N-PHENYL-N'-PHENYLSULFONYLPIPERAZINE DERIVATIVE AND METHOD FOR PRODUCING INTERMEDIATE FOR SAME
    42.
    发明公开
    N-PHENYL-N'-PHENYLSULFONYLPIPERAZINE DERIVATIVE AND METHOD FOR PRODUCING INTERMEDIATE FOR SAME 审中-公开
    N-苯基-N'-苯磺酰基哌嗪衍生物及其制备中间体的方法

    公开(公告)号:EP2832729A1

    公开(公告)日:2015-02-04

    申请号:EP13769121.8

    申请日:2013-03-29

    IPC分类号: C07D263/32 C07B61/00

    CPC分类号: C07D263/32

    摘要: The present invention provides the salt and the crystal thereof of 2-(oxazole-2-yl)phenol derivative which are the intermediate in the process of producing N-phenyl-N'-phenylsulfonyl piperazine derivative, and the process of producing the salt as well as the process of producing N-phenyl-N'-phenylsulfonyl piperazine derivative through the salt.
    A method of producing the salt and the crystal thereof of the compound represented by Formula(I):

    wherein X is halogen;
    and the process of producing the salt as well as the process of producing N-phenyl-N'-phenylsulfonyl piperazine derivative through the salt.

    摘要翻译: 本发明提供作为制备N-苯基-N'-苯磺酰基哌嗪衍生物的方法中的中间体2-(恶唑-2-基)苯酚衍生物的盐及其晶体,以及将该盐制备为 以及通过盐制备N-苯基-N'-苯磺酰基哌嗪衍生物的方法。 由式(I)表示的化合物的盐及其晶体的制备方法:其中X是卤素; 以及生产盐的方法以及通过盐生产N-苯基-N'-苯磺酰基哌嗪衍生物的方法。