Thiadiazole derivative, process for producing it and agricultural and
horticultural fungicide using it as an active ingredient
    6.
    发明授权
    Thiadiazole derivative, process for producing it and agricultural and horticultural fungicide using it as an active ingredient 失效
    噻二唑衍生物,其生产方法和农业和园艺用杀真菌剂作为活性成分

    公开(公告)号:US5478849A

    公开(公告)日:1995-12-26

    申请号:US230789

    申请日:1994-04-21

    摘要: Disclosed is (a) 1,2,5-thiadiazole derivatives represented by the following formulae [I] or [III]: ##STR1## wherein X and Y are the same or different and each represents a hydrogen atom, a halogen atom, an alkyl group having from 1 to 6 carbon atoms, an alkoxy group having from 1 to 4 carbon atoms, a nitro group, a trifluoromethyl group, a carboxyl group, an alkoxycarbonyl group having from 2 to 5 carbon atoms, a naphthyl group or a tetrahydronaphthyl group; and A represents an alkyl group having from 1 to 6 carbon atoms, --C(.dbd.O)OR.sup.1, --C(.dbd.O)NR.sup.2 R.sup.3, a phenyl group which may be substituted by at least one of an alkyl group having from 1 to 6 carbon atoms and an alkoxy group having from 1 to 4 carbon atoms, --CHR.sup.4 C(.dbd.O)R.sup.5 or --C(.dbd.O)R.sup.6, in which R.sup.1 represents an alkyl group having from 1 to 6 carbon atoms, R.sup.2 and R.sup.3 are the same or different and each represents a hydrogen atom or an alkyl group having from 1 to 6 carbon atoms, R.sup.4 represents a hydrogen atom or an alkyl group having from 1 to 4 carbon atoms, R.sup.5 represents an alkoxy group having from 1 to 4 carbon atoms or an amino group which may be substituted by at least one of an alkyl group having from 1 to 4 carbon atoms and a phenyl group which may be substituted by at least one halogen atom, and R.sup.6 represents an alkyl group having from 1 to 6 carbon atoms, (b) a process for producing the compound represented by formula [I] and (c) an agricultural and horticultural fungicide comprising the compound represented by formula [III].

    摘要翻译: 公开了(a)由下式[I]或[III]表示的1,2,5-噻二唑衍生物:相同或不同,表示氢原子,卤素原子,1〜6的烷基 碳原子,具有1至4个碳原子的烷氧基,硝基,三氟甲基,羧基,具有2至5个碳原子的烷氧基羰基,萘基或四氢萘基; 并且A表示具有1至6个碳原子的烷基,-C(= O)OR 1,-C(= O)NR 2 R 3,可被至少一个具有1-6个碳原子的烷基取代的苯基 碳原子和具有1至4个碳原子的烷氧基,-CHR 4 C(= O)R 5或-C(= O)R 6,其中R 1表示具有1至6个碳原子的烷基,R 2和R 3为 相同或不同,各自表示氢原子或具有1至6个碳原子的烷基,R 4表示氢原子或具有1至4个碳原子的烷基,R 5表示具有1至4个碳原子的烷氧基 或可被至少一个具有1至4个碳原子的烷基和可被至少一个卤素原子取代的苯基取代的氨基,R 6表示具有1至6个碳原子的烷基 原子,(b)由式[I]和(c)代表的化合物的制备方法,包括该组合物的农业和园艺杀真菌剂 并由式[III]表示。