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1.
公开(公告)号:WO2011063293A1
公开(公告)日:2011-05-26
申请号:PCT/US2010/057515
申请日:2010-11-19
Applicant: ANACOR PHARMACEUTICALS, INC. , ZHANG, Yong-kang , ZHOU, Huchen , DING, Charles , PLATTNER, Jacob, J. , FREUND, Yvonne
Inventor: ZHANG, Yong-kang , ZHOU, Huchen , DING, Charles , PLATTNER, Jacob, J. , FREUND, Yvonne
CPC classification number: C07F5/025
Abstract: This invention provides, among other things, novel compounds useful for treating helminth infections, pharmaceutical compositions containing such compounds, as well as combinations of these compounds with at least one additional therapeutically effective agent.
Abstract translation: 本发明尤其提供了用于治疗蠕虫感染的新化合物,含有这些化合物的药物组合物,以及这些化合物与至少一种另外的治疗有效药物的组合。
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2.
公开(公告)号:WO2014121124A1
公开(公告)日:2014-08-07
申请号:PCT/US2014/014266
申请日:2014-01-31
Applicant: ANACOR PHARMACEUTICALS, INC. , AKAMA, Tsutomu , EASOM, Eric , FREUND, Yvonne , PLATTNER, Jacob, J. , SLIGAR, Jessica , CHEN, Daitao , FREEMAN, Jennifer , PERALES, Joe
Inventor: AKAMA, Tsutomu , EASOM, Eric , FREUND, Yvonne , PLATTNER, Jacob, J. , SLIGAR, Jessica , CHEN, Daitao , FREEMAN, Jennifer , PERALES, Joe
Abstract: This invention provides, among other things, novel compounds useful for treating protozoal infections, pharmaceutical compositions containing such compounds, as well as combinations of these compounds with at least one additional therapeutically effective agent.
Abstract translation: 本发明尤其提供了可用于治疗原生动物感染的新化合物,含有这些化合物的药物组合物,以及这些化合物与至少一种另外的治疗有效药物的组合。
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公开(公告)号:WO2007095638A3
公开(公告)日:2007-08-23
申请号:PCT/US2007/062350
申请日:2007-02-16
Applicant: ANACOR PHARMACEUTICALS, INC. , BAKER, Stephen, J. , SANDERS, Virginia , AKAMA, Tsutomu , BELLINGER-KAWAHARA, Carolyn , FREUND, Yvonne , MAPLES, Kirk, R. , PLATTNER, Jacob, J. , ZHANG, Yong-Kang , ZHOU, Huchen , HERNANDEZ, Vincent, S.
Inventor: BAKER, Stephen, J. , SANDERS, Virginia , AKAMA, Tsutomu , BELLINGER-KAWAHARA, Carolyn , FREUND, Yvonne , MAPLES, Kirk, R. , PLATTNER, Jacob, J. , ZHANG, Yong-Kang , ZHOU, Huchen , HERNANDEZ, Vincent, S.
Abstract: Methods of treating anti-inflammatory conditions through the use of boron-containing small molecules are disclosed.
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4.BORON-CONTAINING SMALL MOLECULES AS ANTI-INFLAMMATORY AGENTS 审中-公开
Title translation: 含有BORON的小分子作为抗炎剂公开(公告)号:WO2007095638A2
公开(公告)日:2007-08-23
申请号:PCT/US2007062350
申请日:2007-02-16
Applicant: ANACOR PHARMACEUTICALS INC , BAKER STEPHEN J , SANDERS VIRGINIA , AKAMA TSUTOMU , BELLINGER-KAWAHARA CAROLYN , FREUND YVONNE , MAPLES KIRK R , PLATTNER JACOB J , ZHANG YONG-KANG , ZHOU HUCHEN , HERNANDEZ VINCENT S
Inventor: BAKER STEPHEN J , SANDERS VIRGINIA , AKAMA TSUTOMU , BELLINGER-KAWAHARA CAROLYN , FREUND YVONNE , MAPLES KIRK R , PLATTNER JACOB J , ZHANG YONG-KANG , ZHOU HUCHEN , HERNANDEZ VINCENT S
Abstract: Methods of treating anti-inflammatory conditions through the use of boron-containing small molecules are disclosed.
Abstract translation: 公开了通过使用含硼小分子治疗抗炎症状况的方法。
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5.
公开(公告)号:WO2009111676A8
公开(公告)日:2010-09-30
申请号:PCT/US2009036250
申请日:2009-03-05
Applicant: ANACOR PHARMACEUTICALS INC , AKAMA TSUTOMU , ZHANG YONG-KANG , DING CHARLES Z , PLATTNER JACOB J , MAPLES KIRK R , FREUND YVONNE , SANDERS VIRGINIA , XIA YI , BAKER STEPHEN J , NIEMANN JAMES A , LU XIAOSONG , SALES MARCELO , SHARMA RASHMI , SINGH RAJESHWAR , JACOBS ROBERT , CHEN DAITAO , ALLEY MICHAEL RICHARD KEVIN
Inventor: AKAMA TSUTOMU , ZHANG YONG-KANG , DING CHARLES Z , PLATTNER JACOB J , MAPLES KIRK R , FREUND YVONNE , SANDERS VIRGINIA , XIA YI , BAKER STEPHEN J , NIEMANN JAMES A , LU XIAOSONG , SALES MARCELO , SHARMA RASHMI , SINGH RAJESHWAR , JACOBS ROBERT , CHEN DAITAO , ALLEY MICHAEL RICHARD KEVIN
IPC: A61K31/69
CPC classification number: C07F5/025
Abstract: Compounds and methods of treating anti-inflammatory conditions are disclosed.
Abstract translation: 公开了治疗抗炎症的化合物和方法。
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6.BORON-CONTAINING SMALL MOLECULES AS ANTI-INFLAMMATORY AGENTS 审中-公开
Title translation: 含有BORON的小分子作为抗炎剂公开(公告)号:WO2009111676A3
公开(公告)日:2010-04-01
申请号:PCT/US2009036250
申请日:2009-03-05
Applicant: ANACOR PHARMACEUTICALS INC , AKAMA TSUTOMU , ZHANG YONG-KANG , DING CHARLES Z , PLATTNER JACOB J , MAPLES KIRK R , FREUND YVONNE , SANDERS VIRGINIA , XIA YI , BAKER STEPHEN J , NIEMANN JAMES A , LU XIAOSONG , SALES MARCELO , SHARMA RASHMI , SINGH RAJESHWAR , JACOBS ROBERT , CHEN DAITAO , ALLEY MICHAEL RICHARD KEVIN
Inventor: AKAMA TSUTOMU , ZHANG YONG-KANG , DING CHARLES Z , PLATTNER JACOB J , MAPLES KIRK R , FREUND YVONNE , SANDERS VIRGINIA , XIA YI , BAKER STEPHEN J , NIEMANN JAMES A , LU XIAOSONG , SALES MARCELO , SHARMA RASHMI , SINGH RAJESHWAR , JACOBS ROBERT , CHEN DAITAO , ALLEY MICHAEL RICHARD KEVIN
IPC: A61K31/69
CPC classification number: C07F5/025
Abstract: Compounds and methods of treating anti-inflammatory conditions are disclosed.
Abstract translation: 公开了治疗抗炎症状的化合物和方法。
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7.BORON-CONTAINING SMALL MOLECULES AS ANTI-INFLAMMATORY AGENTS 审中-公开
Title translation: 含有BORON的小分子作为抗炎剂公开(公告)号:WO2009111676A2
公开(公告)日:2009-09-11
申请号:PCT/US2009/036250
申请日:2009-03-05
Applicant: ANACOR PHARMACEUTICALS, INC , AKAMA, Tsutomu , ZHANG, Yong-kang , DING, Charles, Z. , PLATTNER, Jacob, J. , MAPLES, Kirk, R. , FREUND, Yvonne , SANDERS, Virginia , XIA, Yi , BAKER, Stephen, J. , NIEMANN, James, A , LU, Xiaosong , SALES, Marcelo , SHARMA, Rashmi , SINGH, Rajeshwar , JACOBS, Robert , CHEN, Daitao , ALLEY, Michael, Richard Kevin
Inventor: AKAMA, Tsutomu , ZHANG, Yong-kang , DING, Charles, Z. , PLATTNER, Jacob, J. , MAPLES, Kirk, R. , FREUND, Yvonne , SANDERS, Virginia , XIA, Yi , BAKER, Stephen, J. , NIEMANN, James, A , LU, Xiaosong , SALES, Marcelo , SHARMA, Rashmi , SINGH, Rajeshwar , JACOBS, Robert , CHEN, Daitao , ALLEY, Michael, Richard Kevin
IPC: A61K31/69
CPC classification number: C07F5/025
Abstract: Compounds and methods of treating anti-inflammatory conditions are disclosed.
Abstract translation: 公开了治疗抗炎症状的化合物和方法。
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