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128 条记录 (耗时 0.017 秒)

    Phenol derivatives
    63.
    发明公开
    Phenol derivatives 失效
    Phenolderivate。

    公开(公告)号：EP0124369A1

    公开(公告)日：1984-11-07

    申请号：EP84302860.6

    申请日：1984-04-27

    申请人： IMPERIAL CHEMICAL INDUSTRIES PLC

    发明人： Crawley, Graham Charles ,  Edwards, Philip Neil ,  Hill, George Beresford ,  Pilgrim, William Robert ,  Tait, Brian Steele ,  Young, Derek William

    IPC分类号： C07C149/36 ,  C07C147/14 ,  C07C147/10 ,  C07C103/76 ,  C07C103/737

    CPC分类号： C07F9/6552 ,  C07C43/225 ,  C07C43/23 ,  C07C45/305 ,  C07C45/44 ,  C07C45/46 ,  C07C45/513 ,  C07C45/60 ,  C07C45/68 ,  C07C49/755 ,  C07C59/64 ,  C07C59/72 ,  C07C62/34 ,  C07C309/00 ,  C07C317/00 ,  C07C323/00 ,  C07C2602/08 ,  C07C2602/10 ,  C07D333/60 ,  C07F7/1852 ,  C07C47/277 ,  C07C49/84

    摘要： A phenol derivative of the formula


    wherein NU is a defined bis-phenolic nucleus including a hydroxyphenyl-hydroxynaphthyl; hydroxyphenyl-hydroxy- indanyl, hydroxyphenyl-hydroxybenzothienyl or di-hydroxyethylene or vinylene nucleus;
    wherein A is alkylene, alkenylene or alkynylene which may be interrupted by phenylene or other linkages,
    wherein R 1 is hydrogen, or alkyl, alkenyl, cycloalkyl, halogenoalkyl, aryl or arylalkyl, or R 1 is joined to R 2 , and wherein X is -CONR2-, -CSNR2-, -NR 12 CO-, -NR 12 CS-, -NR 12 CONR 2- ,
    , -SO 2 NR 2 -or -CO-, or, when R is not hydrogen, is -NR 12 COO-, -S-, -SO- or -SO 2 -, wherein R 2 is hydrogen or alkyl, or R 1 and R 2 together form alkylene;
    wherein R 12 is hydrogen or alkyl, and wherein R 22 is hydrogen, cyano or nitro;
    or a salt thereof when appropriate. The compounds possess antioestrogenic activity and may be used for the treatment of hormone-dependent breast tumours or of anovulatory infertility.

    摘要翻译： 式NU-A-X-R1的酚衍生物，其中NU是包含羟基苯基 - 羟基萘基的定义的双酚核; 羟基苯基 - 羟基苯并噻吩基或二羟基苯基 - 乙烯或亚乙烯基核; 其中A是可以被亚苯基或其它键连接的亚烷基，亚烯基或亚炔基，其中R 1是氢或烷基，烯基，环烷基，卤代烷基，芳基或芳基烷基，或R 1与R 2连接，并且其中X是-CONR 2 - ，-CONR 2 - ， - NR 12 CO - ， - NR 12 CS - ， - NR 12 CONR 2 - ， - SO 2 NR 2 - 或-CO-，或者当R 1不是氢时，是-NR 12 COO - ， - S-，-SO-或 - SO 2 - ，其中R 2是氢或烷基，或者R 1和R 2一起形成亚烷基; 其中R 12是氢或烷基，并且其中R 22是氢，氰基或硝基; 或其盐。 该化合物具有抗雌激素活性，可用于治疗激素依赖性乳腺肿瘤或无排卵性不育症。

    Herbicidal cyclohexane-1,3-dione derivatives
    66.
    发明公开
    Herbicidal cyclohexane-1,3-dione derivatives 失效
    除草环己烷-1,3-二酮衍生物

    公开(公告)号：EP0082694A3

    公开(公告)日：1983-10-12

    申请号：EP82306757

    申请日：1982-12-17

    申请人： ICI AUSTRALIA LIMITED

    发明人： Serban, Alexander ,  Watson, Keith Geoffrey ,  Bird, Graham John ,  Farquharson, Graeme John ,  Houston, Timothy Leslie

    IPC分类号： C07C149/36 ,  A01N35/10 ,  A01N35/06

    CPC分类号： C07C323/00 ,  A01N35/10 ,  A01N41/06

    摘要： The invention concerns novel compounds of the formula I
    wherein:
    R' is selected from alkyl, alkenyl, alkynyl, cycloalkyl benzyl and substituted benzyl; A is selected from hydrogen, halogen, nitro, alkyl, alkoxy, alkylthio, alkenylthio, alkynylthio, cycloalkoxy, cycloalkylthio, sulfamoyl, N-(C 1 to C 6 alkyl) sulfamoyl, N,N-di(C 1 to C 6 alkyl) sulfamoyl, benzylthio and substituted benzylthio; R 2 is selected from hydrogen, alkyl, alkenyl, alkynyl, substituted alkyl, acyl, alkylsulfonyl, benzenesulfonyl, substituted benzenesulfonyl, and an inorganic or organic cation; R 3 is selected from alkyl, alkenyl, alkynyl, substituted alkyl, haloalkenyl and haloalkynyl; and R" is selected from alkyl, fluoroalkyl, alkenyl, alkynyl and phenyl. The compounds are herbicides and in further embodiments the invention provides processes for the preparation of compounds of formula I, intermediates useful in the preparation of compounds of formula I, herbicidal compositions containing as active ingredient a compound of formula I, and processes for severely damaging or killing unwanted plants by applying to the plants or to the growth medium of the plants an effective amount of a compound of formula I.

    摘要翻译： 本发明涉及新的式I化合物，其中：R'选自烷基，烯基，炔基，环烷基苄基和取代的苄基; A选自氢，卤素，硝基，烷基，烷氧基，烷硫基，烯硫基，炔硫基，环烷氧基，环烷硫基，氨磺酰基，N-（C1-C6烷基）氨磺酰基，N，N-二（C1-6烷基）氨磺酰基，苄硫基 和取代的苄硫基; R2选自氢，烷基，链烯基，炔基，取代的烷基，酰基，烷基磺酰基，苯磺酰基，取代的苯磺酰基和无机或有机阳离子; R3选自烷基，烯基，炔基，取代的烷基，卤代烯基和卤代炔基; 化合物是除草剂，并且在进一步的实施方案中，本发明提供了制备式I化合物的方法，可用于制备式I化合物的中间体，除草剂组合物 其含有作为活性成分的式I化合物，以及通过向植物或植物生长介质施用有效量的式I化合物来严重损害或杀死不想要的植物的方法。

    Polyprenyl compounds and preparation thereof
    67.
    发明公开
    Polyprenyl compounds and preparation thereof 失效
    Polyprenylverbindungen und deren Herstellung。

    公开(公告)号：EP0087638A1

    公开(公告)日：1983-09-07

    申请号：EP83101283.6

    申请日：1983-02-10

    申请人： KURARAY CO., LTD.

    发明人： Onishi, Takashi ,  Suzuki, Shigeaki ,  Mori, Fumio ,  Takigawa, Tetsuo ,  Fujita, Yoshiji ,  Mizuno, Masao ,  Nishida, Takashi

    IPC分类号： C07C147/10 ,  C07C33/02 ,  C07D309/12 ,  C07F7/18 ,  C07C149/36 ,  C07C147/14 ,  C07D317/18 ,  C07D405/12 ,  C07D417/12 ,  C07D277/16 ,  C07D213/70

    CPC分类号： C07D405/12 ,  C07C317/00 ,  C07C321/00 ,  C07D309/12 ,  C07D317/18 ,  C07D417/12 ,  C07F7/1852

    摘要： The invention relates to polyprenyl compounds of the general formula


    wherein
    represents a trans-isoprene unit,
    represents a cis-isoprene unit, n is an integer of 11-19, Z' is -CH 2 0H or a functional precursor thereof, and either one of R' and R 2 is a hydrogen atom and the other is -S(O) m R 3 in which m is an integer of 0 (zero), 1 or 2 and R 3 is a phenyl, naphthyl, pyridyl or thiazolinyl group which may optionally have one or more substituents selected from lower alkyl groups and halogen atoms. These polyprenyl compounds can be synthesized by reacting a compound of the general formula

    with a compound of the general formula
    with the aid of an anionizing agent.
    (either one of A and X being a halogen atom and the other being -S(O) m R 3 )
    These polyprenyl compounds can be converted into mammalian dolichols or precursors thereof by reductive elimination of the -S(O) m R 3 group.

    摘要翻译： 本发明涉及通式的聚异戊二烯基化合物... ...表示反异戊二烯单元，...表示顺式异戊二烯单元，n为11〜19的整数，Z 1为-CH 2 OH 或其功能性前体，R 1和R 2中的任一个为氢原子，另一个为-S（O）m R 3，其中m为0（0），1或 2和R 3是苯基，萘基，吡啶基或噻唑啉基，其可以任选地具有一个或多个选自低级烷基和卤素原子的取代基。 这些聚异戊二烯基化合物可以通过使一种通式为...的化合物与一种通式为...的化合物反应而合成... ...借助于阴离子化剂...（A和X中的任一个是卤素 原子，而另一个是-S（O）m R 3）...这些聚异戊二烯基化合物可以通过-S（O）mR 3基团的还原性消除而转化成哺乳动物多烯醇或其前体。