Aminotetralins and use in inducing anesthesia
    92.
    发明授权
    Aminotetralins and use in inducing anesthesia 失效
    氨基丝氨酸和用于诱导麻醉

    公开(公告)号:US4101677A

    公开(公告)日:1978-07-18

    申请号:US806790

    申请日:1977-06-15

    CPC分类号: C07C2102/10 Y10S514/817

    摘要: Covers a compound selected from the group consisting of a member of the formula: ##STR1## wherein R.sub.1 is a radial selected from the group consisting of higher branched or straight chain alkyl and cycloalkyl radicals wherein said R.sub.1 radical contains at least six carbon atoms, R.sub.2 is a radical selected from the group consisting of hydrogen, loweralkyl and loweralkanol radicals, wherein said R.sub.2 radical contains 1 - 3 carbon atoms, and R.sub.3 is methoxy; and nontoxic pharmaceutically acceptable acid addition salts thereof. Also covers the use of said compound as a local anesthetic and pharmaceutical compositions comprising said above compounds as the active ingredient.

    摘要翻译: 包括选自下列成员组成的组的化合物:其中R1是选自由较高支链或直链烷基和环烷基组成的组的放射线,其中所述R 1基团含有至少6个碳原子,R 2 是选自氢,低级烷基和低级烷醇基团的基团,其中所述R 2基团含有1-3个碳原子,并且R 3是甲氧基; 和无毒的药学上可接受的酸加成盐。 还包括所述化合物作为局部麻醉剂的用途和包含所述上述化合物作为活性成分的药物组合物。