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公开(公告)号:US20080081808A1
公开(公告)日:2008-04-03
申请号:US11855183
申请日:2007-09-14
申请人: Martha Sarpong , Nicholas Adams , Jeffrey Axten , Amita Chaudhari , Dashyant Dhanak , Toshihiro Hamajima , Kenneth Newlander , Cynthia Parrish , Jerry Adams , Domingos Silva , Jun Tang
发明人: Martha Sarpong , Nicholas Adams , Jeffrey Axten , Amita Chaudhari , Dashyant Dhanak , Toshihiro Hamajima , Kenneth Newlander , Cynthia Parrish , Jerry Adams , Domingos Silva , Jun Tang
IPC分类号: A61K31/437 , A61K31/4545 , A61K31/496 , A61K31/506 , A61K31/5377 , A61K31/54 , A61P35/00 , C07D471/04
CPC分类号: C07D471/04
摘要: The present invention relates to a compound represented by Formula (I): and pharmaceutically acceptable salts. Compounds of the present invention inhibit Aurora kinase, making them especially suitable for the treatment of a number of diseases, including solid tumor cancers and hematological cancers.
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公开(公告)号:US20070135432A1
公开(公告)日:2007-06-14
申请号:US11600683
申请日:2006-11-15
申请人: Han-Jie Zhou , David Morgans , Gustave Bergnes , Steven Knight , Kenneth Newlander , Dashyant Dhanak , Nicholas Adams
发明人: Han-Jie Zhou , David Morgans , Gustave Bergnes , Steven Knight , Kenneth Newlander , Dashyant Dhanak , Nicholas Adams
IPC分类号: C07D413/02 , C07D403/02 , A61K31/5377 , A61K31/513
CPC分类号: C07D239/36 , C07D231/12 , C07D233/56 , C07D239/47 , C07D239/91 , C07D249/08 , C07D403/06
摘要: Compounds useful for treating cellular proliferative diseases and disorders by modulating the activity of KSP are disclosed.
摘要翻译: 公开了通过调节KSP的活性来治疗细胞增殖性疾病和病症的化合物。
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公开(公告)号:US20060052360A1
公开(公告)日:2006-03-09
申请号:US10538228
申请日:2003-12-12
申请人: Gustave Bergnes , Dashyant Dhanak , Steven Knight , Pu Lu , David Morgans , Kenneth Newlander
发明人: Gustave Bergnes , Dashyant Dhanak , Steven Knight , Pu Lu , David Morgans , Kenneth Newlander
IPC分类号: A61K31/554 , A61K31/55 , A61K31/553 , C07D403/02 , C07D413/02 , C07D417/02
CPC分类号: C07D403/06
摘要: Compounds useful for treating cellular proliferative diseases and disorders by modulating the activity of KSP are disclosed.
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公开(公告)号:US20130053397A1
公开(公告)日:2013-02-28
申请号:US13696362
申请日:2011-05-05
申请人: James Brackley, III , Joelle Lorraine Burgess , Seth Grant , Neil Johnson , Steven D. Knight , Louis Lafrance , William H. Miller , Kenneth Newlander , Stuart Romeril , Meagan B. Rouse , Xinrong Tian , Sharad Kumar Verma
发明人: James Brackley, III , Joelle Lorraine Burgess , Seth Grant , Neil Johnson , Steven D. Knight , Louis Lafrance , William H. Miller , Kenneth Newlander , Stuart Romeril , Meagan B. Rouse , Xinrong Tian , Sharad Kumar Verma
IPC分类号: C07D401/14 , A61P35/00 , A61P35/02 , A61P37/06 , A61P37/00 , A61P31/10 , A61P19/02 , A61K31/496 , A61P1/00
CPC分类号: A61K31/496 , A61K31/405 , A61K31/4439 , A61K31/444 , A61K31/4545 , A61K31/501 , A61K31/506 , A61K31/5377 , A61K31/5383 , A61K31/541 , A61K31/551 , C07D401/12 , C07D401/14 , C07D405/14 , C07D409/14 , C07D417/14 , C07D471/04 , C07D487/04 , C07D487/08 , C07D498/04
摘要: Herein are disclosed indoles of formula (I) where the various groups are defined herein, and which are useful in treating cancer.
摘要翻译: 本文公开了式(I)的吲哚,其中各种基团在本文中定义,并且其可用于治疗癌症。
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公开(公告)号:US20070254870A1
公开(公告)日:2007-11-01
申请号:US11788784
申请日:2007-04-19
申请人: Gustave Bergnes , Dashyant Dhanak , Steven Knight , Pu Lu , David Morgans , Kenneth Newlander
发明人: Gustave Bergnes , Dashyant Dhanak , Steven Knight , Pu Lu , David Morgans , Kenneth Newlander
IPC分类号: A61K31/551 , C07D243/00 , C12N9/99
CPC分类号: C07D403/06
摘要: Compounds useful for treating cellular proliferative diseases and disorders by modulating the activity of KSP are disclosed.
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