Isoxazole carboxylic acid derivative and method for producing the same, and microbicide
    1.
    发明专利
    Isoxazole carboxylic acid derivative and method for producing the same, and microbicide 审中-公开
    异辛唑羧酸衍生物及其制备方法和微生物

    公开(公告)号:JP2009073818A

    公开(公告)日:2009-04-09

    申请号:JP2008209015

    申请日:2008-08-14

    Abstract: PROBLEM TO BE SOLVED: To provide a microbicide expressing excellent control effects in controlling plant diseases, particularly against rice blast, and giving no damage or very little damage to useful plant crops. SOLUTION: The microbicide contains an isoxazole carboxylic acid derivative expressed by general formula (1) as an active ingredient [wherein R 1 and R 2 each independently represents a hydrogen atom, a halogen atom or the like, and at least one of R 1 and R 2 represents a bromine atom; A represents OR 3 , SR 4 , NR 5 R 6 or NR 7 NR 8 R 9 . R 3 and R 4 each represents an 8-12C alkyl group or the like; R 5 represents a hydrogen atom or the like; R 6 represents a 2-pyridyl group or the like which may be substituted; R 7 , R 8 and R 9 each independently represents a 1-12C alkyl group or the like]. COPYRIGHT: (C)2009,JPO&INPIT

    Abstract translation: 要解决的问题:提供在控制植物病害,特别是防稻瘟病方面表现出优异的防治效果的杀微生物剂,并且对有用的植物作物没有损害或非常小的损害。 解决方案:杀微生物剂含有由通式(1)表示的异恶唑羧酸衍生物作为活性成分[其中R SP 1和R SP 2各自独立地表示氢 原子,卤素原子等,R SP 1和R SP 2中的至少一个表示溴原子; A表示OR 3 ,SR 4 ,NR 5 R 6 或NR NR 8 R 9 。 R 3 和R 4 各自表示8-12C烷基等; R 5表示氢原子等; R 6表示可以被取代的2-吡啶基等; R 7 ,R 8 和R 9 各自独立地表示1-12C烷基等〕。 版权所有(C)2009,JPO&INPIT

    Diamine derivative, method for producing the same and fungicide comprising the same as active ingredient
    2.
    发明专利
    Diamine derivative, method for producing the same and fungicide comprising the same as active ingredient 审中-公开
    DIAMINE衍生物,其生产方法及其包含其的活性成分的杀真菌剂

    公开(公告)号:JP2008037796A

    公开(公告)日:2008-02-21

    申请号:JP2006214199

    申请日:2006-08-07

    Abstract: PROBLEM TO BE SOLVED: To provide a fungicide exhibiting excellent control effects on Pyricularia oryzae without damaging useful crops at all. SOLUTION: The fungicide comprises a diamine derivative represented by formula (1) [wherein, R1 is a 1-6C alkyl group or the like; R2 and R7 represent each independently a hydrogen atom, a 1-6C alkyl group or the like; R3 and R4 represent each independently a hydrogen atom, a 1-6C alkyl group or the like (except when both R3 and R4 are hydrogen atoms) or a 3-6C cycloalkyl group containing bound carbon atoms; R5 and R6 represent each independently a hydrogen atom, a 1-6C alkyl group or the like; R8 represents an aryl group or the like which may be substituted; one of X1, X2 and X3 represents a sulfur atom; and all the other represent each an oxygen atom]. A method for producing the diamine derivative is provided and the fungicide comprises the compound as an active ingredient. COPYRIGHT: (C)2008,JPO&INPIT

    Abstract translation: 要解决的问题:提供一种对Pyricularia oryzae显示出优异的防治效果的杀真菌剂,而根本不破坏有用的作物。 解决方案:杀真菌剂包含由式(1)表示的二胺衍生物[其中,R1是1-6C烷基等; R2和R7各自独立地表示氢原子,1-6C烷基等; R3和R4各自独立地表示氢原子,1-6C烷基等(当R3和R4都是氢原子时除外)或含有结合碳原子的3-6C环烷基; R5和R6各自独立地表示氢原子,1-6C烷基等; R8表示可以被取代的芳基等; X 1,X 2和X 3中的一个表示硫原子; 而其他所有的都代表氧原子]。 提供二胺衍生物的制造方法,该杀真菌剂含有作为有效成分的化合物。 版权所有(C)2008,JPO&INPIT

    Pyrazole derivative, method of producing the same, and bactericide
    3.
    发明专利
    Pyrazole derivative, method of producing the same, and bactericide 审中-公开
    吡唑衍生物,其制备方法和杀菌剂

    公开(公告)号:JP2010083763A

    公开(公告)日:2010-04-15

    申请号:JP2008251019

    申请日:2008-09-29

    Abstract: PROBLEM TO BE SOLVED: To provide a bactericide exhibiting an excellent controlling action on plant diseases, particularly on a blast disease of rice. SOLUTION: The bactericide includes a pyrazole derivative represented by formula (1) as an effective component [in the formula, R 1 and R 2 each represents hydrogen, halogen, 1-6C alkyl, 1-6C haloalkyl or the like (provided that at least one of R 1 and R 2 is 1-6C haloalkyl); R 3 represents 1-6C alkyl or the like; R 4 and R 5 each represents hydrogen, halogen, 1-6C alkyl or the like; A represents -OR 6 , -S(O) n R 7 , -NR 8 R 9 , -NR 10 NR 11 R 12 , -NR 13 OR 14 or -ONR 15 R 16 ; n represents 0 to 2; and R 6 to R 16 each represents hydrogen, alkyl or the like]. COPYRIGHT: (C)2010,JPO&INPIT

    Abstract translation: 要解决的问题:提供对植物疾病,特别是稻瘟病病毒具有优异控制作用的杀菌剂。 解决方案:杀菌剂包括由式(1)表示的吡唑衍生物作为有效成分[在该式中,R 1 SP>和< SP> 2< SP> 2< SP>各自表示氢,卤素 ,1-6C烷基,1-6C卤代烷基等(条件是R 1和R 2中的至少一个为1-6个卤代烷基)。 R“3”表示1-6C烷基等; R 4和R 5各自表示氢,卤素,1-6C烷基等; A表示-OR,SP(S),-S(O),-S 9 ,-NR 10 14 或-ONR 15 R 16 ; n表示0〜2; R 16和R 16各自表示氢,烷基等。 版权所有(C)2010,JPO&INPIT

    Diamine derivative, its manufacturing method and bactericide having the same as active ingredient
    4.
    发明专利
    Diamine derivative, its manufacturing method and bactericide having the same as active ingredient 审中-公开
    DIAMINE DERIVATIVE,其制造方法和具有活性成分的杀菌剂

    公开(公告)号:JP2006298785A

    公开(公告)日:2006-11-02

    申请号:JP2005119275

    申请日:2005-04-18

    Abstract: PROBLEM TO BE SOLVED: To provide a novel bactericide which exhibits a broad pest control spectrum against pathogenic bacteria of various crops and solves an urgent problem of resistant bacteria. SOLUTION: The diamine derivative is represented by formula (1) (wherein R1, R2, R5, and R10 are each hydrogen or a substituent such as a 1-6C alkyl group; R3, R4, R6, R7, R8, and R9 are each hydrogen or a substituent such as a 1-6C alkyl group or they are linked with one another to form a carbon-containing 3-6C cycloalkyl group; and Q is an aryl group or a heterocycle), and its manufacturing method is also disclosed, and the bactericide comprises this compound as an active ingredient. COPYRIGHT: (C)2007,JPO&INPIT

    Abstract translation: 要解决的问题:提供一种对各种作物的病原菌具有广泛的害虫控制谱的新型杀菌剂,并解决了抗性细菌的紧迫问题。 解决方案:二胺衍生物由式(1)表示(其中R 1,R 2,R 5和R 10各自为氢或诸如1-6C烷基的取代基; R 3,R 4,R 6,R 7,R 8, 和R9各自为氢或诸如1-6C烷基的取代基或它们彼此连接形成含碳的3-6C环烷基; Q为芳基或杂环)及其制备方法 并且杀菌剂包含该化合物作为活性成分。 版权所有(C)2007,JPO&INPIT

    Diamine derivative, process for producing the same and fungicide containing the derivative as active ingredient
    5.
    发明专利
    Diamine derivative, process for producing the same and fungicide containing the derivative as active ingredient 有权
    DIAMINE DERIVATIVE,其生产方法和含有作为活性成分的衍生物的杀真菌剂

    公开(公告)号:JP2006232803A

    公开(公告)日:2006-09-07

    申请号:JP2005193403

    申请日:2005-07-01

    Abstract: PROBLEM TO BE SOLVED: To provide a novel fungicide that exhibits a wide disease control spectrum against pathogenic fungi acting on various crops and helps resolve worsening drug-resistant strain problems. SOLUTION: The diamine derivatives of the formula (1), a process for producing the same, and fungicides containing the derivatives as an active ingredient are provided. [wherein R1 is a substituent such as C 1-6 alkyl; each of R2 and R5 independently is a hydrogen atom or a substituent such as C 1-6 alkyl; each of R3 and R4 independently is a hydrogen atom or a substituent such as C 1-6 alkyl, or is a C 3-6 cycloalkyl containing carbon atoms mutually bonding therebetween; each of R6, R7, R8 and R9 independently is a hydrogen atom or a substituent such as C 1-6 alkyl; R10 is a hydrogen atom or a substituent such as C 1-6 alkyl; A is an oxygen atom or sulfur atom; and Q is an aryl or heterocycle]. COPYRIGHT: (C)2006,JPO&NCIPI

    Abstract translation: 要解决的问题:提供一种新的杀真菌剂,其对作用于各种作物的致病真菌具有广泛的疾病控制谱,并有助于解决恶化的耐药菌株问题。 解决方案:提供式(1)的二胺衍生物,其制备方法和含有衍生物作为活性成分的杀真菌剂。 [其中R 1是诸如C 1-6烷基的取代基; R 2和R 5各自独立地为氢原子或C 1-6烷基等取代基; R 3和R 4各自独立地是氢原子或C 1-6烷基的取代基,或者是在其间相互结合的含有碳原子的C 3-6环烷基; R6,R7,R8和R9各自独立地为氢原子或C 1-6烷基等取代基; R 10为氢原子或C 1-6烷基等取代基; A是氧原子或硫原子; 并且Q是芳基或杂环]。 版权所有(C)2006,JPO&NCIPI

    Isoxazole derivative and method for producing the same, and fungicide
    7.
    发明专利
    Isoxazole derivative and method for producing the same, and fungicide 审中-公开
    异辛唑衍生物及其制备方法和杀真菌剂

    公开(公告)号:JP2010077090A

    公开(公告)日:2010-04-08

    申请号:JP2008249222

    申请日:2008-09-26

    Abstract: PROBLEM TO BE SOLVED: To provide an isoxazole derivative having high plant disease-controlling activity, especially high disease-controlling activity on rice blast, while entirely harmless to useful crops or almost harmless. SOLUTION: The isoxazole derivative is represented by general formula (1) (wherein, R 1 , R 2 and R 3 are each independently H or the like; A is -OR 4 , -NR 6 R 7 or the like; wherein R 4 is 1-12C alkyl, aryl-substituted 1-6C alkyl, arylaminocarbonyl or the like, and R 6 and R 7 are each independently H, 2-6C alkenyl, aryl-substituted 1-6C alkyl, aryl, arylcarbonyl or the like, provided that R 6 and R 7 are not H at the same time). COPYRIGHT: (C)2010,JPO&INPIT

    Abstract translation: 要解决的问题:提供具有高植物病害控制活性的异恶唑衍生物,特别是对稻瘟病具有高度的防治疾病,同时对有用作物完全无害或几乎无害。 解决方案:异恶唑衍生物由通式(1)表示(其中,R 1,R 2,R 2,R 3和R 3各自为 独立地H等; A是-OR 4,或者其中R 4,R 4, SP>是1-12C烷基,芳基取代的1-6C烷基,芳基氨基羰基等,R 6和R 7各自独立地是H,2-6C烯基 ,芳基取代的1-6C烷基,芳基,芳基羰基等,条件是R 6和R 7不在同一时间。 版权所有(C)2010,JPO&INPIT

    Thiophene carboxylic acid derivative and its manufacturing method, and bactericide
    8.
    发明专利
    Thiophene carboxylic acid derivative and its manufacturing method, and bactericide 审中-公开
    硫酚羧酸衍生物及其制备方法和杀菌剂

    公开(公告)号:JP2009078991A

    公开(公告)日:2009-04-16

    申请号:JP2007247964

    申请日:2007-09-25

    Abstract: PROBLEM TO BE SOLVED: To provide a thiophene carboxylic acid derivative that exhibits excellent plant disease-controlling actions, particularly excellent controlling effects on rice blast disease while causing no injury or very little injury to useful crops. SOLUTION: The thiophene carboxylic acid derivative is represented by general formula (1) [wherein R 1 and R 2 are each a hydrogen atom, a 1-6C haloalkyl group or the like (provided that at least one of R 1 and R 2 is a 1-6C haloalkyl group); R 3 is a hydrogen atom or the like; A is OR 4 , SR 5 , NR 6 R 7 or NR 8 NR 9 R 10 ; R 4 is an 8-12C alkyl group or the like; R 5 is a 1-12C alkyl group or the like; R 6 and R 7 are each a hydrogen atom, an 8-12C alkyl group or the like; and R 8 , R 9 and R 10 are each a hydrogen atom, a 1-12C alkyl group or the like]. COPYRIGHT: (C)2009,JPO&INPIT

    Abstract translation: 待解决的问题:提供一种显示优异的植物病害控制作用的噻吩羧酸衍生物,特别是对稻瘟病病害的防治效果特别优异,同时对有用作物没有损伤或很少的损伤。 解决方案:噻吩羧酸衍生物由通式(1)表示[其中R 1 SP>和R 2 SP 2各自为氢原子,1-6C卤代烷基 基团等(条件是R 1 和R 2 中的至少一个为1-6C卤代烷基); R 3是氢原子等; A是OR 4 ,SR 5 ,NR 6 R 7 或NR 8 NR 9 R 10 ; R SP 4是8-12个C烷基等; R SP 5是1-12C烷基等; R 6和R 7各自为氢原子,8-12个C烷基等; 和R“SP”8,R“SP”9“,”R“SP 10”均为氢原子,1-12C烷基等]。 版权所有(C)2009,JPO&INPIT

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