公开(公告)号：US20160304435A1

公开(公告)日：2016-10-20

申请号：US15103110

申请日：2014-12-08

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Johann SEEBA ,  Günter SCHLEGEL ,  Martin LITTMANN ,  Rafael WARSITZ ,  Mark James FORD

IPC: C07C209/08 ,  C07C209/84

CPC classification number: C07C209/08 ,  C07C209/04 ,  C07C209/14 ,  C07C209/84 ,  C07C211/29

Abstract: The present invention relates to a novel process for preparing halogenated di-substituted benzylamines, particularly halogenated dialkylbenzylamines.

Abstract translation: 本发明涉及制备卤代二取代苄胺，特别是卤代二烷基苄胺的新方法。

公开(公告)号：US20160289194A1

公开(公告)日：2016-10-06

申请号：US15037564

申请日：2014-11-25

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Sergii PAZENOK ,  Norbert LUI ,  Christian FUNKE ,  Arnd NEEFF ,  Vadim Mikhailovich TIMOSHENKO ,  Elena Ivanovna KAMINSKAYA ,  Yuriy Grigorievich SHERMOLOVICH

IPC: C07D231/16 ,  C07D403/04 ,  C07D231/14 ,  C07D231/38

CPC classification number: C07D231/16 ,  C07D231/14 ,  C07D231/38 ,  C07D403/04

Abstract: A new process for the preparation of 5-fluoro-1H-pyrazoles of the general formula (I) as described herein, resulting from the reaction of an olefin with hydrazine in the presence of water and a base.

Abstract translation: 一种制备如本文所述的通式（I）的5-氟-1H-吡唑的新方法，其由在烯烃和碱存在下烯烃与肼的反应得到。

公开(公告)号：US20160280668A1

公开(公告)日：2016-09-29

申请号：US15033928

申请日：2014-11-05

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Werner HALLENBACH ,  Ulrich GOERGENS ,  Andreas TURBERG ,  Kerstin ILG ,  Sebastian HORSTMANN ,  Johannes KOBBERLING

IPC: C07D249/06 ,  C07D409/12 ,  C07D401/04 ,  A01N43/647

CPC classification number: C07D249/06 ,  A01N43/647 ,  C07D401/04 ,  C07D409/12

Abstract: The invention relates inter alia to novel compounds of the general formula (I) in which the A1-A4, T, W, Q, R1 and B1-B4 radicals are each as defined in the description. Also described are processes for preparing the compounds of the formula (I). The inventive compounds are especially suitable for controlling insects, arachnids and nematodes in agriculture, and ectoparasites in veterinary medicine.

Abstract translation: 其中A1-A4，T，W，Q，R1和B1-B4基团各自如说明书中所定义。 还描述了制备式（I）化合物的方法。 本发明化合物特别适用于控制农业中的昆虫，蜘蛛和线虫，以及兽医学中的外寄生虫。

公开(公告)号：US20160280648A1

公开(公告)日：2016-09-29

申请号：US15033987

申请日：2014-11-11

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Wahed Ahmed MORADI ,  Thomas HIMMLER ,  Thomas Norbert MUELLER ,  Albert SCHNATTERER ,  Guenter SCHLEGEL

IPC: C07D213/56

CPC classification number: C07D213/56 ,  C07D213/38 ,  C07D213/57 ,  C07D213/89

Abstract: The present invention relates to a novel catalytic hydrogenation of substituted 2-methyl cyanopyridyl derivatives, in particular 3-chloro-5-(trifluorometyl)pyridin-2-yl]acetonitrile [=Py-CN] to substituted 2-ethylaminopyridine derivatives, in particular 2-[3-chloro-5-(trifluorometyl)pyridin-2-yl]ethanamine [=Py-ethanamine] or salts thereof in the presence of metal catalysts, in particular palladium catalysts.

Abstract translation: 本发明涉及取代的2-甲基氰基吡啶衍生物，特别是3-氯-5-（三氟甲基）吡啶-2-基]乙腈[= Py-CN]到取代的2-乙基氨基吡啶衍生物的催化氢化，特别是 2- [3-氯-5-（三氟甲基）吡啶-2-基]乙胺[= Py-乙胺]或其盐在金属催化剂，特别是钯催化剂存在下。

公开(公告)号：US20160255836A1

公开(公告)日：2016-09-08

申请号：US15029220

申请日：2014-10-15

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Philippe DESBORDES ,  Philippe RINOLFI ,  Tomoki TSUCHIYA ,  Julie GEIST ,  Lionel NICOLAS

IPC: A01N43/56 ,  C07D403/14 ,  C07D405/14 ,  C07D417/14 ,  A01N43/54 ,  A01N43/647 ,  A01N43/10 ,  A01N43/36 ,  C07D401/14 ,  C07D409/14 ,  A01N43/78

CPC classification number: A01N43/56 ,  A01N43/10 ,  A01N43/36 ,  A01N43/54 ,  A01N43/647 ,  A01N43/78 ,  C07D333/18 ,  C07D333/38 ,  C07D401/14 ,  C07D403/14 ,  C07D405/14 ,  C07D409/14 ,  C07D417/14

Abstract: The present invention relates to fungicidal N-cycloalkyl-N-(biheterocyclylmethylene)carboxamide derivatives and their thiocarbonyl derivatives, their process of preparation and intermediate compounds for their preparation, their use as fungicides, particularly in the form of fungicidal compositions and methods for the control of phytopathogenic fungi of plants using these compounds or their compositions.

Abstract translation: 本发明涉及杀真菌N-环烷基-N-（双杂环亚甲基）甲酰胺衍生物及其硫代羰基衍生物，其制备方法及其制备中间体化合物，其用作杀真菌剂，特别是杀真菌组合物和控制方法 使用这些化合物或其组合物的植物致病真菌。

公开(公告)号：US20160251344A1

公开(公告)日：2016-09-01

申请号：US15028923

申请日：2014-10-13

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Britta OLENIK ,  Stefan HILLEBRAND ,  Pierre WASNAIRE ,  Martin WEISS ,  Ulrike WACHENDORFF-NEUMANN

IPC: C07D417/14 ,  A01N43/80

CPC classification number: C07D417/14 ,  A01N43/80 ,  C07B2200/13

Abstract: The present invention relates to a novel crystalline form of 2-{3-[2-(1-{[3,5-bis(difluoromethyl)-1H-pyrazol-1-yl]acetyl}piperidin-4-yl)-1,3-thiazol-4-yl]-4,5-dihydro-1,2-oxazol-5-yl}-3-chlorophenylmethansulphonate, to processes for its preparation and to its use in agrochemical preparations.

Abstract translation: 本发明涉及2- {3- [2-（1 - {[3,5-双（二氟甲基）-1H-吡唑-1-基]乙酰基}哌啶-4-基）-1 ，3-噻唑-4-基] -4,5-二氢-1,2,5-恶唑-5-基} -3-氯苯甲磺酸盐，用于其制备及其在农用化学制剂中的应用。

公开(公告)号：US20160242419A1

公开(公告)日：2016-08-25

申请号：US15026143

申请日：2014-10-22

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： ARNIM KOEHN ,  CHRISTIAN WALDRAFF ,  ELMAR GATZWEILER ,  KLAUS TRABOLD ,  HUBERT MENNE ,  HARTMUT AHRENS ,  SIMON DOERNER-RIEPING ,  RALF BRAUN ,  INES HEINEMANN

IPC: A01N57/20 ,  A01N41/04 ,  A01N47/36 ,  A01N37/34 ,  A01N43/80 ,  A01N43/40 ,  A01N37/10 ,  A01N43/76 ,  A01N43/54 ,  A01N43/707 ,  A01N43/653 ,  A01N43/90 ,  A01N43/56 ,  A01N43/08 ,  A01N51/00 ,  A01N47/32 ,  A01N43/68 ,  A01N43/84 ,  A01N43/42 ,  A01N41/08 ,  A01N37/20 ,  A01N43/82

CPC classification number: A01N57/20 ,  A01N37/10 ,  A01N37/20 ,  A01N37/34 ,  A01N41/04 ,  A01N41/08 ,  A01N43/08 ,  A01N43/40 ,  A01N43/42 ,  A01N43/54 ,  A01N43/56 ,  A01N43/653 ,  A01N43/68 ,  A01N43/707 ,  A01N43/76 ,  A01N43/80 ,  A01N43/82 ,  A01N43/84 ,  A01N43/90 ,  A01N47/32 ,  A01N47/36 ,  A01N47/38 ,  A01N51/00 ,  A01N33/22 ,  A01N37/40 ,  A01N41/10 ,  A01N43/66 ,  A01N47/30

Abstract: What are described are herbicidal compositions comprising active ingredients from the group of the N-(1,3,4-oxadiazol-2-yl)arylcarboxamides and further herbicides and optionally safeners. These herbicidal compositions are particularly suitable for use against harmful plants in crops of useful plants.

Abstract translation: 所描述的是包含来自N-（1,3,4-恶二唑-2-基）芳基羧酰胺和其它除草剂和可选安全剂组的活性成分的除草组合物。 这些除草组合物特别适合用于有效植物作物中的有害植物。

公开(公告)号：US20160135461A1

公开(公告)日：2016-05-19

申请号：US14899709

申请日：2014-06-20

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Stefan HILLEBRAND ,  Matthias RIEDRICH ,  Sebastian HOFFMANN ,  Mark James FORD ,  Joachim TELSER ,  Mazen ES-SAYED ,  Guenter HOEMBERGER ,  Pierre WASNAIRE ,  Ulrike WACHENDORFF-NEUMANN ,  Tomoki TSUCHIYA

IPC: A01N43/80 ,  C07D417/14

CPC classification number: A01N43/80 ,  C07D417/14

Abstract: Piperidinecarboxylic acidderivatives of the formula (I) in which the symbols A, L1, L2, G, p, Q, R1, R2, T and Y are each as defined in the description, and salts, metal complexes and N-oxides of the compounds of the formula (I), and the use thereof for controlling phytopathogenic harmful fungi and processes for preparing compounds of the formula (I).

Abstract translation: 其中符号A，L1，L2，G，p，Q，R1，R2，T和Y各自如说明书中所定义的式（I）的哌啶羧酸衍生物，以及其盐，金属络合物和N-氧化物 式（I）化合物及其用于控制​​植物病原性有害真菌的用途及其制备式（I）化合物的方法。

公开(公告)号：US20160113277A1

公开(公告)日：2016-04-28

申请号：US14895343

申请日：2014-06-02

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Marc MOSRIN ,  Harald JAKOBI ,  Hansjoerg DIETRICH ,  Elmar GATZWEILER ,  Christopher ROSINGER ,  Dirk SCHMUTZLER

IPC: A01N37/36 ,  A01N37/34 ,  C07C255/37 ,  C07C255/36 ,  C07C253/30

CPC classification number: A01N37/36 ,  A01N37/34 ,  A01N53/00 ,  C07C253/30 ,  C07C255/36 ,  C07C255/37 ,  C07C255/53

Abstract: Primarily, the present invention relates to the use of substances of the formula (I) as herbicides, in particular for controlling broad-leaved weeds and/or weed grasses in crops of useful plants and/or as plant growth regulators for influencing the growth of crops of useful plants. The invention furthermore relates to the novel herbicidal substances of the formulae (Ib) and (Ia). The present invention also relates to corresponding compositions comprising one or more of the herbicides of the formula (I) and further agrochemically active substances, and also to plant growth-regulating or herbicidal compositions comprising one or more of these compounds. Moreover, the present invention relates to processes for preparing the compounds of the formula (I).

Abstract translation: 主要地，本发明涉及式（I）的物质作为除草剂的用途，特别是用于控制有用植物作物中的阔叶杂草和/或杂草，和/或作为影响生长的植物生长调节剂 作物的有用植物。 本发明还涉及式（Ib）和（Ia）的新颖除草物质。 本发明还涉及包含一种或多种式（I）的除草剂和其它农业化学活性物质的相应组合物，还涉及包含一种或多种这些化合物的植物生长调节剂或除草组合物。 此外，本发明涉及制备式（I）化合物的方法。

公开(公告)号：US20160075653A1

公开(公告)日：2016-03-17

申请号：US14787530

申请日：2014-04-28

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Anne DECOR ,  Joerg GREUL ,  Eike Kevin HEILMANN ,  Hans-Georg SCHWARZ ,  Ernst Rudolf GESING ,  Jens FRACKENPOHL ,  Hans-Ludwig ELBE ,  Welf Burkhard WIESE ,  Daniela PORTZ ,  Kerstin ILG ,  Olga MALSAM ,  Peter LOESEL ,  Peter LUEMMEN ,  Ulrich GOERGENS ,  Pierre-Yves COQUERON ,  Arianna MARTELLETTI ,  Philippe DESBORDES ,  Stephanie GARY ,  Isabelle CHRISTIAN ,  Claudia WELZ

IPC: C07D213/81 ,  C07D213/82 ,  C07C233/66 ,  C07D231/14

CPC classification number: C07D213/81 ,  A01N43/10 ,  A01N43/18 ,  A01N43/32 ,  A01N43/36 ,  A01N43/40 ,  A01N43/50 ,  A01N43/56 ,  A01N43/60 ,  A01N43/647 ,  A01N43/76 ,  A01N43/78 ,  A01N43/80 ,  C07C233/66 ,  C07C2601/02 ,  C07C2601/04 ,  C07D213/82 ,  C07D231/14

Abstract: The present invention relates to the use of N-(Phenylcycloalkyl)carboxamides and N-(Phenylcycloalkyl)thiocarboxamides for the control of nematodes in agriculture and as anthelmintic agents against endoparasites in animals and humans, compositions containing such compounds and methods for the control of nematodes and helminths and furthermore to novel N-(Phenylcycloalkyl)carboxamides and N-(Phenylcycloalkyl)thiocarboxamides, processes and intermediate compounds for their preparation, their use as nematicides, compositions containing such compounds and methods for the control of nematodes.

Abstract translation: 本发明涉及N-（苯基环烷基）甲酰胺和N-（苯基环烷基）硫代甲酰胺用于控制农业中的线虫和用作动物和人类内寄生虫的驱肠虫剂，含有这些化合物的组合物和控制线虫的方法 并且还涉及新的N-（苯基环烷基）甲酰胺和N-（苯基环烷基）硫代甲酰胺，其制备方法和中间体化合物，它们作为杀线虫剂的用途，含有这些化合物的组合物和用于控制线虫的方法。