Abstract:
PROBLEM TO BE SOLVED: To provide a microbicide expressing excellent control effects in controlling plant diseases, particularly against rice blast, and giving no damage or very little damage to useful plant crops. SOLUTION: The microbicide contains an isoxazole carboxylic acid derivative expressed by general formula (1) as an active ingredient [wherein R 1 and R 2 each independently represents a hydrogen atom, a halogen atom or the like, and at least one of R 1 and R 2 represents a bromine atom; A represents OR 3 , SR 4 , NR 5 R 6 or NR 7 NR 8 R 9 . R 3 and R 4 each represents an 8-12C alkyl group or the like; R 5 represents a hydrogen atom or the like; R 6 represents a 2-pyridyl group or the like which may be substituted; R 7 , R 8 and R 9 each independently represents a 1-12C alkyl group or the like]. COPYRIGHT: (C)2009,JPO&INPIT
Abstract translation:要解决的问题:提供在控制植物病害,特别是防稻瘟病方面表现出优异的防治效果的杀微生物剂,并且对有用的植物作物没有损害或非常小的损害。 解决方案:杀微生物剂含有由通式(1)表示的异恶唑羧酸衍生物作为活性成分[其中R SP 1和R SP 2各自独立地表示氢 原子,卤素原子等,R SP 1和R SP 2中的至少一个表示溴原子; A表示OR 3 SP>,SR 4 SP>,NR 5 SP> R 6 SP>或NR NR 8 SP> R 9 SP>。 R 3 SP>和R 4 SP>各自表示8-12C烷基等; R 5表示氢原子等; R 6表示可以被取代的2-吡啶基等; R 7 SP>,R 8 SP>和R 9 SP>各自独立地表示1-12C烷基等〕。 版权所有(C)2009,JPO&INPIT
Abstract:
PROBLEM TO BE SOLVED: To provide a fungicide exhibiting excellent control effects on Pyricularia oryzae without damaging useful crops at all. SOLUTION: The fungicide comprises a diamine derivative represented by formula (1) [wherein, R1 is a 1-6C alkyl group or the like; R2 and R7 represent each independently a hydrogen atom, a 1-6C alkyl group or the like; R3 and R4 represent each independently a hydrogen atom, a 1-6C alkyl group or the like (except when both R3 and R4 are hydrogen atoms) or a 3-6C cycloalkyl group containing bound carbon atoms; R5 and R6 represent each independently a hydrogen atom, a 1-6C alkyl group or the like; R8 represents an aryl group or the like which may be substituted; one of X1, X2 and X3 represents a sulfur atom; and all the other represent each an oxygen atom]. A method for producing the diamine derivative is provided and the fungicide comprises the compound as an active ingredient. COPYRIGHT: (C)2008,JPO&INPIT
Abstract:
PROBLEM TO BE SOLVED: To provide a bactericide exhibiting an excellent controlling action on plant diseases, particularly on a blast disease of rice. SOLUTION: The bactericide includes a pyrazole derivative represented by formula (1) as an effective component [in the formula, R 1 and R 2 each represents hydrogen, halogen, 1-6C alkyl, 1-6C haloalkyl or the like (provided that at least one of R 1 and R 2 is 1-6C haloalkyl); R 3 represents 1-6C alkyl or the like; R 4 and R 5 each represents hydrogen, halogen, 1-6C alkyl or the like; A represents -OR 6 , -S(O) n R 7 , -NR 8 R 9 , -NR 10 NR 11 R 12 , -NR 13 OR 14 or -ONR 15 R 16 ; n represents 0 to 2; and R 6 to R 16 each represents hydrogen, alkyl or the like]. COPYRIGHT: (C)2010,JPO&INPIT
Abstract:
PROBLEM TO BE SOLVED: To provide a novel bactericide which exhibits a broad pest control spectrum against pathogenic bacteria of various crops and solves an urgent problem of resistant bacteria. SOLUTION: The diamine derivative is represented by formula (1) (wherein R1, R2, R5, and R10 are each hydrogen or a substituent such as a 1-6C alkyl group; R3, R4, R6, R7, R8, and R9 are each hydrogen or a substituent such as a 1-6C alkyl group or they are linked with one another to form a carbon-containing 3-6C cycloalkyl group; and Q is an aryl group or a heterocycle), and its manufacturing method is also disclosed, and the bactericide comprises this compound as an active ingredient. COPYRIGHT: (C)2007,JPO&INPIT
Abstract:
PROBLEM TO BE SOLVED: To provide a novel fungicide that exhibits a wide disease control spectrum against pathogenic fungi acting on various crops and helps resolve worsening drug-resistant strain problems. SOLUTION: The diamine derivatives of the formula (1), a process for producing the same, and fungicides containing the derivatives as an active ingredient are provided. [wherein R1 is a substituent such as C 1-6 alkyl; each of R2 and R5 independently is a hydrogen atom or a substituent such as C 1-6 alkyl; each of R3 and R4 independently is a hydrogen atom or a substituent such as C 1-6 alkyl, or is a C 3-6 cycloalkyl containing carbon atoms mutually bonding therebetween; each of R6, R7, R8 and R9 independently is a hydrogen atom or a substituent such as C 1-6 alkyl; R10 is a hydrogen atom or a substituent such as C 1-6 alkyl; A is an oxygen atom or sulfur atom; and Q is an aryl or heterocycle]. COPYRIGHT: (C)2006,JPO&NCIPI
Abstract translation:要解决的问题:提供一种新的杀真菌剂,其对作用于各种作物的致病真菌具有广泛的疾病控制谱,并有助于解决恶化的耐药菌株问题。 解决方案:提供式(1)的二胺衍生物,其制备方法和含有衍生物作为活性成分的杀真菌剂。 [其中R 1是诸如C 1-6烷基的取代基; R 2和R 5各自独立地为氢原子或C 1-6烷基等取代基; R 3和R 4各自独立地是氢原子或C 1-6烷基的取代基,或者是在其间相互结合的含有碳原子的C 3-6环烷基; R6,R7,R8和R9各自独立地为氢原子或C 1-6烷基等取代基; R 10为氢原子或C 1-6烷基等取代基; A是氧原子或硫原子; 并且Q是芳基或杂环]。 版权所有(C)2006,JPO&NCIPI
Abstract:
PROBLEM TO BE SOLVED: To provide a new germicide which shows a wide pathogen control spectrum against pathogens of agricultural products and solves the problem of drug-resistant strains. SOLUTION: A diamine derivative of formula (1) [wherein R1 is a 1-6C alkyl group or the like; R2, R5 and R10 are each independently a hydrogen atom, a 1-6C alkyl group or the like; R3 and R4, R6 and R7, and R8 and R9 are each independently a hydrogen atom, a 1-6C alkyl group or the like or may be bound to each other to form a 3-6C hydrocarbon ring; A1-A3 are each an oxygen atom or a sulfur atom, provided that at least A2 or A3 is a sulfur atom; and Q is an aryl group or a hetero ring], its preparation method and the germicide containing the compound as an active ingredient are provided. COPYRIGHT: (C)2006,JPO&NCIPI
Abstract:
PROBLEM TO BE SOLVED: To provide an isoxazole derivative having high plant disease-controlling activity, especially high disease-controlling activity on rice blast, while entirely harmless to useful crops or almost harmless. SOLUTION: The isoxazole derivative is represented by general formula (1) (wherein, R 1 , R 2 and R 3 are each independently H or the like; A is -OR 4 , -NR 6 R 7 or the like; wherein R 4 is 1-12C alkyl, aryl-substituted 1-6C alkyl, arylaminocarbonyl or the like, and R 6 and R 7 are each independently H, 2-6C alkenyl, aryl-substituted 1-6C alkyl, aryl, arylcarbonyl or the like, provided that R 6 and R 7 are not H at the same time). COPYRIGHT: (C)2010,JPO&INPIT
Abstract:
PROBLEM TO BE SOLVED: To provide a thiophene carboxylic acid derivative that exhibits excellent plant disease-controlling actions, particularly excellent controlling effects on rice blast disease while causing no injury or very little injury to useful crops. SOLUTION: The thiophene carboxylic acid derivative is represented by general formula (1) [wherein R 1 and R 2 are each a hydrogen atom, a 1-6C haloalkyl group or the like (provided that at least one of R 1 and R 2 is a 1-6C haloalkyl group); R 3 is a hydrogen atom or the like; A is OR 4 , SR 5 , NR 6 R 7 or NR 8 NR 9 R 10 ; R 4 is an 8-12C alkyl group or the like; R 5 is a 1-12C alkyl group or the like; R 6 and R 7 are each a hydrogen atom, an 8-12C alkyl group or the like; and R 8 , R 9 and R 10 are each a hydrogen atom, a 1-12C alkyl group or the like]. COPYRIGHT: (C)2009,JPO&INPIT
Abstract translation:待解决的问题:提供一种显示优异的植物病害控制作用的噻吩羧酸衍生物,特别是对稻瘟病病害的防治效果特别优异,同时对有用作物没有损伤或很少的损伤。 解决方案:噻吩羧酸衍生物由通式(1)表示[其中R 1 SP>和R 2 SP 2各自为氢原子,1-6C卤代烷基 基团等(条件是R 1 SP>和R 2 SP>中的至少一个为1-6C卤代烷基); R 3是氢原子等; A是OR 4 SP>,SR 5 SP>,NR 6 SP> R 7 SP>或NR 8 SP> NR 9 SP> R 10 SP>; R SP 4是8-12个C烷基等; R SP 5是1-12C烷基等; R 6和R 7各自为氢原子,8-12个C烷基等; 和R“SP”8,R“SP”9“,”R“SP 10”均为氢原子,1-12C烷基等]。 版权所有(C)2009,JPO&INPIT
Abstract:
PROBLEM TO BE SOLVED: To provide a compound and an insecticide comprising the same as the active ingredient exhibiting high insecticidal effect and a broad insecticidal spectrum on agricultural/horticultural insect pests but no harm to useful crops at all. SOLUTION: The insecticide comprises a carbazic acid derivative of formula(1)( wherein, R 1 is a 1-6C alkyl or the like; R 2 is a 1-6C alkyl or the like; Xn is 2, 6-Cl 2 -4-CF 3 or the like, and A is CH or the like ) as the active ingredient. COPYRIGHT: (C)2004,JPO
Abstract:
PROBLEM TO BE SOLVED: To provide intermediate aniline derivatives of insecticides having high effectiveness. SOLUTION: The aniline derivatives are represented by general formulae (8), (9). In the formula (8), R 7 is a 1-6C haloalkyl group; and Y 10 , Y 11 , Y 12 , Y 13 may be identical or different and each represents a hydrogen atom, a halogen atom, a 1-6C alkyl group or the like. In the formula (9), R 10 is a 1-6C haloalkyl group which may be substituted by at least one hydroxy group; and R 11 represents a hydrogen atom, a 1-4C alkyl group, a substituted m-nitrobenzoyl group or the like. COPYRIGHT: (C)2010,JPO&INPIT