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公开(公告)号:US20120129862A1
公开(公告)日:2012-05-24
申请号:US13113751
申请日:2011-05-23
申请人: Steven J. Coats , Alexey B. Dyatkin , Wei He , Joseph Lisko , Tamara A. Miskowski , Janet L. Ralbovsky , Mark J. Schulz
发明人: Steven J. Coats , Alexey B. Dyatkin , Wei He , Joseph Lisko , Tamara A. Miskowski , Janet L. Ralbovsky , Mark J. Schulz
IPC分类号: A61K31/53 , C07D403/12 , C07D251/20 , A61P29/00 , C07D251/38 , A61P1/00 , A61P1/12 , A61P35/00 , C07D251/46 , C07D251/30
CPC分类号: C07D239/545 , C07D251/20 , C07D251/34 , C07D251/38 , C07D251/46 , C07D403/12
摘要: The present invention relates to certain novel compounds of Formula (I): and methods for preparing these compounds, compositions, intermediates and derivatives thereof and for the treatment of prokineticin 1 or prokinetin 1 receptor mediated disorders.
摘要翻译: 本发明涉及某些新的式(I)化合物:以及制备这些化合物,组合物,中间体和衍生物以及用于治疗促动蛋白原1或原激素1受体介导的病症的方法。
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公开(公告)号:US20090163505A1
公开(公告)日:2009-06-25
申请号:US12256891
申请日:2008-10-23
申请人: Steven J. COATS , Alexey B. Dyatkin , Wei He , Joseph Lisko , Tamara A. Miskowski , Janet L. Ralbovsky , Mark J. Schulz
发明人: Steven J. COATS , Alexey B. Dyatkin , Wei He , Joseph Lisko , Tamara A. Miskowski , Janet L. Ralbovsky , Mark J. Schulz
IPC分类号: A61K31/53 , C07D403/12 , A61P1/00 , A61P35/00
CPC分类号: C07D251/38 , C07D401/12 , C07D403/12 , C07D405/14
摘要: The present invention relates to certain novel compounds of Formula (I): and methods for preparing these compounds, compositions, intermediates and derivatives thereof and for the treatment of prokineticin 1 or prokinetin 1 receptor mediated disorders.
摘要翻译: 本发明涉及某些新的式(I)化合物:以及制备这些化合物,组合物,中间体及其衍生物以及用于治疗促动蛋白原1或原激素1受体介导的病症的方法。
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公开(公告)号:US08324380B2
公开(公告)日:2012-12-04
申请号:US12256891
申请日:2008-10-23
申请人: Steven J. Coats , Alexey B. Dyatkin , Wei He , Joseph Lisko , Tamara A. Miskowski , Janet L. Ralbovsky , Mark J. Schulz
发明人: Steven J. Coats , Alexey B. Dyatkin , Wei He , Joseph Lisko , Tamara A. Miskowski , Janet L. Ralbovsky , Mark J. Schulz
IPC分类号: C07D251/30 , C07D401/06 , C07D401/14 , C07D403/06 , C07D403/14 , C07D401/12 , C07D403/12 , A61K31/53 , A61P1/12 , A61P1/06 , A61P1/00
CPC分类号: C07D251/38 , C07D401/12 , C07D403/12 , C07D405/14
摘要: The present invention relates to certain novel compounds of Formula (I): and methods for preparing these compounds, compositions, intermediates and derivatives thereof and for the treatment of prokineticin 1 or prokinetin 1 receptor mediated disorders.
摘要翻译: 本发明涉及某些新的式(I)化合物:以及制备这些化合物,组合物,中间体及其衍生物以及用于治疗促动蛋白原1或原激素1受体介导的病症的方法。
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公开(公告)号:US20140038968A1
公开(公告)日:2014-02-06
申请号:US13653452
申请日:2012-10-17
申请人: Steven J. Coats , Alexey B. Dyatkin , Wei He , Joseph Lisko , Tamara A. Miskowski , Janet L. Ralbovsky , Mark J. Schulz
发明人: Steven J. Coats , Alexey B. Dyatkin , Wei He , Joseph Lisko , Tamara A. Miskowski , Janet L. Ralbovsky , Mark J. Schulz
IPC分类号: C07D251/38 , C07D403/12
CPC分类号: C07D251/38 , C07D401/12 , C07D403/12 , C07D405/14
摘要: The present invention relates to certain novel compounds of Formula (I): and methods for preparing these compounds, compositions, intermediates and derivatives thereof and for the treatment of prokineticin 1 or prokinetin 1 receptor mediated disorders.
摘要翻译: 本发明涉及某些新的式(I)化合物:以及制备这些化合物,组合物,中间体及其衍生物以及用于治疗促动蛋白原1或原激素1受体介导的病症的方法。
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公开(公告)号:US08362247B2
公开(公告)日:2013-01-29
申请号:US13113751
申请日:2011-05-23
申请人: Steven J. Coats , Alexey B. Dyatkin , Wei He , Joseph Lisko , Tamara A. Miskowski , Janet L. Ralbovsky , Mark J. Schulz
发明人: Steven J. Coats , Alexey B. Dyatkin , Wei He , Joseph Lisko , Tamara A. Miskowski , Janet L. Ralbovsky , Mark J. Schulz
IPC分类号: C07D403/06 , C07D403/12 , C07D403/14 , C07D401/06 , C07D401/12 , C07D401/14 , A61K31/506 , A61P1/00 , A61P1/06
CPC分类号: C07D239/545 , C07D251/20 , C07D251/34 , C07D251/38 , C07D251/46 , C07D403/12
摘要: The present invention relates to certain novel compounds of Formula (I): and methods for preparing these compounds, compositions, intermediates and derivatives thereof and for the treatment of prokineticin 1 or prokinetin 1 receptor mediated disorders.
摘要翻译: 本发明涉及某些新的式(I)化合物:以及制备这些化合物,组合物,中间体及其衍生物以及用于治疗促动蛋白原1或原激素1受体介导的病症的方法。
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公开(公告)号:US07968710B2
公开(公告)日:2011-06-28
申请号:US11375407
申请日:2006-03-14
申请人: Steven J. Coats , Alexey B. Dyatkin , Wei He , Joseph Lisko , Tamara A. Miskowski , Janet L. Ralbovsky , Mark J. Schulz
发明人: Steven J. Coats , Alexey B. Dyatkin , Wei He , Joseph Lisko , Tamara A. Miskowski , Janet L. Ralbovsky , Mark J. Schulz
IPC分类号: C07D251/30 , C07D401/06 , C07D401/14 , C07D403/06 , C07D403/14 , C07D401/12 , C07D403/12 , A61K31/53 , A61P1/12 , A61P1/06 , A61P1/00
CPC分类号: C07D239/545 , C07D251/20 , C07D251/34 , C07D251/38 , C07D251/46 , C07D403/12
摘要: The present invention relates to certain novel compounds of Formula (I): and methods for preparing these compounds, compositions, intermediates and derivatives thereof and for the treatment of prokineticin 1 or prokinetin 1 receptor mediated disorders.
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公开(公告)号:US07902358B2
公开(公告)日:2011-03-08
申请号:US11647091
申请日:2006-12-28
申请人: Steven J. Coats , Alexey B. Dyatkin , Wei He , Joseph Lisko , Tamara Miskowski , Janet L. Ralbovsky , Mark Schulz
发明人: Steven J. Coats , Alexey B. Dyatkin , Wei He , Joseph Lisko , Tamara Miskowski , Janet L. Ralbovsky , Mark Schulz
IPC分类号: C07D401/06 , C07D401/12 , C07D401/14 , C07D403/06 , C07D403/12 , C07D403/14 , A61K31/506 , A61P1/00 , A61P1/06
CPC分类号: C07D251/26 , C07D251/46 , C07D401/06 , C07D401/12 , C07D403/12 , C07D405/06 , C07D405/14 , C07D417/14 , C07D487/04
摘要: The present invention relates to certain novel compounds of Formula (I): and methods for preparing these compounds, compositions, intermediates and derivatives thereof and for the treatment of prokineticin 1 or prokinetin 1 receptor mediated disorders.
摘要翻译: 本发明涉及某些新的式(I)化合物:以及制备这些化合物,组合物,中间体及其衍生物以及用于治疗促动蛋白原1或原激素1受体介导的病症的方法。
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公开(公告)号:US20080287445A1
公开(公告)日:2008-11-20
申请号:US11646957
申请日:2006-12-28
申请人: Steven J. Coats , Alexey B. Dyatkin , Wei He , Joseph Lisko , Tamara Miskowski , Janet L. Ralbovsky , Mark Schulz
发明人: Steven J. Coats , Alexey B. Dyatkin , Wei He , Joseph Lisko , Tamara Miskowski , Janet L. Ralbovsky , Mark Schulz
IPC分类号: A61K31/505 , A61K31/435 , A61P1/00 , A61K31/53
CPC分类号: A61K31/506 , A61K31/53
摘要: The present invention relates to certain novel compounds of Formula (I): and methods for the treatment of prokineticin 2 or prokinetin 2 receptor mediated disorders.
摘要翻译: 本发明涉及某些新的式(I)化合物:以及用于治疗促动蛋白原2或原激素2受体介导的病症的方法。
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公开(公告)号:US20080269225A1
公开(公告)日:2008-10-30
申请号:US11647091
申请日:2006-12-28
申请人: Steven J. Coats , Alexey B. Dyatkin , Wei He , Joseph Lisko , Tamara Miskowski , Janet L. Ralbovsky , Mark Schulz
发明人: Steven J. Coats , Alexey B. Dyatkin , Wei He , Joseph Lisko , Tamara Miskowski , Janet L. Ralbovsky , Mark Schulz
IPC分类号: A61K31/53 , C07D405/12 , A61P29/00 , A61P1/00
CPC分类号: C07D251/26 , C07D251/46 , C07D401/06 , C07D401/12 , C07D403/12 , C07D405/06 , C07D405/14 , C07D417/14 , C07D487/04
摘要: The present invention relates to certain novel compounds of Formula (I): and methods for preparing these compounds, compositions, intermediates and derivatives thereof and for the treatment of prokineticin 1 or prokinetin 1 receptor mediated disorders.
摘要翻译: 本发明涉及某些新的式(I)化合物:以及制备这些化合物,组合物,中间体及其衍生物以及用于治疗促动蛋白原1或原激素1受体介导的病症的方法。
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公开(公告)号:US20120028997A1
公开(公告)日:2012-02-02
申请号:US12970461
申请日:2010-12-16
申请人: Steven J. Coats , Alexey B. Dyatkin , Wei He , Joseph Lisko , Tamara Miskowski , Janet L. Ralbovsky , Mark Schulz
发明人: Steven J. Coats , Alexey B. Dyatkin , Wei He , Joseph Lisko , Tamara Miskowski , Janet L. Ralbovsky , Mark Schulz
IPC分类号: A61K31/515 , C07D401/06 , C07D403/12 , A61P1/12 , A61P1/00 , A61P35/00 , A61P29/00 , C07D401/12 , A61K31/513
CPC分类号: C07D251/26 , C07D251/46 , C07D401/06 , C07D401/12 , C07D403/12 , C07D405/06 , C07D405/14 , C07D417/14 , C07D487/04
摘要: The present invention relates to certain novel compounds of Formula (I): and methods for preparing these compounds, compositions, intermediates and derivatives thereof and for the treatment of prokineticin 1 or prokinetin 1 receptor mediated disorders.
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