PYRIDAZINE DERIVATIVES
    6.
    发明公开
    PYRIDAZINE DERIVATIVES 审中-公开
    哒嗪衍生物

    公开(公告)号:EP2077997A1

    公开(公告)日:2009-07-15

    申请号:EP07819250.7

    申请日:2007-10-23

    摘要: The present invention relates to novel pyridazine derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: wherein R1 is hydrogen, C1-C6alkyl, C1-C8haloalkyl or C3-C6cycloalkyl; R2 is cycloalkyl, cycloalkylalkyl, halocycloalkyl, cycloalkoxy, halocycloalkoxy, cycloalkylalkoxy, halocycloalkylalkoxy, alkoxyalkyl, cycloalkoxyalkoxyalkyl, haloalkoxyalkyl, trialkylsilyl, alkylthioalkyl, haloalkylthioalkyl, cycloalkylthio, halocycloalkylthio, cycloalkylalkylthio, halocycloalkylalkylthio, alkylsulfinylalkyl, alkylsulfonylalkyl, alkylsulfinyl, haloalkylsulfinyl, alkylsulfonyl, haloalkylsulfonyl, C2-C6alkenyl, C2-C6alkynyl, optionally substituted arylsulfonyl, optionally substituted aryloxy, optionally substituted heteroaryloxy, optionally substituted arylthio, optionally substituted heteroarylthio; or R2 together with an adjacent carbon atom forms an optionally substituted fused ring; R3 is an optionally substituted aryl; R4 is hydrogen, halogen, C1-C6alkyl, C1-C6haloalkyl, C1-C8alkoxy, C1-C6haloalkoxy, hydroxy or cyano; and n is a whole number from 1 to 4; or an agrochemically usable salt form thereof.

    摘要翻译: 本发明涉及式(I),其具有杀微生物活性作为活性成分,特别是杀真菌活性的新颖的哒嗪衍生物:其中R1是氢,C1-C6烷基,C1-C8卤代烷基或C 3 -C 6环烷基; R 2是环烷基,环烷基烷基,卤代环烷基,环烷氧基,卤代环烷氧基,环烷基烷氧基,halocycloalkylalkoxy,烷氧基烷基,cycloalkoxyalkoxyalkyl,卤代烷氧基烷基,三烷基甲硅烷,烷硫基烷基,haloalkylthioalkyl,环烷硫基,halocycloalkylthio,cycloalkylalkylthio,halocycloalkylalkylthio,alkylsulfinylalkyl,烷基磺酰基烷基,烷基亚磺酰基,卤代烷,烷基磺酰基,卤代烷基磺酰基,C2- 任选取代的芳基磺酰基,任选取代的芳基氧基,任选取代的杂芳基氧基,任选取代的芳基硫基,任选取代的杂芳基硫基; 或R2与相邻碳原子一起形成任选取代的稠合环; R3是任选取代的芳基; R 4是氢,卤素,C 1 -C 6烷基,C 1 -C 6卤代烷基,C 1 -C 8烷氧基,C 1 -C 6卤代烷氧基,羟基或氰基; n是从1到4的整数; 或其农业化学可用的盐形式。

    EP0539588A4 -
    9.
    发明公开
    EP0539588A4 - 失效
    EP0539588A4 - Google专利

    公开(公告)号:EP0539588A4

    公开(公告)日:1995-03-15

    申请号:EP91912066

    申请日:1991-07-02

    摘要: A compound represented by general formula (I), its salt, production thereof, and insecticide containing the same wherein R1 represents a 5- or 6-membered nitrogenous aromatic heterocyclic group which may be substituted; X represents alkylene or alkylidene; R2 represents hydrogen, optionally substituted alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, aryl or -Y-R3; Y represents O, S(O)l, CO or CO2; l represents 0, 1 or 2; R3 represents hydrogen, optionally substituted alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl or aryl; A, B and D represent each independently an optionally substituted carbon atom or hetero-atom or a single bond; E represents CO or CS; Q represents hydrogen, optionally substituted alkyl, alkenyl, alkynyl, aryl, nitro, halogen or Z-R4; Z represents CO, CO2 or S(O)m; m represents 0, 1 or 2; and R4 represents optionally substituted alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl or aryl.

    摘要翻译: 通式(I)所示的化合物,其盐,其制造方法以及含有该化合物的杀虫剂,其中,R 1表示可以被取代的5或6元的含氮芳香族杂环基, X代表亚烷基或亚烷基; R2代表氢,任选取代的烷基,烯基,炔基,环烷基,环烯基,芳基或-YR3; Y代表O,S(O)l,CO或CO 2; l代表0,1或2; R 3代表氢,任选取代的烷基,烯基,炔基,环烷基,环烯基或芳基; A,B和D各自独立地表示任选取代的碳原子或杂原子或单键; E代表CO或CS; Q代表氢,任选取代的烷基,烯基,炔基,芳基,硝基,卤素或Z-R4; Z代表CO,CO2或S(O)m; m表示0,1或2; 且R4代表任选取代的烷基,烯基,炔基,环烷基,环烯基或芳基。