公开(公告)号：WO2011042860A3

公开(公告)日：2011-04-14

申请号：PCT/IB2010/054496

申请日：2010-10-05

Applicant: CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE ,  MEIJER, Laurent ,  KUNICK, Conrad ,  BRANDT, Wiebke ,  DOERIG, Christian ,  TECHNISCHE UNIVERSITAT CAROLO-WILHELMINA ZU BRAUNSCHWEIG

Inventor： MEIJER, Laurent ,  KUNICK, Conrad ,  BRANDT, Wiebke ,  DOERIG, Christian

IPC: C07D495/04 ,  C07D495/14 ,  A61K31/4365 ,  A61K31/519 ,  A61P33/06

Abstract: 51 ABSTRACT New derivatives of thieno[2,3-b]pyridine and 5,6,7,8-tetrahydrothieno[2,3-b]quinoline in 5 particular useful in the treatment of malaria The present invention is related to compounds of formula (I) N S R1 R2 R4 R3Ar AA' (I)10 in particular useful for the treatment of malaria, and to pharmaceutical compositions containing them.

公开(公告)号：WO2011042860A2

公开(公告)日：2011-04-14

申请号：PCT/IB2010054496

申请日：2010-10-05

Applicant: CENTRE NAT RECH SCIENT ,  MEIJER LAURENT ,  KUNICK CONRAD ,  BRANDT WIEBKE ,  DOERIG CHRISTIAN ,  TECH UNI CAROLO WILHELMINA ZU BRAUNSCHWEIG

Inventor： MEIJER LAURENT ,  KUNICK CONRAD ,  BRANDT WIEBKE ,  DOERIG CHRISTIAN

IPC: C07D495/04 ,  A61K31/4365 ,  A61K31/519 ,  A61P33/06 ,  C07D495/14

CPC classification number: C07D495/04 ,  C07D495/14

Abstract: 51 ABSTRACT New derivatives of thieno[2,3-b]pyridine and 5,6,7,8-tetrahydrothieno[2,3-b]quinoline in 5 particular useful in the treatment of malaria The present invention is related to compounds of formula (I) N S R1 R2 R4 R3Ar AA' (I)10 in particular useful for the treatment of malaria, and to pharmaceutical compositions containing them.

Abstract translation: 51摘要特别可用于治疗疟疾的噻吩并[2,3-b]吡啶和5,6,7,8-四氢噻吩并[2,3-b]喹啉的新衍生物本发明涉及式 （I）NS R1 R2 R4 R3Ar AA'（I）10特别可用于治疗疟疾，以及含有它们的药物组合物。