发明公开
EP2078010A2 POLYCYCLIC HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS
有权
AS AXL抑制剂SUITABLE环杂芳基取代的三唑
- 专利标题： POLYCYCLIC HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS
- 专利标题（中）： AS AXL抑制剂SUITABLE环杂芳基取代的三唑
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申请号： EP07870107.5申请日： 2007-12-29
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公开(公告)号： EP2078010A2公开(公告)日： 2009-07-15
- 发明人: GOFF, Dane , ZHANG, Jing , SINGH, Rajinder , HOLLAND, Sacha , YU, Jiaxin , HECKRODT, Thilo , DING, Pingyu , LITVAK, Joane
- 申请人： Rigel Pharmaceuticals, Inc.
- 申请人地址： 1180 Veterans Boulevard South San Francisco, CA 94080 US
- 专利权人： Rigel Pharmaceuticals, Inc.
- 当前专利权人： Rigel Pharmaceuticals, Inc.
- 当前专利权人地址： 1180 Veterans Boulevard South San Francisco, CA 94080 US
- 代理机构： Schuster, Thomas
- 优先权： US882850P 20061229; US895400P 20070316; US970931P 20070907
- 国际公布： WO2008083367 20080710
- 主分类号： C07D403/04
- IPC分类号： C07D403/04 ; C07D403/14 ; C07D471/18 ; C07D491/14 ; A61K31/4196 ; A61P19/00 ; A61P35/00 ; C07D401/14 ; C07D405/14 ; C07D417/04 ; C07D417/14 ; C07D451/04 ; C07D471/04 ; C07D487/04 ; C07D487/10 ; C07D491/04 ; C07D491/20 ; C07D495/04 ; C07D519/00
摘要：
Polycyclic heteroaryl substituted triazoles and pharmaceutical compositions containing the compounds are disclosed as being useful in inhibiting the activity of the receptor protein tyrosine kinase Axl. Methods of using the compounds in treating diseases or conditions associated with Axl activity are also disclosed.
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