公开(公告)号：EP2858981A1

公开(公告)日：2015-04-15

申请号：EP13727103.7

申请日：2013-05-29

Applicant: BASF SE

Inventor： WITSCHEL, Matthias ,  STELZER, Frank ,  HUTZLER, Johannes ,  QU, Tao ,  MIETZNER, Thomas ,  KREUZ, Klaus ,  GROßMANN, Klaus ,  APONTE, Raphael ,  HÖFFKEN, Hans Wolfgang ,  CALO, Frederick ,  EHRHARDT, Thomas ,  SIMON, Anja ,  PARRA RAPADO, Liliana

IPC: C07D311/94 ,  A01N43/56 ,  A61K31/4162

CPC classification number: A01N43/90 ,  A01N47/20 ,  C07D311/94 ,  C07D491/052

Abstract: The present invention relates to a pyrazolopyran of the general formula I wherein the variables are defined according to the description, including a tautomer, salt, cleavable prodrug, or mixtures thereof, in particular to said pyrazolopyran for use as a medicament and/or an inhibitor of the enzyme serinehydroxymethyltransferase (SHMT). The invention also relates to a process the preparation of a pyrazolopyran of the formula I, to compositions comprising said compound and processes for the preparation of these compositions. Further it relates to use of the pyrazolopyran of formula I as an herbicide as well as to a method of controlling undesired vegetation.

公开(公告)号：EP2550271A1

公开(公告)日：2013-01-30

申请号：EP11710739.1

申请日：2011-03-22

Applicant: BASF SE

Inventor： SONG, Dschun ,  MAJOR, Julia ,  HUTZLER, Johannes ,  NEWTON, Trevor William ,  WITSCHEL, Matthias ,  MOBERG, William Karl ,  PARRA RAPADO, Liliana ,  QU, Tao ,  STELZER, Frank ,  KLOET, Andree van der ,  SEITZ, Thomas ,  EHRHARDT, Thomas ,  KREUZ, Klaus ,  GROSSMANN, Klaus ,  MICHROWSKA-PIANOWSKA, Anna Aleksandra ,  SIMON, Anja ,  REINGRUBER, Rüdiger ,  KRAUS, Helmut ,  HÖFFKEN, Hans Wolfgang ,  MIETZNER, Thomas ,  DEGASPARI, Nilton

IPC: C07D471/04 ,  A01N43/90

CPC classification number: C07D471/04 ,  A01N43/90

Abstract: Substituted pyridines of the formula (I) in which the variables are defined according to the description, processes and intermediates for preparing the compounds of the formula (I) and their N-oxides, their agriculturally suitable salts, compositions comprising them and their use as herbicides, and also methods for controlling unwanted vegetation.

公开(公告)号：EP2437605A1

公开(公告)日：2012-04-11

申请号：EP10724420.4

申请日：2010-05-31

Applicant: BASF SE

Inventor： SONG, Dschun ,  MAJOR, Julia ,  HUTZLER, Johannes ,  NEWTON, Trevor William ,  WITSCHEL, Matthias ,  MOBERG, William Karl ,  PARRA RAPADO, Liliana ,  QU, Tao ,  STELZER, Frank ,  MICHROWSKA, Anna Aleksandra ,  SEITZ, Thomas ,  EHRHARDT, Thomas ,  KREUZ, Klaus ,  GROßMANN, Klaus ,  SIEVERNICH, Bernd ,  SIMON, Anja ,  NIGGEWEG, Ricarda

IPC: A01N43/60 ,  C07D471/04

CPC classification number: C07D471/04 ,  A01N43/90

Abstract: The invention relates to substituted pyrazines of formula (I), in which the variables are defined according to the description, the agriculturally suitable salts of said pyrazines, methods and intermediate products for producing the pyrazines of formula (I), agents containing said pyrazines and the use of said pyrazines as herbicides, i.e., to control weeds, and a method for controlling unwanted plant growth, in which a quantity of at least one pyrazine compound of formula (I) with a herbicidal action is allowed to act on plants, the seeds thereof, and/or the habitats thereof.

公开(公告)号：EP2350074A1

公开(公告)日：2011-08-03

申请号：EP09784000.3

申请日：2009-10-14

Applicant: BASF SE

Inventor： SONG, Dschun ,  HUPE, Eike ,  PILGER, Christian ,  NEWTON, Trevor, William ,  WITSCHEL, Matthias ,  MOBERG, William, Karl ,  PARRA RAPADO, Liliana ,  QU, Tao ,  STELZER, Frank ,  VESCOVI, Andrea ,  SEITZ, Thomas ,  EHRHARDT, Thomas ,  KREUZ, Klaus ,  GROSSMANN, Klaus ,  REINHARD, Robert ,  SIMON, Anja ,  NIGGEWEG, Ricarda ,  SIEVERNICH, Bernd

IPC: C07D471/04 ,  A01N43/90

CPC classification number: A01N43/90 ,  C07D471/04

Abstract: Disclosed are substituted pyridines of formula (I) in which the variables are defined as indicated in the description, the agriculturally suitable salts thereof, methods and intermediate products for manufacturing the pyridines of formula (I), substances containing said pyridines and the use thereof as herbicides, i.e. to control weeds, and a method for controlling unwanted plant growth in which a herbicidal amount of at least one pyridine compound of formula (I) is made to act on plants, the seeds and/or the habitat thereof.

公开(公告)号：EP2346849A1

公开(公告)日：2011-07-27

申请号：EP09783517.7

申请日：2009-09-29

Applicant: BASF SE

Inventor： PARRA RAPADO, Liliana ,  STELZER, Frank ,  WITSCHEL, Matthias ,  SEITZ, Thomas ,  SIMON, Anja ,  REINHARD, Robert ,  SIEVERNICH, Bernd ,  GROSSMANN, Klaus ,  EHRHARDT, Thomas ,  NEWTON, Trevor William ,  MAJOR, Julia ,  QU, Tao ,  MOBERG, William Karl ,  SONG, Dschun ,  RACK, Michael ,  FRASSETTO, Timo ,  KREUZ, Klaus

IPC: C07D401/06 ,  C07D403/06 ,  A01N43/60

CPC classification number: C07D401/06 ,  C07D403/06

Abstract: The invention relates to piperazine compounds of formula I, where the variables are defined according to the description, agriculturally suitable salts of said piperazine compounds, to a method and intermediate products for the production of the piperazine compounds of formula I, to means comprising said compounds and to the use thereof as herbicides, i.e. to combat weeds, and to a method for combating undesired plant growth wherein an amount of at least one piperazine compound of formula I large enough to have an herbicidal effect is allowed to take effect on plants, seeds and/or habitats thereof.

公开(公告)号：EP2344518A1

公开(公告)日：2011-07-20

申请号：EP09740145.9

申请日：2009-10-26

Applicant: BASF SE

Inventor： PARRA RAPADO, Liliana ,  STELZER, Frank ,  WITSCHEL, Matthias ,  SEITZ, Thomas ,  NEWTON, Trevor, William ,  MAJOR, Julia ,  QU, Tao ,  MOBERG, William, Karl ,  SONG, Dschun ,  RACK, Michael ,  FRASSETTO, Timo ,  SIMON, Anja ,  REINHARD, Robert ,  SIEVERNICH, Bernd ,  GROßMANN, Klaus ,  EHRHARDT, Thomas ,  KREUZ, Klaus

IPC: C07K5/06 ,  A01N37/46

CPC classification number: C07D241/08

Abstract: The invention relates to piperazine compounds of formula (I), where the variables are defined according to the description, to agriculturally suitable salts of said piperazine compounds, to a method and to intermediate products for producing the piperazines of formula (I), to means comprising said piperazines and to the use thereof as herbicides, i.e. for combating weeds, and to a method for combating undesired plant growth wherein an amount of at least one piperazine compound of formula (I) large enough to have a herbicidal effect is allowed to take effect on plants, seeds and/or habitats thereof.

Abstract translation: 本发明涉及式（I）的哌嗪化合物，其中变量根据说明书定义，所述哌嗪化合物的农业上合适的盐，制备式（I）的哌嗪的方法和中间产物， 其包含所述哌嗪及其作为除草剂的用途，即用于防治杂草，并且涉及防止不希望的植物生长的方法，其中允许将至少一种足够大以具有除草效果的式（I）的哌嗪化合物服用 对植物，种子和/或其栖息地的影响。

公开(公告)号：EP2054395A2

公开(公告)日：2009-05-06

申请号：EP08760877.4

申请日：2008-06-11

Applicant: Basf Se

Inventor： HUPE, Eike ,  SEITZ, Thomas ,  WITSCHEL, Matthias ,  SONG, Dschun ,  MOBERG, William Karl ,  PARRA RAPADO, Liliana ,  STELZER, Frank ,  VESCOVI, Andrea ,  NEWTON, Trevor William ,  REINHARD, Robert ,  SIEVERNICH, Bernd ,  GROSSMANN, Klaus ,  EHRHARDT, Thomas ,  RACK, Michael ,  KIBLER, Elmar

IPC: C07D241/08 ,  C07D403/10 ,  C07D407/10 ,  C07D409/10 ,  C07D413/10 ,  C07D417/10 ,  A61K31/495

CPC classification number: C07D241/08 ,  C07D403/10 ,  C07D407/10 ,  C07D409/10 ,  C07D413/10 ,  C07D417/10

Abstract: The invention relates to piperazine compounds of the following defined general formula (I) and to their use as herbicides. The invention also relates to crop protection agents and to a method for combating undesired plant growth. In formula (I), the variables are defined as follows: R1 is selected from halogen, cyano, nitro, Z-C(=O)-R11, phenyl and a 5- or 6-membered heterocyclic group that has 1, 2, 3 or 4 heteroatoms, selected from O, N and S as ring atoms, wherein phenyl and the heterocyclic group are unsubstituted or have 1, 2, 3 or 4 substituents R1a; Z stands for a covalent bond or a CH2 group; R11 represents hydrogen, C1-C6 alkyl, C3-C6 cycloalkyl, C2-C6 alkenyl, C5-C6 cycloalkenyl, C2-C6 alkynyl and similar; R2 represents hydrogen, halogen, nitro, cyano, C1-C4 alkyl, C1-C4 haloalkyl, C2- C4 alkenyl, C1-C4 alkoxy, C1-C4 haloalkoxy, benzyl or a group S(O) nR21, wherein R21 stands for C1-C4 alkyl or C1-C4 haloalkyl and n stands for 0, 1 or 2; R3 represents hydrogen or halogen; R4 represents C1-C4 alkyl, C3- C4 alkenyl or C3-C4 alkynyl; R5 represents hydrogen, C1-C4 alkyl, C3-C4 alkenyl, C3-C4 alkynyl or a group (=O)R51, wherein R51 stands for hydrogen, C1-C4 alkyl, C1-C4 haloalkyl, C1-C4 alkoxy or C1-C4 haloalkoxy; R6 stands for C1-C4 alkyl, C1-C4 hydroxy alkyl or C1-C4 haloalkyl; R7, R8 stand, independently of one another, for hydrogen, OH, C1-C4 alkoxy, C1-C4 haloalkyoxy, C1-C4 alkyl or C1-C4 haloalkyl; R9, R10 are selected, independently of one another, from hydrogen, halogen, CN, NO2, C1-C4 alkyl, C1-C4 haloalkyl, C2-C4 alkenyl, C1-C4 alkoxy and C1-C4 haloalkoxy.

Abstract translation: 本发明涉及下面定义的通式（I）的哌嗪化合物和它们作为除草剂的用途。 本发明还涉及作物保护剂和防治不希望的植物生长的方法。 在式（I）中，变量定义如下：R 1选自卤素，氰基，硝基，ZC（= O）-R 11，苯基和具有1,2,3或4个碳原子的5-或6-元杂环基团 4个选自O，N和S的杂原子作为环原子，其中苯基和杂环基未被取代或具有1,2,3或4个取代基R 1a; Z代表共价键或CH2基团; R 11代表氢，C 1 -C 6烷基，C 3 -C 6环烷基，C 2 -C 6烯基，C 5 -C 6环烯基，C 2 -C 6炔基等; R2表示氢，卤素，硝基，氰基，C1-C4烷基，C1-C4卤代烷基，C2-C4链烯基，C1-C4烷氧基，C1-C4卤代烷氧基，苄基或S（O）nR21基团， -C4烷基或C1-C4卤代烷基，n代表0,1或2; R3代表氢或卤素; R 4代表C 1 -C 4烷基，C 3 -C 4烯基或C 3 -C 4炔基; R 5代表氢，C 1 -C 4烷基，C 3 -C 4烯基，C 3 -C 4炔基或基团（= O）R 51，其中R 51代表氢，C 1 -C 4烷基，C 1 -C 4卤代烷基， C4卤代烷氧基; R6代表C1-C4烷基，C1-C4羟烷基或C1-C4卤代烷基; R 7，R 8彼此独立地代表氢，OH，C 1 -C 4烷氧基，C 1 -C 4卤代烷氧基，C 1 -C 4烷基或C 1 -C 4卤代烷基; R 9，R 10彼此独立地选自氢，卤素，CN，NO 2，C 1 -C 4烷基，C 1 -C 4卤代烷基，C 2 -C 4烯基，C 1 -C 4烷氧基和C 1 -C 4卤代烷氧基。

公开(公告)号：EP2595995A1

公开(公告)日：2013-05-29

申请号：EP11740608.2

申请日：2011-07-20

Applicant: BASF SE

Inventor： MICHROWSKA-PIANOWSKA, Anna Aleksandra ,  MAJOR, Julia ,  HUTZLER, Johannes ,  NEWTON, Trevor William ,  EVANS, Richard Roger ,  KREUZ, Klaus ,  GROßMANN, Klaus ,  SONG, Dschun ,  SIMON, Anja ,  WITSCHEL, Matthias ,  MOBERG, William Karl ,  PARRA RAPADO, Liliana ,  QU, Tao ,  STELZER, Frank ,  KRAUS, Helmut ,  SEITZ, Thomas ,  KLOET, Andree van der ,  REINGRUBER, Rüdiger

IPC: C07D498/04 ,  C07D519/00 ,  A01N43/90

CPC classification number: A01N43/90 ,  A01N43/80 ,  A01N43/84 ,  C07D498/04 ,  C07D513/04 ,  C07D519/00

Abstract: The invention relates to isoxazolo[5,4-b]pyridine compounds of formula (I), to the agriculturally useful salts of isoxazolo[5,4-b]pyridine compounds of formula (I), and to their use as herbicides.

公开(公告)号：EP2315760B1

公开(公告)日：2013-03-06

申请号：EP09780999.0

申请日：2009-07-23

Applicant: BASF SE

Inventor： PARRA RAPADO, Liliana ,  HUPE, Eike ,  WITSCHEL, Matthias ,  SEITZ, Thomas ,  SIMON, Anja ,  REINHARD, Robert ,  SIEVERNICH, Bernd ,  GROßMANN, Klaus ,  EHRHARDT, Thomas ,  NEWTON, Trevor William ,  STELZER, Frank ,  QU, Tao ,  MOBERG, William Karl ,  SONG, Dschun ,  RACK, Michael ,  FRASSETTO, Timo ,  KREUZ, Klaus ,  MAJOR, Julia

IPC: C07D401/06 ,  C07D403/06 ,  A01N43/60

CPC classification number: C07D401/06 ,  A01N43/60 ,  A01N43/78 ,  A01N43/80 ,  A01N43/82 ,  A01N43/84 ,  A01N43/90 ,  C07D403/06 ,  A01N33/18 ,  A01N43/54 ,  A01N2300/00

公开(公告)号：EP2550277A1

公开(公告)日：2013-01-30

申请号：EP11709712.1

申请日：2011-03-22

Applicant: BASF SE

Inventor： SONG, Dschun ,  MAJOR, Julia ,  HUTZLER, Johannes ,  NEWTON, Trevor William ,  WITSCHEL, Matthias ,  MOBERG, William Karl ,  PARRA RAPADO, Liliana ,  QU, Tao ,  STELZER, Frank ,  KLOET, Andree van der ,  SEITZ, Thomas ,  EHRHARDT, Thomas ,  KREUZ, Klaus ,  GROSSMANN, Klaus ,  MICHROWSKA-PIANOWSKA, Anna Aleksandra ,  SIMON, Anja ,  REINGRUBER, Rüdiger ,  KRAUS, Helmut ,  HÖFFKEN, Hans Wolfgang ,  MIETZNER, Thomas

IPC: C07D491/052 ,  A01N43/90

CPC classification number: C07D491/052 ,  A01N43/90

Abstract: Substituted pyridazines of the formula (I) in which the variables are defined according to the description, processes and intermediates for preparing the compounds of the formula (I) and their N-oxides, their agriculturally suitable salts, compositions comprising them and their use as herbicides, and also methods for controlling unwanted vegetation.

Abstract translation: 其中变量根据说明书定义的式（I）取代的哒嗪，制备式（I）化合物及其N-氧化物的方法和中间体，它们的农业上合适的盐，包含它们的组合物和它们作为 除草剂，以及防治不想要的植物的方法。