发明申请
- 专利标题: 1,3-DIAMINOCYCLOPENTANE CARBOXAMIDE DERIVATIVES
- 专利标题(中): 1,3-二氨基环戊烷羧酰胺衍生物
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申请号: PCT/EP2014/001255申请日: 2014-05-09
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公开(公告)号: WO2014202168A1公开(公告)日: 2014-12-24
- 发明人: TSAKLAKIDIS, Christos , STAEHLE, Wolfgang , LEUTHNER, Birgitta , CZODROWSKI, Paul , FUCHSS, Thomas
- 申请人: MERCK PATENT GMBH
- 申请人地址: Frankfurter Strasse 250 64293 Darmstadt DE
- 专利权人: MERCK PATENT GMBH
- 当前专利权人: MERCK PATENT GMBH
- 当前专利权人地址: Frankfurter Strasse 250 64293 Darmstadt DE
- 优先权: EP13003189.1 20130621
- 主分类号: C07D413/14
- IPC分类号: C07D413/14 ; C07D309/04 ; C07D215/12 ; C07D317/50 ; C07D319/18 ; C07D231/12 ; C07D231/56 ; C07D233/26 ; C07D401/04 ; C07D235/06 ; C07D235/18 ; C07D235/26 ; C07D403/04 ; C07D413/04 ; C07D413/12
摘要:
Compounds of the formula I in which R 1 , R 4 , R 6 , R, X 1 , X 2 , X 3 , X 4 , q and W have the meanings indicated in Claim 1, are inhibitors of fatty acid synthase, and can be employed, inter alia, for the treatment of diseases such as cancer, cardiovascular diseases, central nervous system injury and different forms of inflammation.