公开(公告)号：WO2017072792A1

公开(公告)日：2017-05-04

申请号：PCT/IN2016/050364

申请日：2016-10-26

Applicant: SUN PHARMA ADVANCED RESEARCH COMPANY LIMITED

Inventor： PAL, Ranjan Kumar ,  SEDANI, Amit Pravinbhai ,  PRAJAPATI, Kaushikkumar Dhanjibhai ,  RANA, Dijixa Pinakin ,  PATHAK, Sandeep Pankajbhai ,  DESAI, Japan Nitinkumar ,  ARADHYE, Jayraj Dilipbhai ,  PANCHAL, Bhavesh Mohanbhai ,  GHOSH, Indraneel ,  CHITTURI, Trinadha Rao

IPC: C07D311/60 ,  C07D215/12 ,  C07D335/06

CPC classification number: C07D215/12 ,  C07D311/60 ,  C07D335/06 ,  C07D405/10

Abstract: The present invention provides novel heterocyclic compounds as anticancer agents, especially as estrogen receptor (ER) antagonists/ degraders and process for their preparation.

Abstract translation: 本发明提供新的杂环化合物作为抗癌剂，特别是作为雌激素受体（ER）拮抗剂/降解剂及其制备方法。

公开(公告)号：WO2017056115A1

公开(公告)日：2017-04-06

申请号：PCT/IN2016/050333

申请日：2016-10-01

Applicant: SUN PHARMA ADVANCED RESEARCH COMPANY LIMITED

Inventor： SAMANTA, Biswajit ,  PATEL, Poojan Kaushikbhai ,  DESAI, Megha Shringesh ,  AKOLKAR, Nakul Pramodbhai ,  ADHYAPAK, Jay Prakashchandra ,  KUMBHANI, Anil Savajibhai ,  GHOSH, Indraneel ,  CHITTURI, Trinadha Rao

IPC: C07D265/36 ,  C07D413/04 ,  C07D413/12 ,  C07D498/04

CPC classification number: C07D265/36 ,  C07D413/04 ,  C07D413/12 ,  C07D498/04

Abstract: The present invention provides novel N -aryl containing fused heterocyclic compounds as anticancer agents, especially as estrogen receptor (ER) antagonists/ degraders and process for their preparation.

Abstract translation: 本发明提供新的含N-芳基稠合杂环化合物作为抗癌剂，特别是作为雌激素受体（ER）拮抗剂/降解剂及其制备方法。