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1.Substituted Aromatic Carboxamide and Urea Derivatives as Vanilloid Receptor Ligands 失效
标题翻译: 取代芳香酰胺和尿素衍生物作为香草素受体配体公开(公告)号:US20110003795A1
公开(公告)日:2011-01-06
申请号:US12775155
申请日:2010-05-06
申请人: Robert FRANK , Gregor BAHRENBERG , Thomas CHRISTOPH , Klaus SCHIENE , Jean DE VRY , Nils DAMANN , Sven FRORMANN , Bernhard LESCH , Jeewoo LEE , Yong-Soo KIM , Myeong-Seop KIM
发明人: Robert FRANK , Gregor BAHRENBERG , Thomas CHRISTOPH , Klaus SCHIENE , Jean DE VRY , Nils DAMANN , Sven FRORMANN , Bernhard LESCH , Jeewoo LEE , Yong-Soo KIM , Myeong-Seop KIM
IPC分类号: A61K31/55 , C07D223/16 , C07D279/16 , C07D265/36 , C07D265/12 , C07D215/38 , C07D217/02 , C07D249/08 , C07D231/10 , A61K31/5415 , A61K31/536 , A61K31/4709 , A61K31/4725 , A61K31/415 , A61K31/4196 , A61P25/00 , A61P9/12 , A61P11/08 , A61P9/10 , A61P25/30 , A61P25/32
CPC分类号: C07D231/12 , C07D249/08 , C07D401/12 , C07D401/14 , C07D403/12 , C07D405/12 , C07D409/14 , C07D417/12
摘要: The invention relates to substituted aromatic carboxamide and urea derivatives, to processes for the preparation thereof, to pharmaceutical compositions containing these compounds and also to the use of these compounds for preparing pharmaceutical compositions.
摘要翻译: 本发明涉及取代的芳族羧酰胺和脲衍生物,其制备方法,含有这些化合物的药物组合物以及这些化合物用于制备药物组合物的用途。
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2.Substituted Heteroaromatic Pyrazole-Containing Carboxamide and Urea Compounds as Vanilloid Receptor Ligands 审中-公开
标题翻译: 取代的杂芳族吡唑含有羧酰胺和脲化合物作为香草素受体配体公开(公告)号:US20130029962A1
公开(公告)日:2013-01-31
申请号:US13557941
申请日:2012-07-25
IPC分类号: A61K31/4439 , C07D403/12 , A61K31/506 , C07D401/14 , A61P29/00 , A61P25/06 , A61P25/30 , A61P25/28 , A61P25/16 , A61P3/04 , A61P9/12 , A61P11/08 , A61P9/00 , A61P17/02 , A61P25/00 , A61P23/00 , A61P15/00 , C07D401/12
CPC分类号: C07D401/12 , A61K31/4155 , A61K31/4427 , A61K31/506 , C07D401/14 , C07D403/12
摘要: Substituted heteroaromatic pyrazole-containing carboxamide and urea compounds as vanilloid receptor ligands, pharmaceutical compositions containing these compounds and also to a method of using these compounds for treating and/or inhibiting pain and further diseases and/or disorders.
摘要翻译: 含取代的含杂芳基吡唑的甲酰胺和尿素化合物作为香草素受体配体,含有这些化合物的药物组合物,以及使用这些化合物治疗和/或抑制疼痛和其它疾病和/或病症的方法。
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3.Substituted Bicyclic Aromatic Carboxamide and Urea Compounds as Vanilloid Receptor Ligands 有权
标题翻译: 取代的双环芳族羧酰胺和尿素化合物作为香草素受体配体公开(公告)号:US20130029995A1
公开(公告)日:2013-01-31
申请号:US13557863
申请日:2012-07-25
申请人: Robert FRANK , Thomas CHRISTOPH , Bernhard LESCH , Jeewoo LEE
发明人: Robert FRANK , Thomas CHRISTOPH , Bernhard LESCH , Jeewoo LEE
IPC分类号: C07D401/14 , C07D471/04 , C07D401/12 , A61K31/4709 , A61K31/4725 , C07D491/056 , C07D498/04 , A61K31/444 , C07D513/04 , C07D413/14 , C07D417/14 , A61K31/4439 , A61K31/454 , A61K31/517 , A61K31/498 , A61K31/502 , A61P29/00 , A61P25/06 , A61P25/24 , A61P25/00 , A61P25/28 , A61P25/08 , A61P11/00 , A61P11/10 , A61P13/00 , A61P13/10 , A61P1/00 , A61P1/04 , A61P27/02 , A61P17/00 , A61P17/06 , A61P31/22 , A61P1/12 , A61P17/04 , A61P19/10 , A61P19/02 , A61P3/00 , A61P25/30 , A61P25/32 , A61P9/00 , A61P17/02 , A61P15/00 , A61P25/22 , A61P23/02 , A61P25/16 , A61P11/06 , A61P3/04 , A61P9/12 , A61P11/08 , A61K31/4545
CPC分类号: C07D401/12 , C07D471/04
摘要: Substituted bicyclic aromatic carboxamide and urea compounds as vanilloid receptor ligands, pharmaceutical compositions containing these compounds, and a method of using these compounds in the treatment and/or inhibition of pain and further diseases and/or disorders mediated at least in part via the vanilloid receptor 1 (VR1/TRPV1).
摘要翻译: 取代的双环芳族羧酰胺和尿素化合物作为香草素受体配体,含有这些化合物的药物组合物,以及使用这些化合物治疗和/或抑制至少部分通过香草素受体介导的疼痛和其它疾病和/或病症的方法 1(VR1 / TRPV1)。
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