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1.发明授权PHTHALAZINE AND PYRIDO[3,4-D]PYRIDAZINE COMPOUNDS AS H1 RECEPTOR ANTAGONISTS 有权酞嗪和吡啶并[3,4-D]哒嗪AS H1受体拮抗剂的
公开(公告)号：EP2215082B1
公开(公告)日：2011-09-21
申请号：EP08805231.1
申请日：2008-10-10
申请人： Glaxo Group Limited
IPC分类号： C07D403/06 , C07D471/04 , A61K31/502 , A61K31/5025 , A61P29/00 , A61P37/08
CPC分类号： C07D403/06 , C07D471/04
摘要： The present invention relates to compounds of formula (I), and salts thereof, processes for their preparation, to compositions containing them and to their use in the treatment of various diseases, such as allergic rhinitis.
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公开(公告)号：EP0843671A1
公开(公告)日：1998-05-27
申请号：EP96925710.0
申请日：1996-07-11
申请人： GLAXO GROUP LIMITED
发明人： COCKERILL, George Stuart, Glaxo Wellcome plc , CARTER, Malcolm Clive, Glaxo Wellcome plc , McKEOWN, Stephen Karl, Glaxo Wellcome plc , VILE, Sadie , PAGE, Martin John, Glaxo Wellcome plc , HUDSON, Alan Thomas, Long Lodge Cottage , BARRACLOUGH, Paul , FRANZMANN, Karl Witold, 6 Northstead Road
CPC分类号： C07D401/14 , C07D403/12 , C07D405/14 , C07D491/04
摘要： The invention is directed toward substituted heteroaromatic compounds which are protein tyrosine kinase inhibitors, in particular to substituted quinolines and quinazolines. Methods for their preparation, pharmaceutical compositions including such compounds and their use in medicine, for example in the treatment of psoriasis, fibrosis, atherosclerosis, restenosis, auto-immune disease, allergy, asthma, transplantation rejection, inflammation, thrombosis, nervous system diseases, and cancer.
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3.发明公开PYRAZOLE AND TRIAZOLE CARBOXAMIDES AS CRAC CHANNEL INHIBITORS 审中-公开CRAC通道吡唑和TRIAZOLCARBONSÄUREAMIDE作为抑制剂
公开(公告)号：EP2421834A1
公开(公告)日：2012-02-29
申请号：EP10714306.7
申请日：2010-04-22
申请人： Glaxo Group Limited
发明人： COE, Diane, Mary , COOPER, Anthony, William, James , GORE, Paul, Martin , HOUSE, David , SENGER, Stefan , VILE, Sadie
IPC分类号： C07D231/14 , C07D249/04 , A61K31/415 , A61K31/4192 , A61P11/06
CPC分类号： C07D231/14 , C07D249/04
摘要： The present invention relates to amide compounds of formula (I) processes for their preparation, intermediates usable in these processes, pharmaceutical compositions containing these compounds and to their use in therapy.
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公开(公告)号：EP2185542A2
公开(公告)日：2010-05-19
申请号：EP08787173.7
申请日：2008-08-13
申请人： Glaxo Group Limited
发明人： GORE, Paul, Martin , HANCOCK, Ashley, Paul , HODGSON, Simon, Teanby , PROCOPIOU, Panayiotis, Alexandrou , VILE, Sadie
IPC分类号： C07D401/12 , C07D215/233 , A61K31/4709
CPC分类号： C07D409/14 , C07D401/12
摘要： The present invention relates to compounds of formula (I), and salts thereof, processes for their preparation, to compositions containing them and to their use in the treatment of various diseases, such as allergic rhinitis.
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公开(公告)号：EP2091538B1
公开(公告)日：2010-03-03
申请号：EP07857765.7
申请日：2007-12-18
申请人： Glaxo Group Limited
IPC分类号： A61K31/502
CPC分类号： C07D471/04 , C07D237/32
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6.发明公开PHTHALAZINE AND PYRIDO Ý3,4-D¨PYRIDAZ INE COMPOUNDS AS H1 RECEPTOR ANTAGONISTS 有权酞嗪和吡啶并[3,4-D]哒嗪AS H1受体拮抗剂的
公开(公告)号：EP2215082A1
公开(公告)日：2010-08-11
申请号：EP08805231.1
申请日：2008-10-10
申请人： Glaxo Group Limited
IPC分类号： C07D403/06 , C07D471/04 , A61K31/502 , A61K31/5025 , A61P29/00 , A61P37/08
CPC分类号： C07D403/06 , C07D471/04
摘要： The present invention relates to compounds of formula (I), and salts thereof, processes for their preparation, to compositions containing them and to their use in the treatment of various diseases, such as allergic rhinitis.
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公开(公告)号：EP2091538A2
公开(公告)日：2009-08-26
申请号：EP07857765.7
申请日：2007-12-18
申请人： Glaxo Group Limited
IPC分类号： A61K31/502
CPC分类号： C07D471/04 , C07D237/32
摘要： The present invention relates to compounds of formula (I) and salts thereof, processes for their preparation, to compositions containing them and to their use in the treatment of various diseases, such as allergic rhinitis.
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公开(公告)号：EP2421835A1
公开(公告)日：2012-02-29
申请号：EP10714307.5
申请日：2010-04-22
申请人： Glaxo Group Limited
发明人： ALLEN, David, George , COE, Diane, Mary , COOPER, Anthony, William, James , GORE, Paul, Martin , HOUSE, David , SENGER, Stefan , SOLLIS, Steven, Leslie , VILE, Sadie , WILSON, Caroline
IPC分类号： C07D231/40 , A61K31/415 , A61P11/06
CPC分类号： C07D231/40
摘要： The present invention relates to amide compounds, processes for their preparation, pharmaceutical compositions containing these compounds and to their use in the treatment of disorders, conditions or disorders such as allergic disorders, inflammatory disorders and disorders of the immune system.
摘要翻译： 本发明涉及酰胺化合物，其制备方法，含有这些化合物的药物组合物及其在治疗诸如变态反应性疾病，炎性疾病和免疫系统疾病的病症，病症或病症中的用途。
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9.发明公开
公开(公告)号：EP2205585A1
公开(公告)日：2010-07-14
申请号：EP08805283.2
申请日：2008-10-15
申请人： Glaxo Group Limited
发明人： GORE, Paul Martin , HANCOCK, Ashley Paul , HODGSON, Simon Teanby , KRANZ, Michael Joachim , PROCOPIOU, Panayiotis Alexandrou , VILE, Sadie
IPC分类号： C07D401/12 , C07D401/14 , C07D413/14 , A61K31/4709 , A61P11/00 , A61P29/00 , A61P37/00
CPC分类号： C07D401/12 , C07D401/14 , C07D413/14
摘要： The present invention relates to compounds of formula (I) and salts thereof, processes for their preparation, to compositions containing them and to their use in the treatment of various diseases, such as allergic rhinitis.
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