专利检索 ap:("MERCK PATENT GmbH") AND inv:"COLLONGES, Francois" 第 1 页

1.

发明公开
AROYL-O-PIPERIDINE DERIVATIVES FOR THE TREATMENT OF DIABETES-RELATED PROBLEMS 有权
标题翻译：芳-O-哌啶相关的问题与治疗糖尿病

公开(公告)号：EP1753721A1

公开(公告)日：2007-02-21

申请号：EP05742232.1

申请日：2005-05-19

申请人： Merck Patent GmbH

发明人： GUEDAT, Philippe , COLLONGES, Francois , CHEVREUIL, Olivier , DUMAS, Hervé , DENAULT, Marie Noelle , YVON, Stéphane , KANE, Peter , LAINTON, Julia , ROBERTSON, Avril , WENDT, Bernd

IPC分类号： C07D211/46 , C07D401/12 , C07D413/12 , C07D405/12 , C07D409/12 , C07D405/06 , C07D401/06 , C07D211/96 , C07D413/06 , A61K31/435 , A61P3/00

CPC分类号： C07D211/46 , C07D211/96 , C07D213/12 , C07D401/06 , C07D401/12 , C07D405/06 , C07D405/12 , C07D409/06 , C07D409/12 , C07D413/06 , C07D413/12

摘要： The present invention relates to derivatives of aroyl-O-piperidine structure of the general formula (I): in which R1, R2, R3 and R4 are as defined in the description. Application of the compounds of the formula (I) to the treatment of hyper-triglyceridaemia, hypercholesterolaemia and dyslipidaemia, and to the prevention or treatment of obesity.

2.

发明公开
N-BENZODIOXOLYL, N-BENZODIOXANYL AND N-BENZODIOXEPINYL ARYLCARBONXAMIDE DERIVATIVES, AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM 审中-公开
标题翻译： N-二苯并二，N-苯并二和正BENZODIOXEPINYLARYLCARBONSÄUREAMIDDERIVATE和含有药物组合物

公开(公告)号：EP1554263A1

公开(公告)日：2005-07-20

申请号：EP03809266.4

申请日：2003-10-01

申请人： MERCK PATENT GmbH

发明人： DUMAS, Hervé , BARBANTON, Jacques , COLLONGES, Francois , DECERPRIT, Jacques , ORTHOLAND, Jean-Yves , BENZIES, David, W., M. , CAMERON, Stuart , FOSTER, Richard, J. , GUESSREGEN, Stefan, M. , KANE, Peter , LAINTON, Julia, A., H. , ROBERTSON, Avril, A., B. , WENDT, Bernd , WARNE, Mark, R.

IPC分类号： C07D317/46 , C07D319/20 , C07D319/18 , C07D321/10 , C07D405/12 , C07F7/18 , C07C65/24 , C07C65/34 , C07C271/12 , A61K31/357 , A61K31/36 , A61P3/10

CPC分类号： C07D405/12 , C07C65/24 , C07C65/34 , C07C69/007 , C07C69/616 , C07C271/12 , C07D317/46 , C07D319/18 , C07D319/20 , C07D321/10 , C07F7/1856

摘要： The present invention relates to a compound of the formula (I) : in which T, A, R, B Xi, Yi and n are as defined in Claim 1, and to the pharmaceutically usable derivatives, solvates and stereoisomers thereof, comprising a mixture thereof in all proportions, which can be used in the treatment of dyslipidaemia, and to pharmaceutical compositions comprising them.