Pyridine derivatives compounds for controlling invertebrate pests
    1.
    发明授权
    Pyridine derivatives compounds for controlling invertebrate pests 有权
    用于控制无脊椎动物害虫的吡啶衍生物化合物

    公开(公告)号:US09125414B2

    公开(公告)日:2015-09-08

    申请号:US13386473

    申请日:2010-07-15

    摘要: The present invention relates to methods and uses of compounds of formulae I or II and the salts and N-oxides thereof, wherein A is a substituted or unsubstituted 5-membered heterocyclic radical; X1 is S, O or NR1a, wherein R1a is selected from H, C1-C10-alkyl and the like; X2 is OR2a, NR2bR2c, S(O)mR2d; X2 is OR2a, NR2bR2c, S(O)mR2d, wherein m is 0, 1 or 2, R2a is C1-C4-alkyl, C1-C4-haloalkyl and the like, R2b, R2c are H, C1-C4-alkyl, C1-C4-haloalkyl and the like; X3 is a lone pair or oxygen; R1, R2 and R3 are, inter alia, hydrogen, and R1 is H, C1-C10-alkyl and the like. The present invention further relates to a method for controlling invertebrate pests, to a method for protecting plant propagation material and/or the plants which grow therefrom, to plant propagation material, comprising at least one compound according to the present invention, to a method for treating or protecting an animal from infestation or infection by parasites and to an agricultural composition containing at least one compound according to the present invention.

    摘要翻译: 本发明涉及式I或II化合物及其盐和N-氧化物的方法和用途,其中A是取代或未取代的5元杂环基; X1是S,O或NR1a,其中R1a选自H,C1-C10-烷基等; X2是OR2a,NR2bR2c,S(O)mR2d; X2是OR2a,NR2bR2c,S(O)mR2d,其中m是0,1或2,R2a是C1-C4-烷基,C1-C4-卤代烷基等,R2b,R2c是H,C1-C4-烷基, C1-C4卤代烷基等; X3是孤对或氧气; R1,R2和R3尤其是氢,R1是H,C1-C10-烷基等。 本发明还涉及一种控制无脊椎害虫的方法,一种用于保护植物繁殖材料和/或从其生长的植物的方法,包括至少一种根据本发明的化合物的植物繁殖材料的方法, 治疗或保护动物免受寄生虫侵袭或感染,以及含有至少一种本发明化合物的农药组合物。

    Pyridazine compounds for controlling invertebrate pests

    公开(公告)号:US09040537B2

    公开(公告)日:2015-05-26

    申请号:US13634899

    申请日:2011-03-23

    CPC分类号: C07D403/12 A01N43/58

    摘要: The present invention relates to pyridazine compounds of formulae I or II and the salts thereof, the N-oxides thereof and the salts of the N-oxides thereof, where the radical A is of the formula A, wherein # denotes the point of attachment to the remainder of formulae I or II, and wherein A1 is N or C—RA1, A2 is N or C—RA2, A3 is N or C—RA3, A4 is N or C—RA4 and A5 is N or C—RA5, provided that one or two of the variables A1, A2, A3, A4 or A5 is N; RA1, RA5, if present, are H, halogen, CN, NO2, C1-C6-alkyl, C1-C6-haloalkyl and the like; RA2, RA4, if present, are H, halogen, CN, NO2, C1-C10-alkyl, C1-C10-haloalkyl and the like; RA3, if present, is H, halogen, CN, NO2, C1-C10-alkyl, C1-C10-haloalkyl and the like; where W is N or C—RW and V is N or C—RV, provided that one of the variables W or V is N; Rt and Rw, if present, are H, halogen, methyl, C1-haloalkyl and the like; Ru and Rv, if present, are H, halogen, C1-C4-alkyl, C1-C3-haloalkyl and the like; X1 is S, O or NR1a, wherein R1a is H, C1-C10-alkyl and the like; X2 is OR2a, NR2bR2c, S(O)mR2d, wherein m is 0, 1 or 2, R2a is C1-C4-alkyl, C1-C4-haloalkyl and the like, R2b, R2c are H, C1-C4-alkyl, C1-C4-haloalkyl and the like, or R2b and R2c together with the nitrogen atom to which they are bound form a heterocycle, and R2d is C1-C4-alkyl, C1-C4-haloalkyl, C3-C6-cycloalkyl and the like; and R1 is H, CN, C1-C10-alkyl and the like. The present invention further relates to a method for controlling invertebrate pests, to a method for protecting plant propagation material and/or the plants which grow therefrom, to plant propagation material, comprising at least one compound according to the present invention, to a method for treating or protecting an animal from infestation or infection by parasites and to an agricultural composition containing at least one compound according to the present invention.

    Pyridine Compounds for Controlling Invertebrate Pests II
    3.
    发明申请
    Pyridine Compounds for Controlling Invertebrate Pests II 审中-公开
    用于控制无脊椎动物害虫的吡啶化合物

    公开(公告)号:US20130203821A1

    公开(公告)日:2013-08-08

    申请号:US13821745

    申请日:2011-09-12

    摘要: The present invention relates to novel pyridine compounds of the formulae I and II, to their salts, to their tautomers, to their N-oxides, and to the salts of these N-oxides or tautomers. The compounds are useful for combating or controlling invertebrate pests, in particular arthropod pests. The invention also relates to a method for controlling in-vertebrate pests by using these compounds. The invention further relates to plant propagation material and to agricultural compositions comprising said compounds. wherein A is a radical of the formulae A1, A2, A3, A4, A5 or A6 wherein # denotes the binding site to the remainder of formulae I or II; Z is O, S or N—RN; X1 is S, O or NR1a; X2 is OR2a, NR2bR2c, S(O)mR2d; X3 is a lone pair or oxygen; R1, R2 and R3 are, inter alia, hydrogen, and RA1, RA2RA3RA4, RA5, RA6 and RN, are as defined in claim 1.

    摘要翻译: 本发明涉及式I和II的新型吡啶化合物,其盐,其互变异构体,其N-氧化物,以及这些N-氧化物或互变异构体的盐。 这些化合物可用于对抗或控制无脊椎害虫,特别是节肢动物害虫。 本发明还涉及通过使用这些化合物来控制脊椎动物害虫的方法。 本发明还涉及植物繁殖材料和包含所述化合物的农业组合物。 其中A是式A1,A2,A3,A4,A5或A6的基团,其中#表示与式I或II的其余部分的结合位点; Z是O,S或N-RN; X1是S,O或NR1a; X2是OR2a,NR2bR2c,S(O)mR2d; X3是孤对或氧气; R1,R2和R3尤其是氢,RA1,RA2RA3RA4,RA5,RA6和RN如权利要求1中所定义。

    Pyridine compounds for controlling invertebrate pests I
    5.
    发明授权
    Pyridine compounds for controlling invertebrate pests I 有权
    用于控制无脊椎动物害虫的吡啶化合物

    公开(公告)号:US08609700B2

    公开(公告)日:2013-12-17

    申请号:US13821749

    申请日:2011-09-12

    摘要: The present invention relates to novel pyridine compounds of the formulae I and II, to their salts, to their tautomers, to their N-oxides, and to the salts of these N-oxides or tautomers. The compounds are useful for combating or controlling invertebrate pests, in particular arthropod pests. The invention also relates to a method for controlling invertebrate pests by using these compounds. The invention further relates to plant propagation material and to agricultural compositions comprising said compounds. wherein A is a radical of the formulae A1 or A2 # denotes the binding site to the remainder of formulae I or II; n is 0, 1, 2 or 3; Z is O, S or N—RN; X1 is S, O or NR1a; X2 is OR2a, NR2bR2c, S(O)mR2d; X3 is a lone pair or oxygen; R1, R2 and R3 are, inter alia, hydrogen, and RA and RN, are as defined in claim 1.

    摘要翻译: 本发明涉及式I和II的新型吡啶化合物,其盐,其互变异构体,其N-氧化物,以及这些N-氧化物或互变异构体的盐。 这些化合物可用于对抗或控制无脊椎害虫,特别是节肢动物害虫。 本发明还涉及通过使用这些化合物来控制无脊椎害虫的方法。 本发明还涉及植物繁殖材料和包含所述化合物的农业组合物。 其中A是式A1或A2的基团,#表示与式I或II的其余部分的结合位点; n为0,1,2或3; Z是O,S或N-RN; X1是S,O或NR1a; X2是OR2a,NR2bR2c,S(O)mR2d; X3是孤对或氧气; R1,R2和R3尤其是氢,RA和RN如权利要求1中所定义。

    Pyridazine Compounds For Controlling Invertebrate Pests

    公开(公告)号:US20130012380A1

    公开(公告)日:2013-01-10

    申请号:US13634899

    申请日:2011-03-23

    CPC分类号: C07D403/12 A01N43/58

    摘要: The present invention relates to pyridazine compounds of formulae I or II and the salts thereof, the N-oxides thereof and the salts of the N-oxides thereof, where the radical A is of the formula A, wherein # denotes the point of attachment to the remainder of formulae I or II, and wherein A1 is N or C—RA1, A2 is N or C—RA2, A3 is N or C—RA3, A4 is N or C—RA4 and A5 is N or C—RA5, provided that one or two of the variables A1, A2, A3, A4 or A5 is N; RA1, RA5, if present, are H, halogen, CN, NO2, C1-C6-alkyl, C1-C6-haloalkyl and the like; RA2, RA4, if present, are H, halogen, CN, NO2, C1-C10-alkyl, C1-C10-haloalkyl and the like; RA3, if present, is H, halogen, CN, NO2, C1-C10-alkyl, C1-C10-haloalkyl and the like; where W is N or C—RW and V is N or C—RV, provided that one of the variables W or V is N; Rt and Rw, if present, are H, halogen, methyl, C1-haloalkyl and the like; Ru and Rv, if present, are H, halogen, C1-C4-alkyl, C1-C3-haloalkyl and the like; X1 is S, O or NR1a, wherein R1a is H, C1-C10-alkyl and the like; X2 is OR2a, NR2bR2c, S(O)mR2d, wherein m is 0, 1 or 2, R2a is C1-C4-alkyl, C1-C4-haloalkyl and the like, R2b, R2c are H, C1-C4-alkyl, C1-C4-haloalkyl and the like, or R2b and R2c together with the nitrogen atom to which they are bound form a heterocycle, and R2d is C1-C4-alkyl, C1-C4-haloalkyl, C3-C6-cycloalkyl and the like; and R1 is H, CN, C1-C10-alkyl and the like.The present invention further relates to a method for controlling invertebrate pests, to a method for protecting plant propagation material and/or the plants which grow therefrom, to plant propagation material, comprising at least one compound according to the present invention, to a method for treating or protecting an animal from infestation or infection by parasites and to an agricultural composition containing at least one compound according to the present invention.

    Pyridazine compounds for controlling invertebrate pests
    7.
    发明授权
    Pyridazine compounds for controlling invertebrate pests 有权
    用于控制无脊椎害虫的哒嗪化合物

    公开(公告)号:US08710056B2

    公开(公告)日:2014-04-29

    申请号:US13382229

    申请日:2010-07-01

    摘要: The present invention relates to pyridazine compounds of formulae I or II and the salts and N-oxides thereof, wherein A is a substituted or unsubstituted isoxazole or isothiazole radical; V is C(Rv) or N; W is C(Rw) or N; with the proviso that either V or W is N; Rt, Ru, Rv, Rw are H, halogen, C1-C4-alkyl and the like; X1 is S, O or NR1a, wherein R1a is selected H, C1-C10-alkyl and the like; X2 is OR2a, NR2bR2c, S(O)mR2d, wherein m is 0, 1 or 2, R2a is C1-C4-alkyl, C1-C4-haloalkyl and the like, R2b, R2c are H, C1-C4-alkyl, C1-C4-haloalkyl and the like, or R2b and R2c together with the nitrogen atom to which they are bound form a heterocycle, and R2d is C1-C4-alkyl, C1-C4-haloalkyl, C3-C6-cycloalkyl and the like; and R1 is H, CN, C1-C10-alkyl and the like. The present invention further relates to a method for controlling invertebrate pests, to a method for protecting plant propagation material and/or the plants which grow therefrom, to plant propagation material, comprising at least one compound according to the present invention, to a method for treating or protecting an animal from infestation or infection by parasites and to an agricultural composition containing at least one compound according to the present invention.

    摘要翻译: 本发明涉及式I或II的哒嗪化合物及其盐和N-氧化物,其中A是取代或未取代的异恶唑或异噻唑基; V是C(Rv)或N; W是C(Rw)或N; 条件是V或W为N; R 1,R u,R v,R w为H,卤素,C 1 -C 4 - 烷基等; X1是S,O或NR1a,其中R1a选自H,C1-C10-烷基等; X2是OR2a,NR2bR2c,S(O)mR2d,其中m是0,1或2,R2a是C1-C4-烷基,C1-C4-卤代烷基等,R2b,R2c是H,C1-C4-烷基, C1-C4卤代烷基等,或R2b和R2c与它们所结合的氮原子一起形成杂环,R2d是C1-C4-烷基,C1-C4卤代烷基,C3-C6-环烷基等 ; R1为H,CN,C1-C10-烷基等。 本发明还涉及一种控制无脊椎害虫的方法,一种用于保护植物繁殖材料和/或从其生长的植物的方法,包括至少一种根据本发明的化合物的植物繁殖材料的方法, 治疗或保护动物免受寄生虫侵袭或感染,以及含有至少一种本发明化合物的农药组合物。

    Pyridine Compounds for Controlling Invertebrate Pests III
    8.
    发明申请
    Pyridine Compounds for Controlling Invertebrate Pests III 审中-公开
    用于控制无脊椎动物害虫的吡啶化合物

    公开(公告)号:US20130180014A1

    公开(公告)日:2013-07-11

    申请号:US13822529

    申请日:2011-09-12

    摘要: The present invention relates to a method for controlling invertebrate pests, in particular arthropod pests and nematodes, by using pyridine compounds of formulae I or II and the salts thereof, the tautomers thereof, the N-oxides thereof and the salts of the tautomers or N-oxides thereof, where the radical A is of the formula A, wherein # denotes the point of attachment to the remainder of formulae I or II, and wherein A1 is N or C—RA1, A2 is N or C—RA2, A3 is N or C—RA3, A4 is N or C—RA4 and A5 is N or C—RA5, provided that one or two of the variables A1, A2, A3, A4 or A5 is N; RA1, RA5, if present, are H, halogen, CN, NO2, C1-C6-alkyl, C1-C6-haloalkyl and the like; RA2, RA4, if present, are H, halogen, CN, NO2, C1-C10-alkyl, C1-C10-haloalkyl and the like; RA3, if present, is H, halogen, CN, NO2, C1-C10-alkyl, C1-C10-haloalkyl and the like; R1 is H, CN, C1-C10-alkyl, C1-C10-haloalkyl and the like; R2 is H, halogen, methyl, C1-haloalkyl and the like; R3 is H, halogen, C1-C4-alkyl, C1-C3-haloalkyl and the like; X1 is S, O or NR1a, wherein R1a is H, C1-C10-alkyl and the like; X2 is OR2a, NR2bR2c or S(O)mR2d, wherein m is 0, 1 or 2, R2a is C1-C4-alkyl, C1-C4-haloalkyl and the like, R2b and R2c are H, C1-C4-alkyl, C1-C4-haloalkyl and the like, or R2b and R2c together with the nitrogen atom to which they are bound form a heterocycle, and R2d is C1-C4-alkyl, C1-C4-haloalkyl, C3-C6-cycloalkyl and the like. The present invention further relates to a method for protecting plant propagation material and/or the plants which grow therefrom, to plant propagation material, comprising at least one compound of formulae I or II, their salts or N-oxides, and to an agricultural composition containing at least one compound of formulae I or II, their salts or N-oxides.

    摘要翻译: 本发明涉及通过使用式I或II的吡啶化合物及其盐,其互变异构体,其N-氧化物和互变异构体或N的盐来控制无脊椎害虫,特别是节肢动物害虫和线虫的方法 其中基团A为式A,其中#表示与式I或II的其余部分的连接点,其中A1为N或C-RA1,A2为N或C-RA2,A3为 N或C-RA3,A4是N或C-RA4,A5是N或C-RA5,条件是变量A1,A2,A3,A4或A5中的一个或两个为N; RA1,RA5如果存在,是H,卤素,CN,NO 2,C 1 -C 6 - 烷基,C 1 -C 6 - 卤代烷基等; RA2,RA4如果存在,是H,卤素,CN,NO 2,C 1 -C 10 - 烷基,C 1 -C 10 - 卤代烷基等; 如果存在,RA 3是H,卤素,CN,NO 2,C 1 -C 10 - 烷基,C 1 -C 10 - 卤代烷基等; R1是H,CN,C1-C10-烷基,C1-C10-卤代烷基等; R 2是H,卤素,甲基,C 1 - 卤代烷基等; R3是H,卤素,C1-C4-烷基,C1-C3-卤代烷基等; X1是S,O或NR1a,其中R1a是H,C1-C10-烷基等; X2是OR2a,NR2bR2c或S(O)mR2d,其中m是0,1或2,R2a是C1-C4-烷基,C1-C4-卤代烷基等,R2b和R2c是H,C1-C4-烷基, C1-C4卤代烷基等,或R2b和R2c与它们所结合的氮原子一起形成杂环,R2d是C1-C4-烷基,C1-C4卤代烷基,C3-C6-环烷基等 。 本发明还涉及一种用于保护植物繁殖材料和/或从其生长的植物的方法,包括至少一种式I或II化合物,其盐或N-氧化物的植物繁殖材料,以及农业组合物 含有至少一种式I或II的化合物,其盐或N-氧化物。

    Pyrazole Compounds for Controlling Invertebrate Pests
    10.
    发明申请
    Pyrazole Compounds for Controlling Invertebrate Pests 审中-公开
    用于控制无脊椎动物害虫的吡唑化合物

    公开(公告)号:US20130253012A1

    公开(公告)日:2013-09-26

    申请号:US13992108

    申请日:2011-12-09

    摘要: The present invention relates to a method for controlling invertebrate pests, in particular arthropod pests and nematodes, by using pyrazole compounds of formula I and the salts thereof, the tautomers thereof, the N-oxides thereof and the salts of the tautomers or N-oxides thereof, wherein X is N or CH, Y is N or CH, Z is N or CH, provided that either only one of X, Y and Z is N or only two adjacent groups of X, Y and Z are N; and wherein Q is a bivalent 5- or 6-membered carbocyclic radical or a 5- or 6-membered heterocyclic radical having one heteroatom moiety which is selected from the group consisting of O, S, N or N—RQN as ring member and 0, 1 or 2 further heteroatom moieties N as ring members, wherein 0, 1, 2 or 3 of the ring members that are carbon atoms may carry a radical RQ, provided that the pyrazole radical and the 6-membered heteroaromatic radical are bound in ortho- or meta-position of Q with respect to each other, if Q is a 6-membered radical; and wherein RA, if present, is C1-C3-alkyl, C1-C3-haloalkyl or the like; n is 0, 1 or 2; RN is C1-C3-alkyl, C1-C2-haloalkyl, C1-C2-alkoxy-C1-C2-alkyl or the like; Rt and Ru are independently of each other selected from hydrogen, methyl and the like; RQN is hydrogen, C1-C4-alkyl or the like; RQ is hydrogen, halogen, C1-C4-alkyl or the like. The present invention further relates to a method for protecting plant propagation material and/or the plants which grow therefrom, to plant propagation material, comprising at least one compound of formula I, their salts or N-oxides, and to pyrazole compounds of formula I.

    摘要翻译: 本发明涉及通过使用式I的吡唑化合物及其盐,其互变异构体,其N-氧化物和互变异构体或N-氧化物的盐来控制无脊椎害虫,特别是节肢动物害虫和线虫的方法 其中X是N或CH,Y是N或CH,Z是N或CH,条件是X,Y和Z中只有一个是N或只有X,Y和Z的两个相邻基团是N; 并且其中Q是二价5-或6-元碳环基团或具有一个杂原子部分的5-或6-元杂环基团,其选自O,S,N或N-RQN作为环成员,0 ,1个或2个另外的杂原子部分N作为环成员,其中作为碳原子的环成员的0,1,2或3可以携带自由基RQ,条件是吡唑基和6元杂芳族基团在邻位 - 或相对于Q的间位,如果Q是6元基团; 并且其中RA如果存在,是C 1 -C 3 - 烷基,C 1 -C 3 - 卤代烷基等; n为0,1或2; RN是C 1 -C 3烷基,C 1 -C 2卤代烷基,C 1 -C 2烷氧基-C 1 -C 2烷基等; Rt和Ru彼此独立地选自氢,甲基等; RQN是氢,C1-C4烷基等; RQ是氢,卤素,C1-C4烷基等。 本发明还涉及一种用于保护植物繁殖材料和/或从其生长的植物的植物繁殖材料的方法,其包含至少一种式I化合物,其盐或N-氧化物,以及式I的吡唑化合物 。