公开(公告)号：US20160280651A1

公开(公告)日：2016-09-29

申请号：US14899089

申请日：2014-06-27

申请人： THE REGENTS OF THE UNIVERSITY OF CALIFORNIA ,  SYNGENTA PARTICIPATIONS AG

发明人： Sean R. CUTLER ,  Sebastian Volker WENDEBORN ,  Pierre Joseph JUNG ,  Mathilde Denise LACHIA ,  Raphael DUMEUNIER

IPC分类号： C07D215/227 ,  A01N43/42

CPC分类号： C07D215/227 ,  A01N43/42 ,  C07D215/22

摘要： The present invention provides agonist compounds that active ABA receptors, and agricultural formulations comprising the agonist compounds. The agricultural formulations are useful for inducing ABA responses in plant vegetative tissues, reducing abiotic stress in plants, and inhibiting germination of plant seeds. The compounds are also useful for inducing expression of ABA-responsive genes in cells that express endogenous or heterologous ABA receptors.

摘要翻译： 本发明提供了活性ABA受体的激动剂化合物和包含激动剂化合物的农业制剂。 农业制剂可用于在植物营养组织中诱导ABA应答，减少植物中的非生物胁迫并抑制植物种子的萌发。 该化合物也可用于在表达内源性或异源性ABA受体的细胞中诱导ABA反应基因的表达。

公开(公告)号：US20160108001A1

公开(公告)日：2016-04-21

申请号：US14892386

申请日：2014-06-19

申请人： SYNGENTA PARTICIPATIONS AG

发明人： Raphael DUMEUNIER ,  Jilali KESSABI ,  Sebastian Volker WENDEBORN ,  Hannes NUSSBAUMER

IPC分类号： C07D231/14 ,  C07C239/20

CPC分类号： C07D231/14 ,  C07C239/20

摘要： The present invention relates to a process for the enantioselective preparation of the compound of formula (Ib), which process comprises a) reducing the (E)- or (Z)-form of a compound of formula (II), with an enantioselective reagent to a compound of formula (IIIa), and b) acylating the compound of formula (IIIa) with the compound of formula (IV), or c) coupling the compound of formula (IV) with the compound of formula (II), to give a compound of formula (V) and d) reducing compound of formula (V) in the presence of hydrogen, a catalyst and a chiral ligand, to the compound of formula (Ib).

摘要翻译： 本发明涉及式（Ib）化合物的对映选择性制备方法，该方法包括a）用对映选择性试剂还原式（II）化合物的（E） - 或（Z） 与式（Ⅳa）化合物反应，和b）用式（Ⅳ）化合物酰化式（Ⅳa）化合物，或c）将式（Ⅳ）化合物与式（Ⅳ）化合物偶合至 在式（Ⅴ）化合物的存在下，在式（Ⅴ）化合物和d）还原式（Ⅴ）化合物的存在下，将式（Ⅴ）化合物和d）还原化合物在氢气，催化剂和手性配体的存在下反应。

公开(公告)号：US20200315175A1

公开(公告)日：2020-10-08

申请号：US16759147

申请日：2018-10-24

申请人： Syngenta Participations AG

发明人： Ottmar Franz HUETER ,  Mark HOPPE ,  Tomas SMEJKAL ,  Raphael DUMEUNIER ,  Nicolas FEDOU ,  Edouard GODINEAU ,  Philip WEGE ,  Peter MAIENFISCH

IPC分类号： A01N43/78 ,  C07D277/34

摘要： The present inventions concerns use of a specific methoxyacrylate compound to control mosquitoes, and vector control products comprising that methoxyacrylate compound, in particular the invention relates to a substrate, to a composition, for controlling mosquitoes, and to a specific methoxyacrylate compound, processes for the synthesis of mosquitocidal methoxyacrylate compounds and new intermediates.