公开(公告)号：USH811H

公开(公告)日：1990-08-07

申请号：US322460

申请日：1989-03-13

申请人： Rikuo Nasu ,  Terumasa Komyoji ,  Toshio Nakajima ,  Kazumi Suzuki ,  Keiichiro Ito ,  Tekeshi Ohshima ,  Hideshi Yoshimura

发明人： Rikuo Nasu ,  Terumasa Komyoji ,  Toshio Nakajima ,  Kazumi Suzuki ,  Keiichiro Ito ,  Tekeshi Ohshima ,  Hideshi Yoshimura

IPC分类号： A01N43/50 ,  A01N47/14 ,  A01N47/34 ,  A01N47/38 ,  A01N53/00 ,  A01N55/00 ,  A01N57/12 ,  A01N59/20 ,  C07D233/90

CPC分类号： C07D233/90 ,  A01N43/50 ,  A01N63/04 ,  A01N59/20 ,  A01N57/12 ,  A01N55/00 ,  A01N53/00 ,  A01N47/38 ,  A01N47/34 ,  A01N47/14 ,  A01N47/04 ,  A01N43/90 ,  A01N43/80 ,  A01N43/653 ,  A01N43/40 ,  A01N37/36 ,  A01N37/34 ,  A01N37/24 ,  A01N2300/00

摘要： A biocidal composition containing, as active ingredients, at least one imidazole compound represented by formula (I): ##STR1## wherein R.sup.1 represents a phenyl group, a halogen-substituted phenyl group, an alkyl group, or a halogen-substituted alkyl group; and R.sup.2 represents a halogen atom, and at least one other specific compound. The combination of the compound represented by formula (I) and other specific compound can produce an unexpected effect in amount required and biocidal spectrum.

公开(公告)号：US4995898A

公开(公告)日：1991-02-26

申请号：US168070

申请日：1988-03-14

申请人： Rikuo Nasu ,  Terumasa Komyoji ,  Toshio Nakajima ,  Kazumi Suzuki ,  Keiichiro Ito ,  Takeshi Oshima ,  Hideshi Yoshimura

发明人： Rikuo Nasu ,  Terumasa Komyoji ,  Toshio Nakajima ,  Kazumi Suzuki ,  Keiichiro Ito ,  Takeshi Oshima ,  Hideshi Yoshimura

IPC分类号： A01N43/50 ,  A01N31/14 ,  A01N33/00 ,  A01N37/34 ,  A01N43/08 ,  A01N43/84 ,  A01N55/00 ,  A01P3/00 ,  C07D233/84 ,  C07D233/90 ,  C07D233/92 ,  C07D401/04 ,  C07D401/12 ,  C07D405/04 ,  C07D405/14 ,  C07D409/04 ,  C07D409/12 ,  C07F7/08

CPC分类号： C07D401/04 ,  A01N43/50 ,  A01N55/00 ,  C07D233/90 ,  C07D401/12 ,  C07D405/04 ,  C07D405/14 ,  C07D409/04 ,  C07F7/0814

摘要： Novel imidazole compounds are disclosed, which are represented by the following general formula: ##STR1## wherein: R.sub.1 represents a cyano group or a --CSNHR.sub.5 group, wherein R.sub.5 represents a hydrogen atom, a C.sub.1-4 alkyl group, or a --COR.sub.6 group, wherein R.sub.6 represents a C.sub.1-4 alkyl group, a halogenated C.sub.1-4 alkyl group, or a phenyl group;R.sub.2 and R.sub.3 each represents a hydrogen atom; a halogen atom; a nitro group; a cyano group; a trimethylsilyl group; a C.sub.3-6 cycloalkyl group; a naphthyl group; a C.sub.1-12 alkyl group which is optionally substituted with one or more halogen atoms, hydroxyl groups, acetoxy groups, C.sub.1-4 alkoxy groups, halogenated C.sub.1-4 alkoxy groups, phenyl groups, halogenated phenyl groups, or C.sub.1-4 alkylated phenyl groups; a C.sub.2-10 alkenyl group which is optionally substituted with one or more halogen atoms; a C.sub.1-6 alkoxy group which is optionally substituted with one or more halogen atoms; a phenyl group which is optionally substituted with one or more halogen atoms, C.sub.1-4 alkyl groups, halogenated C.sub.1-4 alkyl groups, C.sub.1-4 alkoxy groups, halogenated C.sub.1-4 alkoxy groups, C.sub.1-4 alkylthio groups, halogenated C.sub.1-4 alkylthio groups, nitro groups, cyano groups, or 3,4-methylenedioxy groups; a furyl group which is optionally substituted with one or more halogen atoms or C.sub.1-4 alkyl groups; a thienyl group which is optionally substituted with one or more halogen atoms or C.sub.1-4 alkyl groups; a pyridyl group which is optionally substituted with one or more halogen atoms or C.sub.1-4 alkyl groups; an --SO.sub.n R.sub.7 group, wherein R.sub.7 represents a C.sub.1-6 alkyl group, a C.sub.2-6 alkenyl group, a phenyl group which is optionally substituted with one or more halogen atoms, a benzyl group, a pyridyl group which is optionally substituted with one or more halogen atoms, C.sub.1-4 alkyl groups, or halogenated C.sub.1-4 alkyl groups; or an --NR.sub.8 R.sub.9 group, wherein R.sub.8 and R.sub.9 each represents a C.sub.1-4 alkyl group, and n is 0, 1, or 2; or a --CO(NH).sub.m R.sub.10 group, wherein R.sub.10 represents a C.sub.1-4 alkyl group which is optionally substituted with one or more halogen atoms, a C.sub.1-4 alkoxy group which is optionally substituted with one or more halogen atoms, or a phenyl group which is optionally substituted with one or more halogen atoms; and m is 0 or 1; andR.sub.4 represents a C.sub.1-6 alkyl group which is optionally substituted with one or more halogen atoms; a C.sub.3-6 cycloalkyl group; a phenyl group; a thienyl group; or an --NR.sub.11 R.sub.12 group, wherein R.sub.11 and R.sub.12 each represents a hydrogen atom, a C.sub.1-4 alkyl group which is optionally substituted with one or more halogen atoms, a C.sub.2-4 alkenyl group, or R.sub.11 and R.sub.12 are combined with each other together with a nitrogen atoms adjacent thereto to form a pyrrolidinyl group, a piperidinyl group, a morpholino group, or a thiomorpholino group, provided that R.sub.11 and R.sub.12 are not simultaneously a hydrogen atom;provided that R.sub.2 and R.sub.3 are not simultaneously a halogen atom. The compounds are effective as biocides.

摘要翻译： 由通式I表示的咪唑化合物：其中：R1表示氰基或-CSNHR5基团，其中R5表示氢原子，C1-4烷基或-COR6基团，其中R6表示C1- 4烷基，卤代C 1-4烷基或苯基; R2和R3各自表示氢原子; 卤素原子; 硝基; 氰基; 三甲基甲硅烷基 C 3-6环烷基; 萘基; 任选取代的C 1-12烷基，C 2-10烯基，C 1-6烷氧基，苯基，呋喃基，亚硫酰基或吡啶基; a-SO n R 7基，其中R 7表示C 1-6烷基，C 2-6烯基，苄基，任选取代的苯基或吡啶基; NR8R9基团，其中R8和R9各自表示C1-4烷基，n为0,1或2; 或-CO（NH）m R 10 gorup，其中R 10表示任选取代的C 1-4烷基，C 1-4烷氧基或苯基，m为0或1; 并且R 4表示任选被一个或多个卤素原子取代的C 1-6烷基; C 3-6环烷基; 苯基; 噻吩基; 或-NR 11 R 12基团，其中R 11和R 12各自表示氢原子，任选被一个或多个卤素原子取代的C 1-4烷基，C 2-4链烯基或R 11和R 12一起彼此结合 与其相邻的氮原子形成吡咯烷基，哌啶基，吗啉代基或硫代吗啉基，条件是R 11和R 12不同时为氢原子; 条件是R2和R3不同时为卤素原子。 这些化合物作为杀生物剂是有效的。