Semicarbazide derivatives, processes for preparation thereof and
pharmaceutical composition comprising the same
    91.
    发明授权
    Semicarbazide derivatives, processes for preparation thereof and pharmaceutical composition comprising the same 失效
    氨基脲衍生物,其制备方法和包含其的药物组合物

    公开(公告)号:US4725608A

    公开(公告)日:1988-02-16

    申请号:US673845

    申请日:1984-11-21

    摘要: New semicarbazide derivatives of the formula: ##STR1## wherein R.sup.1 is hydrogen,R.sup.2 is hydrogen, lower alkyl, ar(lower)alkyl, lower alkenyl or aryl,R.sup.3 is lower alkyl, ar(lower)alkyl, lower alkenyl or aryl, orR.sup.2 and R.sup.3 are taken together to form (C.sub.2 -C.sub.6)alkylidene group optionally substituted with aryl or taken together with the adjacent nitrogen atom to form a saturated or unsaturated, 5- or 6-membered heterocyclic group optionally substituted with aryl; orR.sup.1 and R.sup.2 are taken together with the adjacent nitrogen atoms to form a saturated or unsaturated, 5- or 6-membered heterocyclic group or 1,2-diazaspiroalkane-1,2-diyl group,R.sup.3 is hydrogen, lower alkyl, ar(lower)alkyl, lower alkenyl or aryl;R.sup.4 is aryl which may have substituent(s) selected from lower alkyl, halogen, lower alkoxy, lower alkylamino, halo(lower)alkyl, hydroxy, lower alkanoyl, esterified carboxy and carboxy,R.sup.5 is hydrogen or lower alkyl, andX is O or S, provided that the lower alkyl group for R.sup.3 is (C.sub.3 -C.sub.6)alkyl, when R.sup.2 is hydrogen or (C.sub.1 -C.sub.2) alkyl and R.sup.4 is aryl optionally having substituent(s) selected from groups consisting of halogen, lower alkyl, lower alkoxy and halo(lower)alkyl, and pharmaceutically acceptable salts thereof, and processes for preparation thereof and pharmaceutical composition comprising the same.These derivatives and salts thereof are useful as antiinflammatory and analgesic agents.

    摘要翻译: 新的下式的氨基脲衍生物:其中R1是氢,R2是氢,低级烷基,芳基(低级)烷基,低级烯基或芳基,R3是低级烷基,芳基(低级)烷基,低级烯基或芳基,或 R2和R3一起形成任选被芳基取代的(C 2 -C 6)亚烷基或与相邻的氮原子一起形成任选被芳基取代的饱和或不饱和的5或6元杂环基; 或者R1和R2与相邻的氮原子一起形成饱和或不饱和的5或6元杂环基或1,2-二氮杂环烷-1,2-二基,R3是氢,低级烷基,ar( 低级)烷基,低级烯基或芳基; R4是可以具有选自低级烷基,卤素,低级烷氧基,低级烷基氨基,卤代(低级)烷基,羟基,低级烷酰基,酯化羧基和羧基的取代基的芳基,R 5是氢或低级烷基,X是O 或者当R 2为氢或(C 1 -C 2)烷基,且R 4为任选具有选自以下的取代基的芳基时,R 3的低级烷基为(C 3 -C 6)烷基:(C 3 -C 6)烷基,低级烷基, 低级烷氧基和卤代(低级)烷基及其药学上可接受的盐,及其制备方法和包含其的药物组合物。 这些衍生物和其盐可用作抗炎和止痛剂。

    Fused polycyclic compound and organic light-emitting device using the compound
    96.
    发明授权
    Fused polycyclic compound and organic light-emitting device using the compound 有权
    熔融多环化合物和使用该化合物的有机发光装置

    公开(公告)号:US08288016B2

    公开(公告)日:2012-10-16

    申请号:US13056351

    申请日:2009-07-28

    摘要: Provided is an organic light-emitting device having good durability. The organic light-emitting device includes an anode, a cathode, and organic compound layers interposed between the anode and the cathode, and at least one of the organic compound layers contains a fused polycyclic compound represented by the following general formula [1]: wherein R1, R2, R3, R4, R5, R6, R7, R8, R9, R10, R11, R12, R13, R14, R15, R16, R17, and R18 each represent, independently of one another, a hydrogen atom, a halogen atom, an alkyl group having 1 to 20 carbon atoms, a substituted amino group, a substituted or unsubstituted aryl group, or a substituted or unsubstituted heterocyclic group, provided that at least one of R1 to R18 is a substituted phenyl group represented by the following general formula [2]:

    摘要翻译: 提供了具有良好耐久性的有机发光装置。 有机发光器件包括阳极,阴极和介于阳极和阴极之间的有机化合物层,并且至少一个有机化合物层含有由以下通式[1]表示的稠合多环化合物:其中 R1,R2,R3,R4,R5,R6,R7,R8,R9,R10,R11,R12,R13,R14,R15,R16,R17和R18各自独立地表示氢原子, 原子,碳原子数1〜20的烷基,取代氨基,取代或未取代的芳基或取代或未取代的杂环基,条件是R 1〜R 18中的至少一个为以下所示的取代苯基 通式[2]:

    PHOTO-CURABLE TRANSFER SHEET AND METHOD FOR FORMING CONCAVE-CONVEX PATTERN USING THE SAME
    99.
    发明申请
    PHOTO-CURABLE TRANSFER SHEET AND METHOD FOR FORMING CONCAVE-CONVEX PATTERN USING THE SAME 审中-公开
    用于形成使用其的凹凸图案的光固化转印片和方法

    公开(公告)号:US20120175822A1

    公开(公告)日:2012-07-12

    申请号:US13496329

    申请日:2010-09-16

    摘要: The present invention is to provide a photo-curable transfer sheet suitable for the preparation of an intermediate stamper in a nanoimprint method, in which the mold release properties from a mold having a fine concave-convex pattern used in the preparation of the intermediate stamper and the mold release properties of a cured photo-curable resin that is a product having a fine concave-convex pattern transferred from the intermediate stamper are excellent, and the transfer property of the fine concave-convex pattern is good; and a method for forming a concave-convex pattern by using the above-mentioned photo-curable transfer sheet. The photo-curable transfer sheet 10 having a photo-curable transfer layer 11 comprising a photo-curable composition deformable by application of pressure which comprises a polymer and a reactive diluent having a photopolymerizable functional group, wherein the polymer is an acrylic resin comprising a recurring unit derived from (meth)acrylate having an alicyclic group.

    摘要翻译: 本发明提供一种适用于纳米压印法制备中压模的光固化转印片,其中从具有用于制备中间压模的细凹凸图案的模具中脱模性能以及 作为从中间压模转印的具有微细凹凸图案的产品的固化光固化树脂的脱模性优异,并且精细凹凸图案的转印性良好; 以及通过使用上述光固化性转印片形成凹凸图案的方法。 具有光固化性转印层11的光固化性转印片11,其包含通过施加压力而变形的光固化性组合物,所述光固化性组合物包含聚合物和具有光聚合性官能团的反应性稀释剂,其中,所述聚合物为丙烯酸树脂, 衍生自具有脂环族基团的(甲基)丙烯酸酯的单元。