专利检索 ap:("GlaxoSmithKline istrazivacki centar Zagreb d.o.o.") AND inv:"BUKVIC KRAJACIC, Mirjana" 第 1 页

1.

发明公开
9A-CARBAMOYL-Y-AMINOPROPYL- AND 9A-THIOCARBAMOYL-Y-AMINOPROPYL-AZALIDES WITH ANTIMALARIAL ACTIVITY 有权
标题翻译： 9A-羧乙基-Y-氨基丙烯酰胺-9-氨基]亚氨基-γ-氨基丙酸 - 马来酸盐麻醉剂抗菌药物

公开(公告)号：EP1855696A2

公开(公告)日：2007-11-21

申请号：EP06727593.3

申请日：2006-01-13

申请人： GlaxoSmithKline istrazivacki centar Zagreb d.o.o.

发明人： BUKVIC KRAJACIC, Mirjana , KUJUNDZIC, Nedjeljko , IVEZIC, Zrinka , ALIHODZIC, Sulejman , HUTINEC, Antun , FAJDETIC, Andrea

IPC分类号： A61K31/7052 , A61P33/06 , C07H17/08

CPC分类号： A61K31/7052 , C07H17/08 , Y02A50/411

摘要： Novel 9a-N'-substituted-carbamoyl- and thiocarbamoyl-aminoalkyl-9a-aza-9-deoxo-9-dihydro-9a-homoerythromycin A and 3-O-decladinosyl-9a-aza-9-deoxo-9-dihydro-9a-homoerythromycin A compounds having antimalarial activity are claimed. More particularly, the invention relates to 9a-N'-substituted-carbamoyl- and thiocarbamoyl-beta-aminoethyl- or -gamma-aminopropyl-9a-aza-9-deoxo-9-dihydro-9a-homoerythromycin A and 3-O-decladinosyl-9a-aza-9-deoxo-9-dihydro-9a-homoerythromycin A compounds and to pharmaceutically acceptable derivatives thereof having antimalarial activity.

2.

发明授权
9A-CARBAMOYL-Y-AMINOPROPYL- AND 9A-THIOCARBAMOYL-Y-AMINOPROPYL-AZALIDES WITH ANTIMALARIAL ACTIVITY 有权
标题翻译： 9A氨基甲酰-Y-氨丙基和9A-硫代-Y-丙基 - 氮杂内酯抗疟疾活动

公开(公告)号：EP1855696B1

公开(公告)日：2010-04-28

申请号：EP06727593.3

申请日：2006-01-13

申请人： GlaxoSmithKline istrazivacki centar Zagreb d.o.o.

发明人： BUKVIC KRAJACIC, Mirjana , KUJUNDZIC, Nedjeljko , IVEZIC, Zrinka , ALIHODZIC, Sulejman , HUTINEC, Antun , FAJDETIC, Andrea

IPC分类号： A61K31/7052 , A61P33/06 , C07H17/08

CPC分类号： A61K31/7052 , C07H17/08 , Y02A50/411

摘要： Novel 9a-N'-substituted-carbamoyl- and thiocarbamoyl-aminoalkyl-9a-aza-9-deoxo-9-dihydro-9a-homoerythromycin A and 3-O-decladinosyl-9a-aza-9-deoxo-9-dihydro-9a-homoerythromycin A compounds having antimalarial activity are claimed. More particularly, the invention relates to 9a-N'-substituted-carbamoyl- and thiocarbamoyl-beta-aminoethyl- or -gamma-aminopropyl-9a-aza-9-deoxo-9-dihydro-9a-homoerythromycin A and 3-O-decladinosyl-9a-aza-9-deoxo-9-dihydro-9a-homoerythromycin A compounds and to pharmaceutically acceptable derivatives thereof having antimalarial activity.