公开(公告)号：US09512093B2

公开(公告)日：2016-12-06

申请号：US14899755

申请日：2014-06-17

Applicant: BASF SE

Inventor： Timo Frassetto ,  Maximilian Dochnahl ,  Michael Rack ,  Volker Maywald ,  Bernd Wolf ,  Roland Goetz ,  Philip Muelheims ,  Rudolf Haeberle

IPC: C07D265/36 ,  C07C17/16 ,  C07D413/04

CPC classification number: C07D265/36 ,  C07C17/16 ,  C07D413/04 ,  C07C21/22

Abstract: The present invention relates to a process for manufacturing 4-propargylated amino-benzoxazinones of formula (I), comprising the following steps: step a) preparing propargyl chloride by reacting propargyl alcohol with thionyl chloride optionally in the presence of a catalyst; and step b) reacting the propargyl chloride prepared in step (a) with a NH-benzoxazinone of formula (II); wherein the variables are defined according to the description.

公开(公告)号：US20150119572A1

公开(公告)日：2015-04-30

申请号：US14365822

申请日：2012-12-20

Applicant: BASF SE

Inventor： Maximilian Dochnahl ,  Michael Rack ,  Michael Keil ,  Bernd Wolf ,  Uwe Josef Vogelbacher ,  Joachim Gebhardt ,  Timo Frassetto ,  Volker Maywald

IPC: C07C231/24 ,  C07C235/34 ,  C07D207/16 ,  C07C231/12

CPC classification number: C07C231/24 ,  C07C231/12 ,  C07C235/20 ,  C07C235/34 ,  C07D207/06 ,  C07D207/16 ,  C07D211/16 ,  C07D295/185 ,  C07D413/04

Abstract: The present invention relates to a process for manufacturing aryloxyacetamides of formula (I), by reacting haloacetamides of formula (II) with a phenol of formula (III); wherein the variables are defined according to the description, and aryloxyacetamides of formula (I).

Abstract translation: 本发明涉及通过使式（II）的卤代乙酰胺与式（III）的苯酚反应制备式（I）的芳氧基乙酰胺的方法; 其中所述变量根据描述定义，和式（I）的芳氧基乙酰胺。

公开(公告)号：US20150099631A1

公开(公告)日：2015-04-09

申请号：US14402518

申请日：2013-05-15

Applicant: BASF SE

Inventor： Robert Reinhard ,  Tiziana Chiodo ,  Bernd Wolf ,  Stefan Scherer ,  Matthias Bratz ,  Matthias Witschel ,  Trevor William Newton ,  Thomas Seitz

IPC: C07D413/04 ,  A01N43/84

CPC classification number: C07D413/04 ,  A01N43/84 ,  C07B2200/13 ,  A01N25/12 ,  A01N2300/00

Abstract: The present invention relates to a novel crystalline form A of 1,5-dimethyl-6-thioxo-3-(2,2,7-trifluoro-3-oxo-4-(prop-2-ynyl)-3,4-dihydro-2H-benzo[b][1,4]oxazin-6-yl)-1,3,5-triazinane-2,4-dione. The invention also relates to a process for the production of this crystalline form and formulations for plant protection which contains the novel crystalline form of 1,5-dimethyl-6-thioxo-3-(2,2,7-trifluoro-3-oxo-4-(prop-2-ynyl)-3,4-dihydro-2H-benzo[b][1,4]oxazin-6-yl)-1,3,5-triazinane-2,4-dione.

Abstract translation: 本发明涉及1,5-二甲基-6-硫代-3-（2,2,7-三氟-3-氧代-4-（丙-2-炔基）-3,4-二氢 - -2,3-二氢-2H-苯并[b] [1,4]恶嗪-6-基）-1,3,5-三氮杂环戊烷-2,4-二酮。 本发明还涉及生产该结晶形式的方法和用于植物保护的制剂，其含有1,5-二甲基-6-硫代-3-（2,2,7-三氟-3-氧代 -4-（丙-2-炔基）-3,4-二氢-2H-苯并[b] [1,4]恶嗪-6-基）-1,3,5-三氮杂环戊烷-2,4-二酮。