利索-全球专利检索

  1. 登录
  2. 注册

搜索结果

84 条记录 (耗时 0.017 秒)

    MICROBIOCIDAL HETEROCYCLES
    2.
    发明申请
    MICROBIOCIDAL HETEROCYCLES 审中-公开
    微生物杂环

    公开(公告)号：WO2011018415A3

    公开(公告)日：2011-08-18

    申请号：PCT/EP2010061464

    申请日：2010-08-06

    申请人： SYNGENTA PARTICIPATIONS AG ,  SULZER SARAH ,  LAMBERTH CLEMENS ,  QUARANTA LAURA ,  RESPONDEK MATHIAS STEPHAN

    发明人： SULZER SARAH ,  LAMBERTH CLEMENS ,  QUARANTA LAURA ,  RESPONDEK MATHIAS STEPHAN

    IPC分类号： C07D231/12 ,  C07D401/04 ,  C07D401/06 ,  C07D401/12 ,  C07D401/14

    CPC分类号： C07D401/14 ,  C07D231/12 ,  C07D401/04 ,  C07D401/06 ,  C07D401/12

    摘要： The present invention relates to heterocyclic compounds of formula I which have microbiocidal activity, in particular fungicidal activity as well as methods of using the compounds of formula (I) to control microbes: wherein A is x-C(R10R11)-C(=O)-, x-C(R12R13)-C(=S)-, x-O-C(=O)-, x-O-C(=S)-, x-N(R14)-C(=O)-, x-N(R15)-C(=S)-,x-C(R16R17)-SO2- or X-N=C(R30)-,, in each case x indicates the bond that is connected to R1; T is CR18 or N; Y1, Y2, Y3, and Y4 are independently CR19 or N; Q is O or S; n is 1 or 2; p is 1 or 2, providing that when n is 2, p is 1. R1 is phenyl, pyridyl, imidazolyl, or pyrazolyl; wherein the phenyl, pyridyl, imidazolyl and pyrazolyl are each optionally substituted by 1 to 3 substituents independently selected from C1-C4 alkyl, C1-C4 haloalkyl, halogen, cyano, hydroxy and amino; R2, R3, R4, R5, R6, R7, R10, R11, R12, R13, R16, R17, R18,R19 and R30 each independently are hydrogen, halogen, cyano, C1-C4alkyl, or C1-C4haloalkyl; R8, R14 and R15 each independently are hydrogen or C1-C4alkyl; and R9 is phenyl, benzyl or group (a): wherein the phenyl, benzyl and group (a) are each optionally substituted with 1 to 3 substituents independently selected from C1-C4 alkyl, C1-C4 haloalkyl, halogen, cyano, hydroxy and amino; or a salt or a N-oxide thereof.

    摘要翻译： 本发明涉及具有杀微生物活性，特别是杀真菌活性的式I杂环化合物以及使用式（I）化合物控制微生物的方法：其中A是xC（R 10 R 11）-C（= O） - ，xC（R 12 R 13）-C（= S） - ，xOC（= O） - ，xOC（= S） - ，xN（R 14）-C（= O） ，xC（R 16 R 17）-SO 2 - 或XN = C（R 30） - ，在每种情况下，x表示连接至R 1的键; T是CR18或N; Y1，Y2，Y3和Y4独立地为CR19或N; Q是O或S; n是1或2; p是1或2，条件是当n是2时，p是1。 其中所述苯基，吡啶基，咪唑基和吡唑基各自任选被1至3个独立地选自C 1 -C 4烷基，C 1 -C 4卤代烷基，卤素，氰基，羟基和氨基的取代基取代; R2，R3，R4，R5，R6，R7，R10，R11，R12，R13，R16，R17，R18，R19和R30各自独立地为氢，卤素，氰基，C1-4烷基或C1-4卤代烷基; R8，R14和R15各自独立地为氢或C1-C4烷基; （a）：其中苯基，苄基和基团（a）各自任选被1至3个取代基取代，所述取代基独立地选自C 1 -C 4烷基，C 1 -C 4卤代烷基，卤素，氰基，羟基和 氨基; 或其盐或N-氧化物。

    MICROBIOCIDAL HETEROCYCLES
    3.
    发明申请
    MICROBIOCIDAL HETEROCYCLES 审中-公开
    微生物杂交

    公开(公告)号：WO2011018415A2

    公开(公告)日：2011-02-17

    申请号：PCT/EP2010/061464

    申请日：2010-08-06

    申请人： SYNGENTA PARTICIPATIONS AG ,  SULZER, Sarah ,  LAMBERTH, Clemens ,  QUARANTA, Laura ,  RESPONDEK, Mathias, Stephan

    发明人： SULZER, Sarah ,  LAMBERTH, Clemens ,  QUARANTA, Laura ,  RESPONDEK, Mathias, Stephan

    CPC分类号： C07D401/14 ,  C07D231/12 ,  C07D401/04 ,  C07D401/06 ,  C07D401/12

    摘要： The present invention relates to heterocyclic compounds of formula I which have microbiocidal activity, in particular fungicidal activity as well as methods of using the compounds of formula (I) to control microbes: wherein A is x-C(R 10 R 11 )-C(=O)-, x-C(R 12 R 13 )-C(=S)-, x-O-C(=O)-, x-O-C(=S)-, x-N(R 14 )-C(=O)-, x-N(R 15 )-C(=S)-,x-C(R 16 R 17 )-SO 2 - or X-N=C(R 30 )-,, in each case x indicates the bond that is connected to R 1 ; T is CR 18 or N; Y 1 , Y 2 , Y 3 , and Y 4 are independently CR 19 or N; Q is O or S; n is 1 or 2; p is 1 or 2, providing that when n is 2, p is 1. R 1 is phenyl, pyridyl, imidazolyl, or pyrazolyl; wherein the phenyl, pyridyl, imidazolyl and pyrazolyl are each optionally substituted by 1 to 3 substituents independently selected from C 1 -C 4 alkyl, C 1 -C 4 haloalkyl, halogen, cyano, hydroxy and amino; R 2 , R 3 , R 4 , R 5 , R 6 , R 7 , R 10 , R 11 , R 12 , R 13 , R 16 , R 17 , R 18 ,R 19 and R 30 each independently are hydrogen, halogen, cyano, C 1 -C 4 alkyl, or C 1 -C 4 haloalkyl; R 8 , R 14 and R 15 each independently are hydrogen or C 1 -C 4 alkyl; and R 9 is phenyl, benzyl or group (a): wherein the phenyl, benzyl and group (a) are each optionally substituted with 1 to 3 substituents independently selected from C 1 -C 4 alkyl, C 1 -C 4 haloalkyl, halogen, cyano, hydroxy and amino; or a salt or a N-oxide thereof.

    摘要翻译： 本发明涉及具有杀微生物活性，特别是杀真菌活性的式I的杂环化合物以及使用式（I）化合物来控制微生物的方法：其中A是xC（R10R11）-C（= O） - ，xC（R12R13）-C（= S） - ，xOC（= O） - ，xOC（= S） - ，xN（R14）-C（= O） - ，xN（R15）-C（= S） ，xC（R16R17）-SO2-或XN = C（R30） - ，在各种情况下，x表示与R1连接的键; T为CR18或N; Y1，Y2，Y3和Y4独立地为CR19或N; Q是O或S; n为1或2; p为1或2，条件是当n为2时，p为1. R1为苯基，吡啶基，咪唑基或吡唑基; 其中苯基，吡啶基，咪唑基和吡唑基各自任选被1至3个独立地选自C 1 -C 4烷基，C 1 -C 4卤代烷基，卤素，氰基，羟基和氨基的取代基取代; R2，R3，R4，R5，R6，R7，R10，R11，R12，R13，R16，R17，R18，R19和R30各自独立地为氢，卤素，氰基，C1-C4烷基或C1-C4卤代烷基; R8，R14和R15各自独立地为氢或C1-C4烷基; 并且R 9为苯基，苄基或基团（a）：其中苯基，苄基和基团（a）各自任选被1至3个独立地选自C 1 -C 4烷基，C 1 -C 4卤代烷基，卤素，氰基，羟基和 氨基; 或其盐或N-氧化物。

    PROCESS FOR THE PRODUCTION OF NITROBENZOLES
    8.
    发明申请
    PROCESS FOR THE PRODUCTION OF NITROBENZOLES 审中-公开
    生产硝基苯酚的方法

    公开(公告)号：WO2006087222A1

    公开(公告)日：2006-08-24

    申请号：PCT/EP2006/001507

    申请日：2006-02-20

    申请人： SYNGENTA PARTICIPATIONS AG ,  WALTER, Harald ,  CORSI, Camilla ,  EHRENFREUND, Josef ,  LAMBERTH, Clemens ,  SCHNEIDER, Hermann ,  TOBLER, Hans

    发明人： WALTER, Harald ,  CORSI, Camilla ,  EHRENFREUND, Josef ,  LAMBERTH, Clemens ,  SCHNEIDER, Hermann ,  TOBLER, Hans

    IPC分类号： C07C201/12 ,  C07C205/06 ,  C07C205/19 ,  C07C309/65 ,  A01N33/18

    CPC分类号： C07C201/12 ,  C07C303/28 ,  C07C309/65 ,  C07C2601/02 ,  C07C205/06 ,  C07C205/11 ,  C07C205/19 ,  C07C205/45

    摘要： The present invention relates to a process for the preparation of compounds of formula (I) wherein the substituents are as defined in claim 1 , by a) reaction of a compound of formula (II) wherein the substituents are as defined in claim 1 , with a reducing agent to form a compound of formula (III) wherein the substituents are as defined in claim 1 , and b) reaction of that compound either b1 ) with triphenylphosphine dibromide or triphenylphosphine dichloride or b2) with RSO2CI, wherein R is Ci-C4alkyl, CrC4fluoroalkyl, benzyl, phenyl, nitrophenyl, halophenyl or CrC6alkylphenyl, in the presence of a base, to form a compound of formula (IV) wherein the substituents are as defined in claim 1 ; and c) conversion of that compound in the presence of a base into a compound of formula (I); and also to novel nitrobenzene intermediates for use in that process.

    摘要翻译： 本发明涉及一种制备式（I）化合物的方法，其中取代基如权利要求1所定义，通过a）将式（Ⅱ）化合物（其中取代基如权利要求1所定义）与 还原剂形成式（III）的化合物，其中取代基如权利要求1所定义，和b）该化合物b1）与三苯基膦二溴化物或三苯基膦二氯化物或b2）与RSO2Cl的反应，其中R是C 1 -C 4烷基 ，C 1 -C 4氟烷基，苄基，苯基，硝基苯基，卤代苯基或C 1 -C 6烷基苯基，以形成式（IV）的化合物，其中取代基如权利要求1所定义; 和c）将所述化合物在碱存在下转化为式（I）的化合物; 以及用于该方法的新型硝基苯中间体。

    PROCESS FOR THE PREPARATION OF 4,4-DIFLUORO-3-OXOBUTANOIC ACID ESTERS
    9.
    发明申请
    PROCESS FOR THE PREPARATION OF 4,4-DIFLUORO-3-OXOBUTANOIC ACID ESTERS 审中-公开
    制备4,4-二氟-3-氧代戊酸的方法

    公开(公告)号：WO2006005612A1

    公开(公告)日：2006-01-19

    申请号：PCT/EP2005/007635

    申请日：2005-07-13

    申请人： SYNGENTA PARTICIPATIONS AG ,  WALTER, Harald ,  CORSI, Camilla ,  EHRENFREUND, Josef ,  LAMBERTH, Clemens ,  TOBLER, Hans

    发明人： WALTER, Harald ,  CORSI, Camilla ,  EHRENFREUND, Josef ,  LAMBERTH, Clemens ,  TOBLER, Hans

    IPC分类号： C07C67/343

    CPC分类号： C07C67/343 ,  C07C69/716

    摘要： The present invention relates to a process for the preparation of a compound of the formula (I), wherein R is C 1-12 alkyl, by the contact of a compound of the general formula (II) , wherein R 1 and R 2 are each, independently, C 1-12 alkyl; or R 1 and R 2 join together with the nitrogen atom to which they are attached to form an alicyclic amine ring containing 4 to 7 carbon atoms or a morpholine ring, with an acetic acid ester of the general formula (III) CH 3 COOR, wherein R is as defined under formula (I), in the presence of a base.

    摘要翻译： 本发明涉及制备式（I）化合物的方法，其中R是C 1-12烷基，通过通式（II）的化合物与 其中R 1和R 2各自独立地为C 1-12烷基; 或R 1和R 2 2与它们所连接的氮原子一起形成含有4至7个碳原子的脂环族胺环或吗啉环，其中 （III）CH 3 COOR的乙酸酯，其中R如式（I）所定义，在碱的存在下。