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公开(公告)号:WO2017072792A1
公开(公告)日:2017-05-04
申请号:PCT/IN2016/050364
申请日:2016-10-26
Applicant: SUN PHARMA ADVANCED RESEARCH COMPANY LIMITED
Inventor: PAL, Ranjan Kumar , SEDANI, Amit Pravinbhai , PRAJAPATI, Kaushikkumar Dhanjibhai , RANA, Dijixa Pinakin , PATHAK, Sandeep Pankajbhai , DESAI, Japan Nitinkumar , ARADHYE, Jayraj Dilipbhai , PANCHAL, Bhavesh Mohanbhai , GHOSH, Indraneel , CHITTURI, Trinadha Rao
IPC: C07D311/60 , C07D215/12 , C07D335/06
CPC classification number: C07D215/12 , C07D311/60 , C07D335/06 , C07D405/10
Abstract: The present invention provides novel heterocyclic compounds as anticancer agents, especially as estrogen receptor (ER) antagonists/ degraders and process for their preparation.
Abstract translation: 本发明提供新的杂环化合物作为抗癌剂,特别是作为雌激素受体(ER)拮抗剂/降解剂及其制备方法。 p>