubstituted or substituted 5- or 6-membered heterocycle containing 1-3 hetero atoms selected from O, N and S, and m is 0-4; salts thereof; an agrohorticultural disease controller containing said derivative or salt; and method for using said disease controller.

    摘要翻译: 由通式(I)表示的1,2,3-噻二唑衍生物或其盐:其中R 1是H,(卤素)C 1 -C 4烷基,含有1至3个相同或不同的O的5或6元杂环, N或S等,A是下式的基团:其中R2和R3是H,卤素,氰基,甲酰基,烷硫基,烷氧基羰基,取代或未取代的苯基等,或R2和R3, 可以形成可被-O-,-S(O)n - (n为0-2),-CO-或-NR 8 - (R 8(R 8))截断的C 2 -C 6亚烷基的3-至7-元环 是H,卤素等),B是氰基或含有1-3个选自O,N和S的杂原子的未取代或取代的5-或6-元杂环,m是0-4; 的盐; 含有所述衍生物或盐的农业疾病控制器; 以及使用所述疾病控制器的方法。

    1,2,3-thiadiazole derivatives, plant disease controller and method for using the same
    7.
    发明授权
    1,2,3-thiadiazole derivatives, plant disease controller and method for using the same 失效
    1,2,3-噻二唑衍生物,植物病害控制剂及其使用方法

    公开(公告)号:US06348460B1

    公开(公告)日:2002-02-19

    申请号:US09437240

    申请日:1999-11-10

    IPC分类号: A01N4386

    摘要: A 1,2,3-thiadiazole derivative represented by general formula (I): [wherein R1 is hydrogen atom, halogen atom, (C1-C6) alkyl, phenyl, etc., R2 is the following group (A) or group (B): (wherein R3 is halogen atom, cyano, etc., R4 is hydrogen atom, halogen atom, cyano, etc., X and Y, same or different, are oxygen atom or sulfur atom, n is 0-3, R5 is hydrogen atom, (C1-C20) alkyl, etc., R6 is (C1-C20) alkyl, (C2-C20) alkenyl, etc., and m is 0-2)]; a plant disease controller containing said compound as active ingredient; and a method for using said controller.

    摘要翻译: 由通式(I)表示的1,2,3-噻二唑衍生物:其中R1是氢原子,卤素原子,(C1-C6)烷基,苯基等,R2是下列基团(A)或基团 B):(其中R3是卤素原子,氰基等,R4是氢原子,卤原子,氰基等,X和Y相同或不同,是氧原子或硫原子,n是0-3,R5 是(C 1 -C 20)烷基等,R 6是(C 1 -C 20)烷基,(C 2 -C 20)烯基等,m是0-2)]。 含有所述化合物作为活性成分的植物病害防除剂; 以及使用所述控制器的方法。

    Bis-thiadiazole derivatives or salts thereof and agrohorticultural disease controller and method for using the same
    8.
    发明授权
    Bis-thiadiazole derivatives or salts thereof and agrohorticultural disease controller and method for using the same 失效
    双噻二唑衍生物或其盐和农业园艺病控制剂及其使用方法

    公开(公告)号:US06313154B1

    公开(公告)日:2001-11-06

    申请号:US09276706

    申请日:1999-03-26

    IPC分类号: C07D41714

    CPC分类号: A01N43/82 C07D285/06

    摘要: A bis-thiadiazole derivative represented by general formula (I): wherein R1 and R2 represent H, C1-C8 alkyl, halo C1-C4 alkyl, unsubstituted or substituted phenyl, 5- or 6-membered heterocycle containing 1 to 3 hetero atoms selected from O, S and N, or the like; X1 and X2 represent O or S; Y1 and Y2 represent O, S or —N(R3)—; R represents C0-C30 alkylene. —(C)a(R3)(R4)— (R3 and R4 represent H, halogen, OH, C1-C4 alkyl, halo C1-C4 alkyl or the like) or the like; and a is 0 to 30; or a salt thereof, and an agrohorticultural disease controller containing said derivative or salt as an active ingredient.

    摘要翻译: 由通式(I)表示的双噻二唑衍生物:其中R1和R2表示H,C1-C8烷基,卤代C1-C4烷基,未取代或取代的苯基,含有1至3个杂原子的5-或6-元杂环选择 来自O,S和N等; X1和X2表示O或S; Y1和Y2表示O,S或-N(R3) - ; R表示C 0 -C 30亚烷基。 - (C)a(R3)(R4) - (R3和R4表示H,卤素,OH,C1-C4烷基,卤代C1-C4烷基等)等; a为0〜30; 或其盐,以及含有所述衍生物或盐作为活性成分的农业园艺疾病控制剂。